Search results
- 1.0575132 - ÚOCHB 2024 RIV US eng J - Journal Article
Solntseva, E. I. - Bukanova, J. V. - Kondratenko, R. - Kudová, Eva
Corticosteroids as Selective and Effective Modulators of Glycine Receptors.
ACS Chemical Neuroscience. Roč. 14, č. 17 (2023), s. 3132-3142. ISSN 1948-7193. E-ISSN 1948-7193
R&D Projects: GA MŠMT(CZ) LX22NPO5104
Institutional support: RVO:61388963
Keywords : GABAA receptor * glycine receptor * corticosteroids * structure-activity relationship study
OECD category: Neurosciences (including psychophysiology
Impact factor: 5, year: 2022
Method of publishing: Open access
https://doi.org/10.1021/acschemneuro.3c00287
Permanent Link: https://hdl.handle.net/11104/0344992File Download Size Commentary Version Access 10.1021acschemneuro.3c00287.pdf 0 4 MB Publisher’s postprint open-access - 2.0392261 - ÚOCHB 2014 RIV US eng J - Journal Article
Slavíková, Barbora - Bujons, J. - Matyáš, Libor - Vidal, M. - Babot, Z. - Krištofíková, Z. - Suňol, C. - Kasal, Alexander
Allopregnanolone and Pregnanolone Analogues Modified in the C Ring: Synthesis and Activity.
Journal of Medicinal Chemistry. Roč. 56, č. 6 (2013), s. 2323-2336. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GAP303/12/1464
Institutional support: RVO:61388963
Keywords : steroids * synthesis of neurosteroid analogues * GABAA receptor * [3H]flunitrazepam binding * intact neurons in culture * 3D-QSAR analysis
Subject RIV: FR - Pharmacology ; Medidal Chemistry
Impact factor: 5.480, year: 2013
Permanent Link: http://hdl.handle.net/11104/0221183 - 3.0352785 - ÚOCHB 2011 RIV CZ cze P - Patent Document
Kasal, Alexander - Buděšínský, Miloš - Mareš, Pavel - Krištofíková, Z.
3alfa-Hydroxy-21ksí,22-oxido-21-homo-5alfa-pregnan-20-on, způsob jeho výroby a použití.
[3alpha-Hydroxy-21xi, 22-oxide-21-homo-5alpha-pregnan-20-one, process if its preparation and its use.]
Praha: Úřad průmyslového vlastnictví, 2010. Owner: Ústav organické chemie a biochemie AV ČR, v. v. i. - Fyziologický ústav AV ČR, v. v. i. - Psychiatrické centrum Praha. Date of the patent acceptance: 06.08.2010. Patent Number: 302050
Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50110509
Keywords : neurosteroids * receptors of gamma-aminobutyric acid * GABAA * TBPS * epilepsy
Subject RIV: CC - Organic Chemistry
http://spisy.upv.cz/Patents/FullDocuments/302/302050.pdf
Permanent Link: http://hdl.handle.net/11104/0192211 - 4.0346335 - ÚOCHB 2011 RIV FR eng J - Journal Article
Dansey, M. V. - Di Chenna, P. - Valeiro, A. S. - Krištofíková, Z. - Chodounská, Hana - Kasal, Alexander - Burton, G.
Synthesis and GABAA receptor activity of A-homo analogues of neuroactive steroids.
European Journal of Medicinal Chemistry. Roč. 45, č. 7 (2010), s. 3063-3069. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA203/08/1498
Institutional research plan: CEZ:AV0Z40550506
Keywords : A-homopregnane * neurosteroid * gamma-aminobutyric acid * GABAA receptor
Subject RIV: CC - Organic Chemistry
Impact factor: 3.193, year: 2010
Permanent Link: http://hdl.handle.net/11104/0187392 - 5.0324227 - ÚOCHB 2009 RIV CZ eng J - Journal Article
Kapras, Vojtěch - Šťastná, Eva - Chodounská, Hana - Pouzar, Vladimír - Krištofíková, Zdena
Preparation of steroid sulfamates and their interaction with GABAA receptor.
[Příprava steroidních sulfamátů a jejich interakce s MNDA receptory.]
Collection of Czechoslovak Chemical Communications. Roč. 74, č. 4 (2009), s. 643-650. ISSN 0010-0765
R&D Projects: GA ČR(CZ) GA203/08/1498
Institutional research plan: CEZ:AV0Z40550506
Keywords : sulfamates * neurosteroids * GABAA receptors * pregnane
Subject RIV: CC - Organic Chemistry
Impact factor: 0.856, year: 2009
Permanent Link: http://hdl.handle.net/11104/0171978 - 6.0042101 - ÚOCHB 2007 RIV US eng J - Journal Article
Havlíková, H. - Hill, M. - Kancheva, L. - Vrbíková, J. - Pouzar, Vladimír - Černý, Ivan - Kancheva, R. - Stárka, L.
Serum profiles of free and conjugated neuroactive pregnanolone isomers in nonpregnant women of fertile age.
[Sérové profily volných a konjugovaných neuroaktivních pregnanolonových isomerů u netěhotných žen v produktivním věku.]
Journal of Clinical Endocrinology and Metabolism. Roč. 91, č. 8 (2006), s. 3092-3099. ISSN 0021-972X. E-ISSN 1945-7197
R&D Projects: GA MZd(CZ) NR7768
Institutional research plan: CEZ:AV0Z40550506
Keywords : pregnanolone isomers * GABAA * steroids
Subject RIV: CC - Organic Chemistry
Impact factor: 5.799, year: 2006
Permanent Link: http://hdl.handle.net/11104/0135409 - 7.0041903 - ÚOCHB 2007 RIV US eng J - Journal Article
Suňol, C. - García, D. A. - Bujons, J. - Krištofíková, Zdena - Matyáš, Libor - Babot, Z. - Kasal, Alexander
Activity of B-Nor Analogues of Neurosteroids on the GABAA Receptor in Primary Neuronal Cultures.
[Účinky B-noranalog neurosteroidů na GABAA receptor měřené na primární kultuře neuronů.]
Journal of Medicinal Chemistry. Roč. 49, č. 11 (2006), s. 3225-3224. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GA203/06/1605
Grant - others:FEDER(ES) SAF20003-04930; CIRIT(ES) 2001SGR00355
Institutional research plan: CEZ:AV0Z40550506
Keywords : neurosteroid * GABAA receptor * B-nor steroids * 7-nor steroids
Subject RIV: CC - Organic Chemistry
Impact factor: 5.115, year: 2006
Permanent Link: http://hdl.handle.net/11104/0135246