Search results
- 1.0540277 - ÚMG 2021 RIV US eng J - Journal Article
Tykvart, J. - Navrátil, V. - Kugler, Michael - Šácha, P. - Schimer, J. - Hlaváčková, A. - Tenora, L. - Zemanová, J. - Dejmek, M. - Král, Vlastimil - Potáček, M. - Majer, P. - Jahn, U. - Brynda, Jiří - Řezáčová, Pavlína - Konvalinka, J.
Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA).
SLAS Discovery. Roč. 25, č. 9 (2020), s. 1026-1037. ISSN 2472-5552. E-ISSN 2472-5560
Institutional support: RVO:68378050
Keywords : high-throughput screening * carbonic anhydrase IX * drug discovery * DNA-linked inhibitor antibody assay
OECD category: Biochemistry and molecular biology
Impact factor: 2.918, year: 2020
Method of publishing: Limited access
https://journals.sagepub.com/doi/10.1177/2472555220918836
Permanent Link: http://hdl.handle.net/11104/0317971 - 2.0525049 - ÚOCHB 2021 RIV US eng J - Journal Article
Tykvart, Jan - Navrátil, Václav - Kugler, Michael - Šácha, Pavel - Schimer, Jiří - Hlavačková, Anna - Tenora, Lukáš - Zemanová, Jitka - Dejmek, Milan - Král, V. - Potáček, M. - Majer, Pavel - Jahn, Ullrich - Brynda, Jiří - Řezáčová, Pavlína - Konvalinka, Jan
Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA).
SLAS Discovery. Roč. 25, č. 9 (2020), s. 1026-1037. ISSN 2472-5552. E-ISSN 2472-5560
R&D Projects: GA ČR(CZ) GA19-10280S; GA ČR(CZ) GA17-14510S; GA MŠMT(CZ) EF16_019/0000729; GA MŠMT(CZ) LO1304
Institutional support: RVO:61388963
Keywords : high-throughput screening * carbonic anhydrase IX * drug discovery * DNA-linked inhibitor antibody assay
OECD category: Biochemistry and molecular biology
Impact factor: 2.918, year: 2020
Method of publishing: Limited access
https://journals.sagepub.com/doi/10.1177/2472555220918836
Permanent Link: http://hdl.handle.net/11104/0309265 - 3.0476344 - ÚEB 2018 RIV FR eng J - Journal Article
Řezníčková, Eva - Tenora, L. - Pospíšilová, Pavlína - Galeta, J. - Jorda, Radek - Berka, K. - Majer, Pavel - Potáček, M. - Kryštof, Vladimír
ALK5 kinase inhibitory activity and synthesis of 2,3,4-substituted 5,5-dimethyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles.
European Journal of Medicinal Chemistry. Roč. 127, FEB 15 (2017), s. 632-642. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA MŠMT(CZ) LO1204; GA ČR(CZ) GA15-15264S; GA MŠMT(CZ) LM2015047
Institutional support: RVO:61389030 ; RVO:61388963
Keywords : i-receptor kinase * beta signaling pathway * small-molecule inhibitor * tgf-beta * domain inhibitors * growth * fibrosis * cancer * potent * series * Transforming growth factor beta receptor I * Protein kinase * Inhibitor * Substituted pyrrolo[1,2-b]pyrazoles
OECD category: Pharmacology and pharmacy; Pharmacology and pharmacy (UOCHB-X)
Impact factor: 4.816, year: 2017
Permanent Link: http://hdl.handle.net/11104/0272863File Download Size Commentary Version Access 2017_Reznickova_EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY_632.pdf 4 1.3 MB Other open-access - 4.0468499 - ÚEB 2017 RIV US eng J - Journal Article
Tenora, L. - Galeta, J. - Řezníčková, Eva - Kryštof, Vladimír - Potáček, M.
Application of Pd-Catalyzed Cross-Coupling Reactions in the Synthesis of 5,5-Dimethy1-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles that Inhibit ALK5 Kinase.
Journal of Organic Chemistry. Roč. 81, č. 23 (2016), s. 11841-11856. ISSN 0022-3263. E-ISSN 1520-6904
R&D Projects: GA ČR(CZ) GA15-15264S
Institutional support: RVO:61389030
Keywords : c-h functionalization * pyridine n-oxides * receptor-type-i * direct arylation * tgf-beta * galunisertib ly2157299 * domain inhibitors * bond activation * growth * withasomnine
Subject RIV: FR - Pharmacology ; Medidal Chemistry
Impact factor: 4.849, year: 2016
Permanent Link: http://hdl.handle.net/11104/0266335File Download Size Commentary Version Access 2016_Tenora_JOURNAL OF ORGANIC CHEMISTRY_11841.pdf 0 2.4 MB Other open-access - 5.0192497 - UOCHB-X 960167 RIV US eng J - Journal Article
Dostál, J. - Bochořáková, H. - Táborská, E. - Slavík, J. - Potáček, M. - Buděšínský, Miloš - Hoffmann, E.
Structure of Sanguinarine Base.
Journal of Natural Products. Roč. 59, č. 6 (1996), s. 599-602. ISSN 0163-3864. E-ISSN 1520-6025
Impact factor: 1.243, year: 1996
Permanent Link: http://hdl.handle.net/11104/0088223