Search results

  1. 1.
    0569736 - MBÚ 2024 RIV NL eng J - Journal Article
    Bavlovič, J. - Pávková, I. - Balonová, L. - Benada, Oldřich - Štulík, J. - Klimentová, J.
    Intact O-antigen is critical structure for the exceptional tubular shape of outer membrane vesicles in Francisella tularensis.
    Microbiological Research. Roč. 269, April 2023 (2023), č. článku 127300. ISSN 0944-5013. E-ISSN 1618-0623
    R&D Projects: GA ČR(CZ) GA22-06771S
    Institutional support: RVO:61388971
    Keywords : Francisella tularensis * Outer membrane vesicles * Nanotubes * Lipopolysaccharide * Capsule * O-antigen
    OECD category: Microbiology
    Impact factor: 6.7, year: 2022
    Method of publishing: Limited access
    https://www.sciencedirect.com/science/article/pii/S0944501323000010?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0342544
     
     
  2. 2.
    0556370 - FGÚ 2023 RIV FR eng J - Journal Article
    Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
    Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
    European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
    Institutional support: RVO:67985823
    Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.7, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1016/j.ejmech.2022.114193
    Permanent Link: http://hdl.handle.net/11104/0330742
     
     
  3. 3.
    0545566 - ÚOCHB 2022 RIV CZ eng J - Journal Article
    Kubelková, K. - Hubálek, Martin - Řehulka, P. - Řehulková, H. - Friedecký, D. - Žáková, J. - Macela, A.
    Molecular characterization of alcohol–ether extract from bovine tissue.
    Military Medical Science Letters. Roč. 90, č. 3 (2021), s. 120-136. ISSN 0372-7025. E-ISSN 2571-113X
    Institutional support: RVO:61388963
    Keywords : bovine tissue extract * Juvenil * molecular composition * psychobiotics * biological response modifier * antimicrobial peptides * defensin * hemocidin
    OECD category: Analytical chemistry
    Method of publishing: Open access
    http://doi.org/10.31482/mmsl.2021.012
    Permanent Link: http://hdl.handle.net/11104/0322253
     
     
  4. 4.
    0543492 - ÚEM 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA ČR(CZ) GA20-12047S
    Institutional support: RVO:68378041
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320802
     
     
  5. 5.
    0543350 - FGÚ 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, Kristína - Kletečková, Lenka - Chvojková, Markéta - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Krausová, B. - Horák, Martin - Valeš, Karel - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, Apr (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320571
     
     
  6. 6.
    0542659 - FGÚ 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
    OECD category: Pharmacology and pharmacy
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0320032
     
     
  7. 7.
    0541833 - ÚEM 2022 RIV CH eng J - Journal Article
    Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
    Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
    Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
    R&D Projects: GA MZd(CZ) NU20-08-00296
    Research Infrastructure: e-INFRA CZ - 90140
    Institutional support: RVO:68378041
    Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/1/3
    Permanent Link: http://hdl.handle.net/11104/0319349
     
     
  8. 8.
    0541714 - ÚOCHB 2022 RIV CH eng J - Journal Article
    Hudáčová, M. - Hamuľaková, S. - Konkoľová, Eva - Jendželovský, R. - Vargová, J. - Ševc, J. - Fedoročko, P. - Soukup, O. - Janočková, J. - Ihnatová, V. - Kučera, T. - Bzonek, P. - Nováková, N. - Jun, D. - Junová, L. - Korábečný, J. - Kuča, K. - Kožurková, M.
    Synthesis of New Biscoumarin Derivatives, In Vitro Cholinesterase Inhibition, Molecular Modelling and Antiproliferative Effect in A549 Human Lung Carcinoma Cells.
    International Journal of Molecular Sciences. Roč. 22, č. 8 (2021), č. článku 3830. E-ISSN 1422-0067
    Institutional support: RVO:61388963
    Keywords : biscoumarin * Alzheimer’s disease * blood–brain barrier * cholinesterase * antiproliferative activity * A549
    OECD category: Biochemistry and molecular biology
    Impact factor: 6.208, year: 2021
    Method of publishing: Open access
    https://doi.org/10.3390/ijms22083830
    Permanent Link: http://hdl.handle.net/11104/0319265
     
     
  9. 9.
    0541685 - FGÚ 2022 RIV CH eng J - Journal Article
    Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
    Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
    Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
    Research Infrastructure: e-INFRA CZ - 90140
    Institutional support: RVO:67985823
    Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/1/3
    Permanent Link: http://hdl.handle.net/11104/0319216
     
     
  10. 10.
    0541608 - MBÚ 2022 RIV GB eng J - Journal Article
    Kubelková, K. - Hudcovic, Tomáš - Kozáková, Hana - Pejchal, J. - Macela, A.
    Early infection-induced natural antibody response.
    Scientific Reports. Roč. 11, č. 1 (2021), č. článku 1541. ISSN 2045-2322. E-ISSN 2045-2322
    R&D Projects: GA ČR(CZ) GA19-08294S
    Institutional support: RVO:61388971
    Keywords : live vaccine strain * bacterium francisella-tularensis * early protective immunity * intracellular bacterium * t-cells
    OECD category: Infectious Diseases
    Impact factor: 4.997, year: 2021
    Method of publishing: Open access
    https://www.nature.com/articles/s41598-021-81083-0
    Permanent Link: http://hdl.handle.net/11104/0319141
     
     

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