- Anticancer kiteplatin pyrophosphate derivatives show unexpected targe…
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Anticancer kiteplatin pyrophosphate derivatives show unexpected target selectivity for DNA

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    SYSNO ASEP0486058
    Druh ASEPJ - Článek v odborném periodiku
    Zařazení RIVJ - Článek v odborném periodiku
    Poddruh JČlánek ve WOS
    NázevAnticancer kiteplatin pyrophosphate derivatives show unexpected target selectivity for DNA
    Tvůrce(i) Kašpárková, Jana (BFU-R) RID, ORCID
    Kostrhunová, Hana (BFU-R) RID, ORCID
    Novohradský, Vojtěch (BFU-R) ORCID
    Prachařová, J. (CZ)
    Curcio, A. (IT)
    Margiotta, N. (IT)
    Natile, G. (IT)
    Brabec, Viktor (BFU-R) RID, ORCID
    Celkový počet autorů8
    Zdroj.dok.Dalton Transactions. - : Royal Society of Chemistry - ISSN 1477-9226
    Roč. 46, č. 41 (2017), s. 14139-14148
    Poč.str.10 s.
    Forma vydáníTištěná - P
    Jazyk dok.eng - angličtina
    Země vyd.GB - Velká Británie
    Klíč. slovacancer-chemotherapy ; platinum complexes ; cross-links
    Vědní obor RIVCE - Biochemie
    Obor OECDBiochemistry and molecular biology
    CEPGA17-05302S GA ČR - Grantová agentura ČR
    Institucionální podporaBFU-R - RVO:68081707
    UT WOS000413638400011
    DOI https://doi.org/10.1039/c7dt02633a
    AnotaceOne of the promising new antitumor platinum complexes is a large-ring chelate complex [PtCl2(cis-1,4-DACH)] (DACH = diaminocyclohexane) (kiteplatin). Recently, new platinum(II) derivatives of kiteplatin with pyrophosphate as a carrier ligand have been synthesized and tested on a panel of human cancer cell lines. These derivatives of kiteplatin were found to be more effective than clinically used anticancer platinum drugs. The design of kiteplatin pyrophosphate derivatives was based on the concept of pyrophosphate coordinated platinum complexes, phosphaplatins. Phosphaplatins have been shown to function without binding to DNA and hence DNA has been excluded as the target of phosphaplatins in contrast to conventional antitumor platinum drugs. Cytotoxicity, major cellular targets and DNA interactions of the new anticancer platinum drug were characterized by standard biochemical methods and methods of molecular and cellular biology. We demonstrate that, in contrast to what has been reported on closely related phosphaplatins, the derivatives of kiteplatin with the pyrophosphate carrier ligand are activated in the cellular environment. This activation, which yields species capable of platination of DNA, very likely comprises the hydrolytic release of the pyrophosphate ligand that could be enzymatically catalyzed. Collectively, these data provide convincing evidence that unexpectedly DNA is an important target for the biological activity of the kiteplatin pyrophosphate derivatives, although the overall mechanism of action might be different from those of conventional platinum drugs.
    PracovištěBiofyzikální ústav
    KontaktJana Poláková, polakova@ibp.cz, Tel.: 541 517 244
    Rok sběru2018
Počet záznamů: 1  

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