Search results
- 1.0569736 - MBÚ 2024 RIV NL eng J - Journal Article
Bavlovič, J. - Pávková, I. - Balonová, L. - Benada, Oldřich - Štulík, J. - Klimentová, J.
Intact O-antigen is critical structure for the exceptional tubular shape of outer membrane vesicles in Francisella tularensis.
Microbiological Research. Roč. 269, April 2023 (2023), č. článku 127300. ISSN 0944-5013. E-ISSN 1618-0623
R&D Projects: GA ČR(CZ) GA22-06771S
Institutional support: RVO:61388971
Keywords : Francisella tularensis * Outer membrane vesicles * Nanotubes * Lipopolysaccharide * Capsule * O-antigen
OECD category: Microbiology
Impact factor: 6.7, year: 2022
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0944501323000010?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0342544 - 2.0556370 - FGÚ 2023 RIV FR eng J - Journal Article
Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
OECD category: Pharmacology and pharmacy
Impact factor: 6.7, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2022.114193
Permanent Link: http://hdl.handle.net/11104/0330742 - 3.0545566 - ÚOCHB 2022 RIV CZ eng J - Journal Article
Kubelková, K. - Hubálek, Martin - Řehulka, P. - Řehulková, H. - Friedecký, D. - Žáková, J. - Macela, A.
Molecular characterization of alcohol–ether extract from bovine tissue.
Military Medical Science Letters. Roč. 90, č. 3 (2021), s. 120-136. ISSN 0372-7025. E-ISSN 2571-113X
Institutional support: RVO:61388963
Keywords : bovine tissue extract * Juvenil * molecular composition * psychobiotics * biological response modifier * antimicrobial peptides * defensin * hemocidin
OECD category: Analytical chemistry
Method of publishing: Open access
http://doi.org/10.31482/mmsl.2021.012
Permanent Link: http://hdl.handle.net/11104/0322253 - 4.0543492 - ÚEM 2022 RIV US eng J - Journal Article
Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
R&D Projects: GA ČR(CZ) GA20-12047S
Institutional support: RVO:68378041
Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
OECD category: Pharmacology and pharmacy
Impact factor: 6.100, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bcp.2021.114460
Permanent Link: http://hdl.handle.net/11104/0320802 - 5.0543350 - FGÚ 2022 RIV US eng J - Journal Article
Kaniaková, Martina - Korábečný, J. - Holubová, Kristína - Kletečková, Lenka - Chvojková, Markéta - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Krausová, B. - Horák, Martin - Valeš, Karel - Soukup, O.
7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
Biochemical Pharmacology. Roč. 186, Apr (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
OECD category: Pharmacology and pharmacy
Impact factor: 6.100, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bcp.2021.114460
Permanent Link: http://hdl.handle.net/11104/0320571 - 6.0542659 - FGÚ 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
OECD category: Pharmacology and pharmacy
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0320032 - 7.0541833 - ÚEM 2022 RIV CH eng J - Journal Article
Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
R&D Projects: GA MZd(CZ) NU20-08-00296
Research Infrastructure: e-INFRA CZ - 90140
Institutional support: RVO:68378041
Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
OECD category: Pharmacology and pharmacy
Impact factor: 6.064, year: 2021
Method of publishing: Open access
https://www.mdpi.com/2218-273X/11/1/3
Permanent Link: http://hdl.handle.net/11104/0319349 - 8.0541714 - ÚOCHB 2022 RIV CH eng J - Journal Article
Hudáčová, M. - Hamuľaková, S. - Konkoľová, Eva - Jendželovský, R. - Vargová, J. - Ševc, J. - Fedoročko, P. - Soukup, O. - Janočková, J. - Ihnatová, V. - Kučera, T. - Bzonek, P. - Nováková, N. - Jun, D. - Junová, L. - Korábečný, J. - Kuča, K. - Kožurková, M.
Synthesis of New Biscoumarin Derivatives, In Vitro Cholinesterase Inhibition, Molecular Modelling and Antiproliferative Effect in A549 Human Lung Carcinoma Cells.
International Journal of Molecular Sciences. Roč. 22, č. 8 (2021), č. článku 3830. E-ISSN 1422-0067
Institutional support: RVO:61388963
Keywords : biscoumarin * Alzheimer’s disease * blood–brain barrier * cholinesterase * antiproliferative activity * A549
OECD category: Biochemistry and molecular biology
Impact factor: 6.208, year: 2021
Method of publishing: Open access
https://doi.org/10.3390/ijms22083830
Permanent Link: http://hdl.handle.net/11104/0319265 - 9.0541685 - FGÚ 2022 RIV CH eng J - Journal Article
Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
Research Infrastructure: e-INFRA CZ - 90140
Institutional support: RVO:67985823
Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
OECD category: Pharmacology and pharmacy
Impact factor: 6.064, year: 2021
Method of publishing: Open access
https://www.mdpi.com/2218-273X/11/1/3
Permanent Link: http://hdl.handle.net/11104/0319216 - 10.0541608 - MBÚ 2022 RIV GB eng J - Journal Article
Kubelková, K. - Hudcovic, Tomáš - Kozáková, Hana - Pejchal, J. - Macela, A.
Early infection-induced natural antibody response.
Scientific Reports. Roč. 11, č. 1 (2021), č. článku 1541. ISSN 2045-2322. E-ISSN 2045-2322
R&D Projects: GA ČR(CZ) GA19-08294S
Institutional support: RVO:61388971
Keywords : live vaccine strain * bacterium francisella-tularensis * early protective immunity * intracellular bacterium * t-cells
OECD category: Infectious Diseases
Impact factor: 4.997, year: 2021
Method of publishing: Open access
https://www.nature.com/articles/s41598-021-81083-0
Permanent Link: http://hdl.handle.net/11104/0319141