Search results
- 1.0573825 - FGÚ 2024 RIV GB eng J - Journal Article
Vojtěchová, Iveta - Tučková, K. - Jůza, R. - Stuchlík, Aleš - Kelemen, E. - Korábečný, J. - Soukup, O. - Petrásek, Tomáš
Dopaminergic and glutamatergic models of psychosis show differential sensitivity to aripiprazole and a novel experimental compound modulating D2/5-HT receptor activity.
Progress in Neuro-Psychopharmacology & Biological Psychiatry. Roč. 127, 20 Dec (2023), č. článku 110819. ISSN 0278-5846. E-ISSN 1878-4216
R&D Projects: GA MZd(CZ) NU22-04-00526
Institutional support: RVO:67985823
Keywords : schizophrenia * dizocilpine * amphetamine * antipsychotic * aripiprazole
OECD category: Neurosciences (including psychophysiology
Impact factor: 5.6, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.pnpbp.2023.110819
Permanent Link: https://hdl.handle.net/11104/0344177 - 2.0556370 - FGÚ 2023 RIV FR eng J - Journal Article
Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
OECD category: Pharmacology and pharmacy
Impact factor: 6.7, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2022.114193
Permanent Link: http://hdl.handle.net/11104/0330742 - 3.0546462 - FGÚ 2022 RIV CH eng J - Journal Article
Jůza, R. - Štefková, K. - Dehaen, W. - Randáková, Alena - Petrásek, T. - Vojtěchová, I. - Kobrlová, T. - Pulkrábková, L. - Mucková, L. - Mecava, M. - Prchal, L. - Mezeiová, E. - Musílek, K. - Soukup, O. - Korábečný, J.
Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D-2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
Biomolecules. Roč. 11, č. 9 (2021), č. článku 1262. E-ISSN 2218-273X
Institutional support: RVO:67985823
Keywords : aripiprazole * dopamine receptor * blood–brain barrier * molecular modeling studies * schizophrenia
OECD category: Pharmacology and pharmacy
Impact factor: 6.064, year: 2021
Method of publishing: Open access
https://www.mdpi.com/2218-273X/11/9/1262
Permanent Link: http://hdl.handle.net/11104/0322976