Search results
- 1.0469894 - ÚOCHB 2017 RIV DE eng J - Journal Article
Machara, A. - Konvalinka, Jan - Kotora, M.
A Modular Synthesis of N-Benzotriazole Ureas Using Alkylation of 5-Nitrobenzotriazole.
ChemistrySelect. Roč. 1, č. 1 (2016), s. 101-107. ISSN 2365-6549. E-ISSN 2365-6549
R&D Projects: GA ČR GA13-19561S
Institutional support: RVO:61388963
Keywords : benzotriazole * alkylation * urea * isocyanate * reduction
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0267663 - 2.0463882 - ÚOCHB 2017 RIV FR eng J - Journal Article
Albinana, C. B. - Machara, A. - Řezáčová, Pavlína - Pachl, Petr - Konvalinka, Jan - Kožíšek, Milan
Kinetic, thermodynamic and structural analysis of tamiphosphor binding to neuraminidase of H1N1 (2009) pandemic influenza.
European Journal of Medicinal Chemistry. Roč. 121, Oct 4 (2016), s. 100-109. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR GA13-19561S; GA MŠMT LO1302; GA MŠMT(CZ) LO1304
Institutional support: RVO:61388963
Keywords : influenza neuraminidase * oseltamivir * tamiphosphor * isothermal titration calorimetry * crystal structure * lattice-translocation defect
Subject RIV: CE - Biochemistry
Impact factor: 4.519, year: 2016
Permanent Link: http://hdl.handle.net/11104/0262963 - 3.0463437 - ÚOCHB 2017 RIV GB eng J - Journal Article
Kožíšek, Milan - Štěpánek, Ondřej - Parkan, Kamil - Albinana, C. B. - Pávová, Marcela - Weber, Jan - Kräusslich, H. G. - Konvalinka, Jan - Machara, A.
Synthesis and evaluation of 2-pyridinylpyrimidines as inhibitors of HIV-1 structural protein assembly.
Bioorganic and Medicinal Chemistry Letters. Roč. 26, č. 15 (2016), s. 3487-3490. ISSN 0960-894X. E-ISSN 1464-3405
R&D Projects: GA ČR GA13-19561S; GA MŠMT(CZ) LK11207
Institutional support: RVO:61388963
Keywords : assay * assembly * capsid * inhibition * pyrimidine
Subject RIV: CE - Biochemistry
Impact factor: 2.454, year: 2016
http://www.sciencedirect.com/science/article/pii/S0960894X16306503
Permanent Link: http://hdl.handle.net/11104/0262633 - 4.0458499 - ÚOCHB 2017 RIV US eng J - Journal Article
Machara, A. - Lux, V. - Kožíšek, Milan - Grantz Šašková, Klára - Štěpánek, O. - Kotora, M. - Parkan, Kamil - Pávová, Marcela - Glass, B. - Sehr, P. - Lewis, J. - Müller, B. - Kräusslich, H. G. - Konvalinka, Jan
Specific Inhibitors of HIV Capsid Assembly Binding to the C-Terminal Domain of the Capsid Protein: Evaluation of 2-Arylquinazolines as Potential Antiviral Compounds.
Journal of Medicinal Chemistry. Roč. 59, č. 2 (2016), s. 545-558. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR GA13-19561S
EU Projects: European Commission(XE) 201095 - HIV ACE
Institutional support: RVO:61388963
Keywords : HIV-1 assembly * capsid * high-throughput screening * AlphaScreen assay
Subject RIV: CE - Biochemistry
Impact factor: 6.259, year: 2016
Permanent Link: http://hdl.handle.net/11104/0258765