Search results
- 1.0531944 - FGÚ 2021 RIV US eng J - Journal Article
Hrčka Krausová, Barbora - Kysilov, Bohdan - Černý, Jiří - Vyklický, Vojtěch - Smejkalová, Tereza - Ladislav, Marek - Balík, Aleš - Kořínek, Miloslav - Chodounská, Hana - Kudová, Eva - Vyklický ml., Ladislav
Site of Action of Brain Neurosteroid Pregnenolone Sulfate at the N-Methyl-D-Aspartate Receptor.
Journal of Neuroscience. Roč. 40, č. 31 (2020), s. 5922-5936. ISSN 0270-6474. E-ISSN 1529-2401
R&D Projects: GA ČR(CZ) GA17-02300S; GA ČR(CZ) GJ16-03913Y; GA TA ČR(CZ) TN01000013; GA ČR(CZ) GA20-17945S; GA MŠMT(CZ) LQ1604
Institutional support: RVO:67985823 ; RVO:61388963
Keywords : glutamate receptors * neurosteroids * patch clamp * structure
OECD category: Neurosciences (including psychophysiology
Impact factor: 6.167, year: 2020 ; AIS: 2.649, rok: 2020
Method of publishing: Open access with time embargo
Result website:
https://doi.org/10.1523/JNEUROSCI.3010-19.2020DOI: https://doi.org/10.1523/JNEUROSCI.3010-19.2020
Permanent Link: http://hdl.handle.net/11104/0310574 - 2.0531929 - FGÚ 2021 RIV GB eng J - Journal Article
Kořínek, Miloslav - González-González, I. M. - Smejkalová, Tereza - Hajduković, Dragana - Skřenková, Kristýna - Krůšek, Jan - Horák, Martin - Vyklický ml., Ladislav
Cholesterol modulates presynaptic and postsynaptic properties of excitatory synaptic transmission.
Scientific Reports. Roč. 10, č. 1 (2020), č. článku 12651. ISSN 2045-2322. E-ISSN 2045-2322
R&D Projects: GA ČR(CZ) GA17-02300S; GA ČR(CZ) GJ16-03913Y; GA TA ČR(CZ) TN01000013; GA MŠMT(CZ) LQ1604
Institutional support: RVO:67985823
Keywords : synaptic transmission * cholesterol * NMDA receptor * NMDA receptor * neuroprotection * synapse * membrane
OECD category: Neurosciences (including psychophysiology
Impact factor: 4.380, year: 2020 ; AIS: 1.285, rok: 2020
Method of publishing: Open access
Result website:
https://www.nature.com/articles/s41598-020-69454-5DOI: https://doi.org/10.1038/s41598-020-69454-5
Permanent Link: http://hdl.handle.net/11104/0310562 - 3.0517459 - FGÚ 2020 RIV CH eng J - Journal Article
Černý, Jiří - Božíková, P. - Balík, Aleš - Marques, S. M. - Vyklický ml., Ladislav
NMDA Receptor Opening and Closing-Transitions of a Molecular Machine Revealed by Molecular Dynamics.
Biomolecules. Roč. 9, č. 10 (2019), č. článku 546. ISSN 2218-273X. E-ISSN 2218-273X
R&D Projects: GA ČR(CZ) GA17-02300S; GA TA ČR(CZ) TN01000013; GA MŠMT(CZ) ED1.1.00/02.0109
Research Infrastructure: CESNET II - 90042; CERIT-SC - 90085; ELIXIR-CZ - 90047
Institutional support: RVO:67985823
Keywords : glutamate receptor gating * molecular modeling * molecular dynamics simulations * NMDA receptor transition * open and closed state
OECD category: Neurosciences (including psychophysiology
Impact factor: 4.082, year: 2019
Method of publishing: Open access
Result website:
https://doi.org/10.3390/biom9100546DOI: https://doi.org/10.3390/biom9100546
Permanent Link: http://hdl.handle.net/11104/0302760 - 4.0501437 - ÚOCHB 2020 RIV US eng J - Journal Article
Matoušová, Marika - Souček, Radko - Tloušťová, Eva - Slavíková, Barbora - Chodounská, Hana - Mertlíková-Kaiserová, Helena - Kudová, Eva
Pregn-5-en-3beta-ol and androst-5-en-3beta-ol dicarboxylic acid esters as potential therapeutics for NMDA hypofunction: In vitro safety assessment and plasma stability.
Steroids. Roč. 147, Jul (2019), s. 4-9. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA ČR(CZ) GA17-02300S; GA MZd(CZ) NV15-29370A; GA MŠMT LO1302
Institutional support: RVO:61388963
Keywords : neurosteroid * NMDA receptor hypofunction * hepatotoxicity * mitotoxicity * Caco-2 permeability * plasma stability
OECD category: Neurosciences (including psychophysiology
Impact factor: 1.948, year: 2019 ; AIS: 0.481, rok: 2019
Method of publishing: Limited access
Result website:
https://www.sciencedirect.com/science/article/abs/pii/S0039128X18301752?via%3DihubDOI: https://doi.org/10.1016/j.steroids.2018.09.012
Permanent Link: http://hdl.handle.net/11104/0296235 - 5.0498559 - ÚOCHB 2019 RIV CH eng J - Journal Article
Adla, Santosh Kumar - Slavíková, Barbora - Chodounská, Hana - Vyklický, Vojtěch - Ladislav, Marek - Hubálková, Pavla - Krausová, Barbora - Smejkalová, Tereza - Nekardová, Michaela - Šmídková, Markéta - Monincová, Lenka - Souček, Radko - Vyklický ml., Ladislav - Kudová, Eva
Strong Inhibitory Effect, Low Cytotoxicity and High Plasma Stability of Steroidal Inhibitors of N-Methyl-D-Aspartate Receptors With C-3 Amide Structural Motif.
Frontiers in Pharmacology. Roč. 9, Nov 12 (2018), č. článku 1299. ISSN 1663-9812. E-ISSN 1663-9812
R&D Projects: GA TA ČR(CZ) TE01020028; GA ČR(CZ) GBP208/12/G016; GA ČR(CZ) GA17-02300S; GA ČR(CZ) GJ16-03913Y; GA MZd(CZ) NV15-29370A; GA MŠMT LO1302; GA MŠMT(CZ) ED1.1.00/02.0109
Grant - others:AV ČR(CZ) MSM200111601
Program: Program na podporu mezinárodní spolupráce začínajících výzkumných pracovníků
Institutional support: RVO:61388963 ; RVO:67985823
Keywords : neurosteroid * amide * NMDA receptor * plasma stability * structure-activity relationship
OECD category: Biochemistry and molecular biology
Impact factor: 3.845, year: 2018 ; AIS: 1.047, rok: 2018
Result website:
https://www.frontiersin.org/articles/10.3389/fphar.2018.01299/fullDOI: https://doi.org/10.3389/fphar.2018.01299
Permanent Link: http://hdl.handle.net/11104/0291127 - 6.0490287 - FGÚ 2019 RIV US eng J - Journal Article
Krausová, Barbora - Slavíková, Barbora - Nekardová, Michaela - Hubálková, Pavla - Vyklický, Vojtěch - Chodounská, Hana - Vyklický ml., Ladislav - Kudová, Eva
Positive Modulators of the N-Methyl-D-aspartate Receptor: Structure-Activity Relationship Study of Steroidal 3-Hemiesters.
Journal of Medicinal Chemistry. Roč. 61, č. 10 (2018), s. 4505-4516. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GA17-02300S; GA ČR(CZ) GBP208/12/G016; GA TA ČR(CZ) TE01020028; GA MZd(CZ) NV15-29370A; GA MŠMT(CZ) ED1.1.00/02.0109
Grant - others:AV ČR(CZ) MSM200111601
Program: Program na podporu mezinárodní spolupráce začínajících výzkumných pracovníků
Institutional support: RVO:67985823 ; RVO:61388963
Keywords : neurosteroids * N-Methyl-D-aspartate receptor * positive modulators
OECD category: Neurosciences (including psychophysiology
Impact factor: 6.054, year: 2018 ; AIS: 1.522, rok: 2018
DOI: https://doi.org/10.1021/acs.jmedchem.8b00255
Permanent Link: http://hdl.handle.net/11104/0284547 - 7.0489301 - FGÚ 2019 RIV CH eng J - Journal Article
Ladislav, Marek - Černý, Jiří - Krůšek, Jan - Horák, Martin - Balík, Aleš - Vyklický ml., Ladislav
The LILI Motif of M3-S2 Linkers Is a Component of the NMDA Receptor Channel Gate.
Frontiers in Molecular Neuroscience. Roč. 11, Apr 6 (2018), č. článku 113. ISSN 1662-5099. E-ISSN 1662-5099
R&D Projects: GA ČR(CZ) GA17-02300S; GA TA ČR(CZ) TE01020028; GA MZd(CZ) NV15-29370A; GA MŠMT(CZ) LQ1604; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:67985823
Keywords : glutamate receptor gating * electrophysiology * spontaneous activity * channel open probability * protein block alphabet * molecular modeling
OECD category: Neurosciences (including psychophysiology
Impact factor: 3.720, year: 2018 ; AIS: 1.346, rok: 2018
DOI: https://doi.org/10.3389/fnmol.2018.00113
Permanent Link: http://hdl.handle.net/11104/0283746 - 8.0489295 - FGÚ 2019 RIV CH eng J - Journal Article
Vyklický, Vojtěch - Krausová, Barbora - Černý, Jiří - Ladislav, Marek - Smejkalová, Tereza - Kysilov, Bohdan - Kořínek, Miloslav - Danačíková, Šárka - Horák, Martin - Chodounská, Hana - Kudová, Eva - Vyklický ml., Ladislav
Surface Expression, Function, and Pharmacology of Disease-Associated Mutations in the Membrane Domain of the Human GluN2B Subunit.
Frontiers in Molecular Neuroscience. Roč. 11, Apr 6 (2018), č. článku 110. ISSN 1662-5099. E-ISSN 1662-5099
R&D Projects: GA ČR(CZ) GA17-02300S; GA ČR(CZ) GJ16-03913Y; GA TA ČR(CZ) TE01020028; GA MZd(CZ) NV15-29370A; GA MŠMT(CZ) ED1.1.00/02.0109
Grant - others:AV ČR(CZ) MSM200111601
Program: Program na podporu mezinárodní spolupráce začínajících výzkumných pracovníků
Institutional support: RVO:67985823 ; RVO:61388963
Keywords : NMDA receptor * GluN2B * de novo missense mutations * neuropsychiatric disorder * neurosteroids
OECD category: Neurosciences (including psychophysiology
Impact factor: 3.720, year: 2018 ; AIS: 1.346, rok: 2018
DOI: https://doi.org/10.3389/fnmol.2018.00110
Permanent Link: http://hdl.handle.net/11104/0283743 - 9.0475702 - FGÚ 2018 RIV US eng J - Journal Article
Petrovič, Miloš - da Silva, S. V. - Clement, J. P. - Vyklický ml., Ladislav - Mulle, C. - González-González, I. M. - Henley, J. M.
Metabotropic action of postsynaptic kainate receptors triggers hippocampal long-term potentiation.
Nature Neuroscience. Roč. 20, č. 4 (2017), s. 529-539. ISSN 1097-6256. E-ISSN 1546-1726
R&D Projects: GA ČR(CZ) GA17-02300S
Institutional support: RVO:67985823
Keywords : hippocampus * long-term potentiation * membrane proteins
OECD category: Neurosciences (including psychophysiology
Impact factor: 19.912, year: 2017 ; AIS: 10.1, rok: 2017
DOI: https://doi.org/10.1038/nn.4505
Permanent Link: http://hdl.handle.net/11104/0272353