Search results
- 1.0585351 - FGÚ 2025 RIV NL eng J - Journal Article
Bencze, Michal - Boroš, Almoš - Behuliak, Michal - Vavřínová, Anna - Vaněčková, Ivana - Zicha, Josef
Changes in cardiovascular autonomic control induced by chronic inhibition of acetylcholinesterase during pyridostigmine or donepezil treatment of spontaneously hypertensive rats.
European Journal of Pharmacology. Roč. 971, 15 May (2024), č. článku 176526. ISSN 0014-2999. E-ISSN 1879-0712
R&D Projects: GA MŠMT(CZ) LX22NPO5104; GA ČR(CZ) GA21-03810S
Institutional support: RVO:67985823
Keywords : parasympathetic tone * sympathetic tone * sympathovagal control of heart rate * spontaneously hypertensive rats * Wistar-Kyoto rats * acetylcholinesterase inhibitors
OECD category: Physiology (including cytology)
Impact factor: 5, year: 2022
Method of publishing: Open access
https://doi.org/10.1016/j.ejphar.2024.176526
Permanent Link: https://hdl.handle.net/11104/0353070File Download Size Commentary Version Access 24_0040_0585351.pdf 0 7.3 MB Publisher’s postprint open-access - 2.0584241 - ÚEM 2025 RIV NL eng J - Journal Article
Mezeiová, E. - Prchal, L. - Hrabinová, M. - Mucková, L. - Pulkrabková, L. - Soukup, O. - Misiachna, Anna - Janoušek, J. - Fibigar, J. - Kučera, T. - Horák, Martin - Makhaeva, G.F. - Korabecný, J.
Morphing cholinesterase inhibitor amiridine into multipotent drugs for the
treatment of Alzheimer’s disease.
Biomedicine & Pharmacotherapy. Roč. 173, april. (2024), č. článku 116399. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
Keywords : amiridine * acetylcholinesterase * antioxidant capacity * butyrylcholinesterase * multi-target directed ligands * NMDA receptors
OECD category: Neurosciences (including psychophysiology
Impact factor: 7.5, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S075333222400283X?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0352201File Download Size Commentary Version Access Mezeirová 2024.pdf 1 1.7 MB Author´s preprint open-access - 3.0578898 - ÚEB 2024 RIV US eng J - Journal Article
Šachlevičiūtė, U. - Gonzalez, G. - Kvasnicová, M. - Štěpánková, Š. - Kleizienė, N. - Bieliauskas, A. - Zatloukal, M. - Strnad, Miroslav - Sløk, F. A. - Kvasnica, Miroslav - Šačkus, A. - Žukauskaitė, A.
Synthesis and neuroprotective activity of 3-aryl-3-azetidinyl acetic acid methyl ester derivatives.
Archiv der Pharmazie. Roč. 356, č. 12 (2023), č. článku 2300378. ISSN 0365-6233. E-ISSN 1521-4184
R&D Projects: GA ČR(CZ) GA23-05389S
Institutional support: RVO:61389030
Keywords : acetylcholinesterase * Alzheimer disease * azetidine * neuroprotection * Parkinson disease
OECD category: Biochemistry and molecular biology
Impact factor: 5.1, year: 2022
Method of publishing: Open access
https://doi.org/10.1002/ardp.202300378
Permanent Link: https://hdl.handle.net/11104/0347819File Download Size Commentary Version Access 2023_Sachleviciute_ARCHIV DER PHARMAZIE_e2300378..pdf 1 3.6 MB Other open-access - 4.0572189 - ÚEM 2024 RIV CH eng J - Journal Article
Svobodová, B. - Pulkrabová, L. - Pánek, D. - Misiachna, Anna - Kolcheva, Marharyta - Andrýs, R. - Handl, J. - Čapek, J. - Nývltová, P. - Roušar, T. - Prchal, L. - Hepnarová, V. - Hrabinová, M. - Mucková, L. - Tosnerová, D. - Karabanovich, G. - Finger, V. - Soukup, O. - Horák, Martin - Korabecný, J.
Structure-Guided Design of N-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer’s Disease.
International Journal of Molecular Sciences. Roč. 24, č. 11 (2023), č. článku 9124. ISSN 1661-6596
R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) LX22NPO5107
Institutional support: RVO:68378041
Keywords : Alzheimer’s disease * acetylcholinesterase * enzyme inhibition * N-methyl-d-aspartate receptor * multi-target directed ligands * monoamine oxidase A/B
OECD category: Pharmacology and pharmacy
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://doi.org/10.3390/ijms24119124
Permanent Link: https://hdl.handle.net/11104/0342960File Download Size Commentary Version Access Svobodová 2023.pdf 2 3.8 MB Publisher’s postprint open-access - 5.0570474 - ÚEB 2024 RIV GB eng J - Journal Article
Gonzalez, G. - Kvasnica, Miroslav - Svrčková, K. - Štěpánková, Š. - Santos, J. R. C. - Peřina, M. - Jorda, R. - Lopes, S. M.M. - Melo, T.
Ring-fused 3 beta-acetoxyandrost-5-enes as novel neuroprotective agents with cholinesterase inhibitory properties.
Journal of Steroid Biochemistry and Molecular Biology. Roč. 225, JAN (2023), č. článku 106194. ISSN 0960-0760
R&D Projects: GA ČR GA20-15621S
Institutional support: RVO:61389030
Keywords : Neuroprotective agents * Cholinesterase inhibitors * Acetylcholinesterase and butyrylcholinesterase * enzymes * Hexacyclic steroids * SteroidalN-sulfonyl-1-azadiene
OECD category: Biochemistry and molecular biology
Impact factor: 4.1, year: 2022
Method of publishing: Open access
https://doi.org/10.1016/j.jsbmb.2022.106194
Permanent Link: https://hdl.handle.net/11104/0341775File Download Size Commentary Version Access 2023_Gonzalez_JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY_106194.pdf 1 5.7 MB Other open-access - 6.0566059 - ÚEM 2023 RIV cze P - Patent Document
Soukup, O. - Korábečný, J. - Horák, Martin - Misiachna, Anna - Valeš, K. - Vyklický, L.
7-Fenoxytakrin a jeho použití.
[7-Phenoxytacrine and its use.]
2022. Owner: Fakultní nemocnice Hradec Králové - Ústav experimentální medicíny AV ČR, v. v. i. - Národní ústav duševního zdraví, p. o. - Fyziologický ústav AV ČR, v. v. i. Date of the patent acceptance: 22.04.2022. Patent Number: 309225
R&D Projects: GA MZd(CZ) NU20-08-00296
Institutional support: RVO:68378041
Keywords : NMDA receptor * dual drugs * Alzheimer's disease * acetylcholinesterase
OECD category: Pharmacology and pharmacy
https://isdv.upv.cz/doc/FullFiles/Patents/FullDocuments/309/309225.pdf
Permanent Link: https://hdl.handle.net/11104/0337498 - 7.0566057 - ÚEM 2023 RIV cze P - Patent Document
Soukup, O. - Korábečný, J. - Horák, Martin - Misiachna, Anna - Valeš, K. - Vyklický, L.
Duálně účinné deriváty takrinu a jejich použití.
[Tacrine derivatives possessing dual activity and their use.]
2022. Owner: Fakultní nemocnice Hradec Králové - Ústav experimentální medicíny AV ČR, v. v. i. - Národní ústav duševního zdraví, p. o. - Fyziologický ústav AV ČR, v. v. i. Date of the patent acceptance: 18.05.2022. Patent Number: 309262
Institutional support: RVO:68378041
Keywords : NMDA receptor * dual drugs * Alzheimer's disease * acetylcholinesterase
OECD category: Pharmacology and pharmacy
https://isdv.upv.cz/doc/FullFiles/Patents/FullDocuments/309/309262.pdf
Permanent Link: https://hdl.handle.net/11104/0337634 - 8.0564447 - FGÚ 2023 RIV cze P - Patent Document
Soukup, O. - Korábečný, J. - Horák, Martin - Misiachna, A. - Valeš, K. - Vyklický ml., Ladislav
7-Fenoxytakrin a jeho použití.
[7-Phenoxytacrine and its use.]
2022. Owner: Fakultní nemocnice Hradec Králové - Ústav experimentální medicíny AV ČR, v. v. i. - Národní ústav duševního zdraví, p. o. - Fyziologický ústav AV ČR, v. v. i. Date of the patent acceptance: 22.04.2022. Patent Number: 309225
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : NMDA receptor * dual drugs * Alzheimer´s disease * acetylcholinesterase
OECD category: Pharmacology and pharmacy
https://isdv.upv.cz/doc/FullFiles/Patents/FullDocuments/309/309225.pdf
Permanent Link: https://hdl.handle.net/11104/0336111 - 9.0564438 - FGÚ 2023 RIV cze P - Patent Document
Soukup, O. - Korábečný, J. - Horák, Martin - Misiachna, A. - Valeš, K. - Vyklický ml., Ladislav
Duálně účinné deriváty takrinu a jejich použití.
[Tacrine derivatives possessing dual activity and their use.]
2022. Owner: Fakultní nemocnice Hradec Králové - Ústav experimentální medicíny AV ČR, v. v. i. - Národní ústav duševního zdraví, p. o. - Fyziologický ústav AV ČR, v. v. i. Date of the patent acceptance: 18.05.2022. Patent Number: 309262
Institutional support: RVO:67985823
Keywords : NMDA receptor * dual drugs * Alzheimer´s disease * acetylcholinesterase
OECD category: Pharmacology and pharmacy
https://isdv.upv.cz/doc/FullFiles/Patents/FullDocuments/309/309262.pdf
Permanent Link: https://hdl.handle.net/11104/0336106 - 10.0561212 - FZÚ 2023 RIV US eng J - Journal Article
Nepovímová, E. - Svobodová, L. - Doležal, R. - Rostohar, Danijela … Total 30 authors
Tacrine – benzothiazoles: novel class of potential multitarget anti-Alzheimer's drugs dealing with cholinergic, amyloid and mitochondrial systems.
Bioorganic Chemistry. Roč. 107, Feb (2021), č. článku 104596. ISSN 0045-2068. E-ISSN 1090-2120
EU Projects: European Commission(XE) 654148 - LASERLAB-EUROPE
Institutional support: RVO:68378271
Keywords : Alzheimer's disease * tacrine * benzothiazole * acetylcholinesterase Inhibitors * amyloid beta * ABAD * MTDLs
OECD category: Optics (including laser optics and quantum optics)
Impact factor: 5.307, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bioorg.2020.104596
Permanent Link: https://hdl.handle.net/11104/0333898