Search results
- 1.0521898 - ÚACH 2020 FR eng A - Abstract
Nekvinda, Jan - Holub, Josef - Brynda, Jiří - Pospíšilová, Klára - Řezáčová, Pavlína - Grüner, Bohumír
Alkylsulfonamido carboranes: the isomer dependence observed in inhibitory activity towards Carbonic Anhydrase IX.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "O48".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
R&D Projects: GA ČR(CZ) GA15-05677S; GA ČR(CZ) GA18-27648S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : Carbonic Anhydrase
OECD category: Inorganic and nuclear chemistry; Biochemistry and molecular biology (UMG-J)
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306442 - 2.0520890 - ÚOCHB 2020 GB eng A - Abstract
Řezáčová, Pavlína - Kugler, Michael - Brynda, Jiří - Grüner, Bohumír - Hajdúch, M. - Nekvinda, Jan - Pospíšilová, Klára - Das, V. - Holub, Josef
Structure-assisted design of Carborane inhibitors of human Carbonic anhydrase IX.
Acta Crystallographica Section A-Foundation and Advances. Oxford Blackwell. Roč. 74, Suppl (2018), „e197“. ISSN 2053-2733. E-ISSN 2053-2733.
[European Crystallography Meeting /31./. 22.08.2018-27.08.2018, Oviedo]
R&D Projects: GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LO1304; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : anti-tumor agents * carborane inhibitors * Carbonic anhydrase IX
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Permanent Link: http://hdl.handle.net/11104/0305557 - 3.0484844 - ÚACH 2018 CN eng A - Abstract
Grüner, Bohumír - Holub, Josef - Nekvinda, Jan - Šícha, Václav - Štěpánková, J. - Hajdúch, M. - Pospíšilová, K. - Řezáčová, Pavlína - Brynda, Jiří
Rational Design and Synthesis of Carborane and Metallacarborane Sulfonamides as Inhibitors of Carbonic AnhydraseIX.
IMEBORON 16 Programme. Hong Kong: Chinese University of Hong Kong, 2017.
[IMEBORON: International Meeting on Boron Chemistry /16./. 09.07.2017-13.07.2017, Hong Kong]
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : carboranes
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UMG-J)
Permanent Link: http://hdl.handle.net/11104/0279972 - 4.0469489 - ÚACH 2017 RU eng A - Abstract
Grüner, Bohumír - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Štěpánková, J. - Hajdúch, M. - Řezáčová, Pavlína - Brynda, Jiří
Metallacarborane chemistry: Site-directed substitutions designed for specific inhibition activity towards CA-IX.
EuroBoron 7 : Book of Abstracts. Moscow: Federal Agency for Scientific Organisations, 2016. s. 20.
[International Congress on Neutron Capture Theraphy /17./. 02.10.2016-07.10.2016, Columbia]
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:61388980 ; RVO:61388963 ; RVO:68378050
Keywords : metallacarborane inhibitors
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UOCHB-X); FR - Pharmacology ; Medidal Chemistry (UMG-J)
http://icnct17.org/AbstractBook17.pdf
Permanent Link: http://hdl.handle.net/11104/0267272 - 5.0469464 - ÚACH 2017 US eng A - Abstract
Grüner, Bohumír - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Štěpánková, J. - Hajdúch, M. - Řezáčová, Pavlína - Brynda, Jiří
Carborane and metallacarborane inhibitors of Carbonic Anhydrase IX, compounds with possible double action.
The 17th International Congress on Neutron Capture Theraphy : Abstracts for presentation. Columbia: University of Missouri, 2016. s. 89.
[International Congress on Neutron Capture Theraphy /17./. 02.10.2016-07.10.2016, Columbia]
R&D Projects: GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028
Institutional support: RVO:61388980 ; RVO:61388963 ; RVO:68378050
Keywords : metallacarborane inhibitors
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UOCHB-X); FR - Pharmacology ; Medidal Chemistry (UMG-J)
http://icnct17.org/AbstractBook17.pdf
Permanent Link: http://hdl.handle.net/11104/0267255 - 6.0452109 - ÚOCHB 2016 GB eng A - Abstract
Koháryová, M. - Brynda, Jiří - Řezáčová, Pavlína - Kollárová, M.
Thioredoxin reductase from s. Coelicolor as a drug target.
FEBS Journal. Roč. 282, Suppl 1 (2015), s. 396. ISSN 1742-464X. E-ISSN 1742-4658.
[Congress of the Federation of European Biochemical Societies (FEBS) - The Biochemical Basis of Life /40./. 04.07.2015-09.07.2015, Berlin]
Institutional support: RVO:61388963 ; RVO:68378050
Keywords : thioredoxin reductase * protein structure * drugs
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0253136 - 7.0451586 - ÚACH 2016 GB eng A - Abstract
Grüner, Bohumír - Šícha, Václav - Holub, Josef - Nekvinda, Jan - Cígler, Petr - Štěpánková, P. - Mašek, V. - Matějíček, P. - Pokorná, Jana - Konvalinka, Jan - Hajduch, M. - Brynda, Jiří - Řezáčová, Pavlína
Metallacarboranes as hydrophobic pharmacophores; state of the art. Are these compounds worthy of further study?
Medical chemistry of boron compounds conference : oral presentation abstracts. Cambridge: Zing Conferences, 2015. s. 28.
[Medical chemistry of boron compounds conference. 04.10.2015-07.10.2015, Oropesa]
R&D Projects: GA ČR GA15-05677S
Institutional support: RVO:61388980 ; RVO:61388963 ; RVO:68378050
Keywords : metallacarboranes * pharmacophores
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UOCHB-X); EB - Genetics ; Molecular Biology (UMG-J)
Permanent Link: http://hdl.handle.net/11104/0252718 - 8.0443491 - ÚOCHB 2016 CZ eng A - Abstract
Kovářová, Zuzana - Hobizalová, Radka - Žebrakovská, Iva - Brynda, Jiří - Řezáčová, Pavlína - Horn, Martin - Mareš, Michael
Proteolytic system of blood-feeding ticks: An update on protein structures.
Materials Structure in Chemistry, Biology, Physics and Technology. Czech and Slovak Crystallographic Association. Roč. 22, č. 1 (2015), s. 43-44. ISSN 1211-5894.
[Discussions in Structural Molecular Biology. Annual Meeting of the Czech Society for Structural Biology /13./. 19.03.2015-21.03.2015, Nové Hrady]
Institutional support: RVO:61388963 ; RVO:68378050
Keywords : blood-feeding ticks * protein structure * proteolytic system
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0246297 - 9.0443483 - ÚOCHB 2016 CZ eng A - Abstract
Jílková, Adéla - Horn, Martin - Řezáčová, Pavlína - Marešová, Lucie - Fajtová, Pavla - Brynda, Jiří - Vondrášek, Jiří - McKerrow, J. H. - Caffrey, C. R. - Mareš, Michael
Activation route of the Schistosoma mansoni cathepsin B1 drug target.
Materials Structure in Chemistry, Biology, Physics and Technology. Czech and Slovak Crystallographic Association. Roč. 22, č. 1 (2015), s. 39. ISSN 1211-5894.
[Discussions in Structural Molecular Biology. Annual Meeting of the Czech Society for Structural Biology /13./. 19.03.2015-21.03.2015, Nové Hrady]
Institutional support: RVO:61388963 ; RVO:68378050
Keywords : Schistosoma mansoni * cathepsin B1 * sulfated polysaccharides
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0246295 - 10.0443405 - ÚOCHB 2016 CZ eng A - Abstract
Brynda, Jiří - Pachl, Petr - Šícha, Václav - Fábry, Milan - Grüner, Bohumír - Cígler, Petr - Řezáčová, Pavlína
Carborane-based inhibitors of carbonic anhydrases.
Materials Structure in Chemistry, Biology, Physics and Technology. Czech and Slovak Crystallographic Association. Roč. 22, č. 1 (2015), s. 3. ISSN 1211-5894.
[Discussions in Structural Molecular Biology. Annual Meeting of the Czech Society for Structural Biology /13./. 19.03.2015-21.03.2015, Nové Hrady]
R&D Projects: GA ČR GA15-05677S
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : carboranes * carbonic anhydrase
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0246131