Search results
- 1.0558143 - ÚMCH 2023 RIV CH eng J - Journal Article
Studenovský, Martin - Rumlerová, Anna - Kovářová, Jiřina - Dvořáková, Barbora - Sivák, Ladislav - Kostka, Libor - Berdár, Daniel - Etrych, Tomáš - Kovář, Marek
HPMA copolymer mebendazole conjugate allows systemic administration and possesses antitumour activity in vivo.
Pharmaceutics. Roč. 14, č. 6 (2022), č. článku 1201. E-ISSN 1999-4923
R&D Projects: GA ČR(CZ) GA19-05649S; GA MŠMT(CZ) LTAUSA18083
Grant - others:AV ČR(CZ) JSPS-22-01
Program: Bilaterální spolupráce
Institutional support: RVO:61389013 ; RVO:61388971
Keywords : mebendazole * drug delivery * cancer therapy
OECD category: Polymer science; Pharmacology and pharmacy (MBU-M)
Impact factor: 5.4, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1999-4923/14/6/1201
Permanent Link: https://hdl.handle.net/11104/0333076 - 2.0558142 - ÚMCH 2023 RIV US eng J - Journal Article
Kostka, Libor - Sivák, Ladislav - Šubr, Vladimír - Kovářová, Jiřina - Šírová, Milada - Říhová, Blanka - Sedláček, Radislav - Etrych, Tomáš - Kovář, Marek
Simultaneous delivery of doxorubicin and protease inhibitor derivative to solid tumors via star-shaped polymer nanomedicines overcomes P-gp- and STAT3-mediated chemoresistance.
Biomacromolecules. Roč. 23, č. 6 (2022), s. 2522-2535. ISSN 1525-7797. E-ISSN 1526-4602
R&D Projects: GA ČR(CZ) GA19-05649S; GA MZd(CZ) NU21-03-00273; GA MŠMT(CZ) LTAUSA18083; GA MŠMT(CZ) LM2018126; GA MŠMT(CZ) ED1.1.00/02.0109
Research Infrastructure: CCP II - 90126
Institutional support: RVO:61389013 ; RVO:61388971 ; RVO:68378050
Keywords : HPMA * RAFT * star-like
OECD category: Polymer science; Microbiology (MBU-M); Genetics and heredity (medical genetics to be 3) (UMG-J)
Impact factor: 6.2, year: 2022
Method of publishing: Limited access
https://pubs.acs.org/doi/10.1021/acs.biomac.2c00256
Permanent Link: https://hdl.handle.net/11104/0332796 - 3.0550778 - MBÚ 2022 RIV GB eng J - Journal Article
Tomala, Jakub - Weberová, Petra - Tomalová, Barbora - Zákostelská, Zuzana - Sivák, Ladislav - Kovářová, Jiřina - Kovář, Marek
IL-2/JES6-1 mAb complexes dramatically increase sensitivity to LPS through IFN-gamma production by CD25(+)Foxp3(-) T cells.
eLife. Roč. 10, DEC 21 2021 (2021), č. článku e62432. ISSN 2050-084X. E-ISSN 2050-084X
R&D Projects: GA ČR GA13-12885S; GA ČR(CZ) GA18-12973S; GA MZd(CZ) NV19-03-00179
Institutional support: RVO:61388971
Keywords : il-2 * tolerance * responses * suppression * il-2 * anti-il-2 mab complexes * cd25 * T cells * IFN-gamma * lps * hyperreactivity * Mouse
OECD category: Immunology
Impact factor: 8.713, year: 2021
Method of publishing: Open access
https://elifesciences.org/articles/62432
Permanent Link: http://hdl.handle.net/11104/0326088 - 4.0542896 - MBÚ 2022 RIV NL eng J - Journal Article
Sivák, Ladislav - Šubr, Vladimír - Kovářová, Jiřina - Dvořáková, Barbora - Šírová, Milada - Říhová, Blanka - Randárová, Eva - Kraus, Michal - Tomala, Jakub - Studenovský, Martin - Vondráčková, Michaela - Sedláček, Radislav - Makovický, Peter - Fučíková, J. - Vošahlíková, Š. - Spíšek, R. - Kostka, Libor - Etrych, Tomáš - Kovář, Marek
Polymer-ritonavir derivate nanomedicine with pH-sensitive activation possesses potent anti-tumor activity in vivo via inhibition of proteasome and STAT3 signaling.
Journal of Controlled Release. Roč. 332, APR 10 2021 (2021), s. 563-580. ISSN 0168-3659. E-ISSN 1873-4995
R&D Projects: GA ČR(CZ) GA19-05649S; GA MŠMT(CZ) LM2015040; GA MŠMT(CZ) ED1.1.00/02.0109
Research Infrastructure: CCP - 90040
Institutional support: RVO:61388971 ; RVO:61389013 ; RVO:68378050
Keywords : Ritonavir derivate * Polymer carrier * pH-controlled release * Antitumor activity * Proteasome inhibition * STAT3 signaling inhibition
OECD category: Microbiology; Polymer science (UMCH-V)
Impact factor: 11.467, year: 2021
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0168365921001267
Permanent Link: http://hdl.handle.net/11104/0320232 - 5.0481666 - ÚMCH 2019 RIV NL eng J - Journal Article
Studenovský, Martin - Sivák, Ladislav - Sedláček, Ondřej - Konefal, Rafal - Horková, Veronika - Etrych, Tomáš - Kovář, Marek - Říhová, Blanka - Šírová, Milada
Polymer nitric oxide donors potentiate the treatment of experimental solid tumours by increasing drug accumulation in the tumour tissue.
Journal of Controlled Release. Roč. 269, 10 January (2018), s. 214-224. ISSN 0168-3659. E-ISSN 1873-4995
R&D Projects: GA ČR(CZ) GA14-12742S; GA MZd(CZ) NV16-28600A; GA MŠMT(CZ) LQ1604; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61389013 ; RVO:61388971
Keywords : enhanced permeability and retention effect * nitric oxide donor * polymer-based cytotoxic drugs
OECD category: Polymer science; Microbiology (MBU-M)
Impact factor: 7.901, year: 2018
Permanent Link: http://hdl.handle.net/11104/0278289 - 6.0473557 - MBÚ 2018 RIV GB eng J - Journal Article
Sivák, Ladislav - Šubr, Vladimír - Tomala, Jakub - Říhová, Blanka - Strohalm, Jiří - Etrych, Tomáš - Kovář, Marek
Overcoming multidrug resistance via simultaneous delivery of cytostatic drug and P-glycoprotein inhibitor to cancer cells by HPMA copolymer conjugate.
Biomaterials. Roč. 115, JAN 2017 (2017), s. 65-80. ISSN 0142-9612. E-ISSN 1878-5905
R&D Projects: GA ČR(CZ) GAP301/12/1254; GA MŠMT(CZ) LQ1604; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61388971 ; RVO:61389013
Keywords : Multidrug resistance * P-glycoprotein * Doxorubicin
OECD category: Microbiology; Polymer science (UMCH-V)
Impact factor: 8.806, year: 2017
Permanent Link: http://hdl.handle.net/11104/0270692 - 7.0466229 - ÚMCH 2017 RIV NL eng J - Journal Article
Braunová, Alena - Kostka, Libor - Sivák, Ladislav - Cuchalová, Lucie - Hvězdová, Zuzana - Laga, Richard - Filippov, Sergey K. - Černoch, Peter - Pechar, Michal - Janoušková, Olga - Šírová, Milada - Etrych, Tomáš
Tumor-targeted micelle-forming block copolymers for overcoming of multidrug resistance.
Journal of Controlled Release. Roč. 245, 10 January (2017), s. 41-51. ISSN 0168-3659. E-ISSN 1873-4995
R&D Projects: GA MZd(CZ) NV16-28600A; GA MŠMT(CZ) LO1507; GA MŠMT(CZ) LQ1604; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61389013 ; RVO:61388971
Keywords : multidrug resistance * P-glycoprotein inhibitor * EPR effect
OECD category: Polymer science; Microbiology (MBU-M)
Impact factor: 7.877, year: 2017
Permanent Link: http://hdl.handle.net/11104/0264763 - 8.0459478 - ÚMCH 2017 RIV NL eng J - Journal Article
Koziolová, Eva - Janoušková, Olga - Cuchalová, Lucie - Hvězdová, Zuzana - Hraběta, J. - Eckschlager, T. - Sivák, Ladislav - Ulbrich, Karel - Etrych, Tomáš - Šubr, Vladimír
Overcoming multidrug resistance in Dox-resistant neuroblastoma cell lines via treatment with HPMA copolymer conjugates containing anthracyclines and P-gp inhibitors.
Journal of Controlled Release. Roč. 233, 10 July (2016), s. 136-146. ISSN 0168-3659. E-ISSN 1873-4995
R&D Projects: GA ČR(CZ) GAP301/12/1254; GA MŠMT(CZ) LO1507
Institutional support: RVO:61389013 ; RVO:61388971
Keywords : N-(2-hydroxypropyl)methacrylamide copolymers * multidrug resistance * P-glycoprotein inhibitors
Subject RIV: CD - Macromolecular Chemistry; FD - Oncology ; Hematology (MBU-M)
Impact factor: 7.786, year: 2016
Permanent Link: http://hdl.handle.net/11104/0259686 - 9.0431003 - ÚMCH 2015 RIV US eng J - Journal Article
Šubr, Vladimír - Sivák, Ladislav - Koziolová, Eva - Braunová, Alena - Pechar, Michal - Strohalm, Jiří - Kabešová, Martina - Říhová, Blanka - Ulbrich, Karel - Kovář, Marek
Synthesis of poly[N-(2-hydroxypropyl)methacrylamide] conjugates of inhibitors of the ABC transporter that overcome multidrug resistance in doxorubicin-resistant P388 cells in vitro.
Biomacromolecules. Roč. 15, č. 8 (2014), s. 3030-3043. ISSN 1525-7797. E-ISSN 1526-4602
R&D Projects: GA ČR GAP301/12/1254; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61389013 ; RVO:61388971
Keywords : N-(2-hydroxypropyl)methacrylamide copolymers * multidrug resistance * P-glycoprotein inhibitors
Subject RIV: CD - Macromolecular Chemistry; FD - Oncology ; Hematology (MBU-M)
Impact factor: 5.750, year: 2014
Permanent Link: http://hdl.handle.net/11104/0236142