Search results
- 1.0574151 - ÚACH 2024 RIV CH eng J - Journal Article
Oboňová, B. - Habala, L. - Litecká, Miroslava - Herich, P. - Bilková, A. - Bilka, F. - Horváth, B.
Antimicrobially Active Zn(II) Complexes of Reduced Schiff Bases Derived from Cyclohexane-1,2-diamine and Fluorinated Benzaldehydes—Synthesis, Crystal Structure and Bioactivity.
Life. Roč. 13, č. 7 (2023), č. článku 1516. E-ISSN 2075-1729
Institutional support: RVO:61388980
Keywords : antimicrobial activity * metal complexes * fluorinated compounds * medicinal chemistry * Schiff bases * zinc
OECD category: Inorganic and nuclear chemistry
Impact factor: 3.2, year: 2022
Method of publishing: Open access
Permanent Link: https://hdl.handle.net/11104/0344533File Download Size Commentary Version Access Antimicrobially.pdf 0 2.4 MB CC BY licence Publisher’s postprint open-access Antimicrobially SI.pdf 0 2.8 MB CC BY licence Publisher’s postprint open-access
Research data: MDPI - 2.0543050 - ÚOCHB 2022 RIV GB eng J - Journal Article
Kalčic, Filip - Dračínský, Martin - Janeba, Zlatko
Diverse synthetic approaches towards C1′-branched acyclic nucleoside phosphonates.
Organic & Biomolecular Chemistry. Roč. 19, č. 32 (2021), s. 6958-6963. ISSN 1477-0520. E-ISSN 1477-0539
R&D Projects: GA MŠMT LTAUSA18086
Institutional support: RVO:61388963
Keywords : tenofovir alafenamide * medicinal chemistry * nucleotide analogs
OECD category: Organic chemistry
Impact factor: 3.890, year: 2021
Method of publishing: Limited access
https://doi.org/10.1039/D1OB00751C
Permanent Link: http://hdl.handle.net/11104/0320358 - 3.0539170 - ÚMG 2021 RIV GB eng J - Journal Article
Kugler, Michael - Holub, J. - Brynda, Jiří - Pospíšilová, K. - El Anwar, S. - Bavol, D. - Havránek, M. - Král, Vlastimil - Fábry, Milan - Gruner, B. - Řezáčová, Pavlína
The structural basis for the selectivity of sulfonamido dicarbaboranes toward cancer-associated carbonic anhydrase IX.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 35, č. 1 (2020), s. 1800-1810. ISSN 1475-6366. E-ISSN 1475-6374
Institutional support: RVO:68378050
Keywords : tumor hypoxia * medicinal chemistry * drug discovery * binding-sites * inhibition * boron * pharmacophores * opportunities * conjugation * metastasis * Carbonic anhydrase IX * carborane * enzyme inhibitors * structure-activity relationship
OECD category: Biochemistry and molecular biology
Impact factor: 5.051, year: 2020
Method of publishing: Open access
https://www.tandfonline.com/doi/full/10.1080/14756366.2020.1816996
Permanent Link: http://hdl.handle.net/11104/0316870 - 4.0534661 - ÚACH 2021 RIV DE eng J - Journal Article
Nekvinda, Jan - Kugler, Michael - Holub, Josef - El Anwar, Suzan - Brynda, Jiří - Pospíšilová, K. - Růžičková, Z. - Řezáčová, Pavlína - Grüner, Bohumír
Direct Introduction of an Alkylsulfonamido Group on C-sites of Isomeric Dicarba-closo-dodecaboranes: The Influence of Stereochemistry on Inhibitory Activity against the Cancer-Associated Carbonic Anhydrase IX Isoenzyme.
Chemistry - A European Journal. Roč. 26, č. 69 (2020), s. 16541-16553. ISSN 0947-6539. E-ISSN 1521-3765
R&D Projects: GA ČR(CZ) GA18-27648S; GA ČR(CZ) GA15-05677S
Grant - others:AV ČR(CZ) L200321851
Program: Program podpory perspektivníchlidských zdrojů - postdoktorandů
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : medicinal chemistry * indomethacin * carbonic anhydrase * dicarba-closo-dodecaboranes * inhibitors * sulfonamide
OECD category: Inorganic and nuclear chemistry; Biochemistry and molecular biology (UMG-J)
Impact factor: 5.236, year: 2020
Method of publishing: Open access with time embargo
Permanent Link: http://hdl.handle.net/11104/0314883File Download Size Commentary Version Access Direct.pdf 2 1.8 MB Author’s postprint open-access Direct SI.pdf 0 5.2 MB Author’s postprint open-access - 5.0511423 - ÚOCHB 2020 RIV US eng J - Journal Article
Grüner, B. - Brynda, Jiří - Das, V. - Šícha, V. - Štěpánková, J. - Nekvinda, J. - Holub, J. - Pospíšilová, Klára - Fábry, M. - Pachl, Petr - Král, V. - Kugler, Michael - Mašek, V. - Medvedíková, M. - Matějková, Stanislava - Nová, A. - Lišková, B. - Gurská, S. - Džubák, P. - Hajdúch, M. - Řezáčová, Pavlína
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX.
Journal of Medicinal Chemistry. Roč. 62, č. 21 (2019), s. 9560-9575. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963
Keywords : cobalt bis(1,2-dicarbollide) * carborane complexes * medicinal chemistry
OECD category: Biochemistry and molecular biology
Impact factor: 6.205, year: 2019
Method of publishing: Limited access
https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.9b00945
Permanent Link: http://hdl.handle.net/11104/0301695 - 6.0506196 - ÚMG 2020 RIV US eng J - Journal Article
Brennecke, P. - Rasina, D. - Aubi, O. - Herzog, K. - Landskron, J. - Cautain, B. - Vicente, F. - Quintana, J. - Mestres, J. - Stechmann, B. - Ellinger, B. - Brea, J. - Kolanowski, J. L. - Pilarski, R. - Orzaez, M. - Pineda-Lucena, A. - Laraia, L. - Nami, F. - Zielenkiewicz, P. - Paruch, K. - Hansen, E. - von Kries, J.P. - Neuenschwander, M. - Specker, E. - Bartůněk, Petr - Šímová, Šárka - Lesnikowski, Z. - Krauss, S. - Lehtio, L. - Bilitewski, U. - Broenstrup, M. - Tasken, K. - Jirgensons, A. - Lickert, H. - Clausen, M. H. - Andersen, J. H. - Vicent, M. J. - Genilloud, O. - Martinez, A. - Nazare, M. - Fecke, W. - Gribbon, P.
EU-OPENSCREEN: A Novel Collaborative Approach to Facilitate Chemical Biology.
SLAS Discovery. Roč. 24, č. 3 (2019), s. 398-413. ISSN 2472-5552. E-ISSN 2472-5560
R&D Projects: GA MŠMT LO1220; GA MŠMT LM2015063
Institutional support: RVO:68378050
Keywords : chemical biology * screening * medicinal chemistry * open access * compound library
OECD category: Biochemical research methods
Impact factor: 2.195, year: 2019
Method of publishing: Open access
https://journals.sagepub.com/doi/10.1177/2472555218816276
Permanent Link: http://hdl.handle.net/11104/0297510 - 7.0502856 - ÚMG 2019 RIV US eng J - Journal Article
Bartůněk, Petr - Šímová, Šárka … Total 42 authors
EU-OPENSCREEN: A Novel Collaborative Approach to Facilitate Chemical Biology.
SLAS Discovery. Roč. 24, č. 3 (2019), s. 398-413. ISSN 2472-5552. E-ISSN 2472-5560
R&D Projects: GA MŠMT LO1220; GA MŠMT LM2015063
Institutional support: RVO:68378050
Keywords : chemical biology * screening * medicinal chemistry * open access * compound library
OECD category: Cell biology
Impact factor: 2.195, year: 2019
Permanent Link: http://hdl.handle.net/11104/0294735 - 8.0482693 - ÚOCHB 2018 RIV US eng J - Journal Article
Kolář, Michal H. - Tabarrini, O.
Halogen Bonding in Nucleic Acid Complexes.
Journal of Medicinal Chemistry. Roč. 60, č. 21 (2017), s. 8681-8690. ISSN 0022-2623. E-ISSN 1520-4804
Institutional support: RVO:61388963
Keywords : aldose reductase inhibition * minor groove binders * medicinal chemistry
OECD category: Physical chemistry
Impact factor: 6.253, year: 2017
Permanent Link: http://hdl.handle.net/11104/0278100 - 9.0446581 - ÚOCHB 2016 RIV DE eng J - Journal Article
Šála, Michal - Dejmek, Milan - Procházková, Eliška - Hřebabecký, Hubert - Rybáček, Jiří - Dračínský, Martin - Novák, Pavel - Rosenbergová, Šárka - Rosenberg, Ivan - Nencka, Radim
A New Analogue of Locked Cyclohexane Nucleic Acids.
Synthesis. Roč. 47, č. 17 (2015), s. 2654-2662. ISSN 0039-7881. E-ISSN 1437-210X
R&D Projects: GA ČR GPP207/12/P625; GA ČR GA13-26526S
Institutional support: RVO:61388963
Keywords : nucleosides * bicyclic compounds * oligonucleotides * carbocycles * medicinal chemistry
Subject RIV: CC - Organic Chemistry
Impact factor: 2.652, year: 2015
Permanent Link: http://hdl.handle.net/11104/0248634 - 10.0443641 - ÚACH 2016 US eng O - Others
Grüner, Bohumír - Štíbr, Bohumil
15th International Conference on Boron Chemistry (IMEBORON XV).
Pure and Applied Chemistry. Walter de Gruyter. Roč. 87, č. 2 (2015), s. 121. ISSN 0033-4545. E-ISSN 1365-3075
Institutional support: RVO:61388980
Keywords : boranes * boron * boron materials * carboranes * IMEBORON XV * medicinal chemistry
Subject RIV: CA - Inorganic Chemistry
Permanent Link: http://hdl.handle.net/11104/0246364