Počet záznamů: 1
Hydroxyethylamine isostere of an HIV-1 protease inhibitor prefers its amine to the hydroxy group in binding to catalytic aspartates. A synchrotron study of HIV-1 protease in complex with a peptidomimetic inhibitor
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$a Hydroxyethylamine isostere of an HIV-1 protease inhibitor prefers its amine to the hydroxy group in binding to catalytic aspartates. A synchrotron study of HIV-1 protease in complex with a peptidomimetic inhibitor 215 $a 7 s. 463 -1
$1 001 cav_un_epca*0257026 $1 011 $a 0022-2623 $e 1520-4804 $1 200 1 $a Journal of Medicinal Chemistry $v Roč. 45, č. 7 (2002), s. 1432-1438 $1 210 $c American Chemical Society 610 1-
$a HIV-1 protease 610 1-
$a hydroxyethylamine-containing inhibitor 610 1-
$a aspartate 700 -1
$3 cav_un_auth*0103012 $a Dohnálek $b Jan $p UMCH-V $w Structure and dynamics of macromolecules $4 070 $T Ústav makromolekulární chemie AV ČR, v. v. i. 701 -1
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Počet záznamů: 1