Search results

  1. 1.
    0582133 - ÚEM 2025 RIV NL eng J - Journal Article
    Misiachna, Anna - Svobodová, B. - Netolický, Jakub - Chvojková, M. - Kletečková, L. - Prchal, L. - Novák, M. - Hrabinová, M. - Kučera, T. - Mucková, L. - Moravcová, Z. - Karasová-Ždárová, J. - Pejchal, J. - Blažek, F. - Maliňák, D. - Hakenová, K. - Hrčka Krausová, Barbora - Kolcheva, Marharyta - Ladislav, Marek - Korábečný, J. - Pahnke, J. - Valeš, K. - Horák, Martin - Soukup, O.
    Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition.
    European Journal of Medicinal Chemistry. Roč. 266, feb. (2024), č. článku 116130. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA TA ČR(CZ) TO01000078; GA MŠMT(CZ) EH22_008/0004562
    Institutional support: RVO:68378041
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 6.7, year: 2022
    Method of publishing: Open access
    https://www.sciencedirect.com/science/article/pii/S0223523424000102?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0350209
    FileDownloadSizeCommentaryVersionAccess
    Misiachna 2024.pdf45 MBPublisher’s postprintopen-access
     
     
  2. 2.
    0551558 - ÚEM 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
    Institutional support: RVO:68378041
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
    OECD category: Medicinal chemistry
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0326821
     
     
  3. 3.
    0543492 - ÚEM 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA ČR(CZ) GA20-12047S
    Institutional support: RVO:68378041
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320802
     
     
  4. 4.
    0543350 - FGÚ 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, Kristína - Kletečková, Lenka - Chvojková, Markéta - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Krausová, B. - Horák, Martin - Valeš, Karel - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, Apr (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320571
     
     
  5. 5.
    0542659 - FGÚ 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
    OECD category: Pharmacology and pharmacy
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0320032
     
     


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