Search results

  1. 1.
    0546462 - FGÚ 2022 RIV CH eng J - Journal Article
    Jůza, R. - Štefková, K. - Dehaen, W. - Randáková, Alena - Petrásek, T. - Vojtěchová, I. - Kobrlová, T. - Pulkrábková, L. - Mucková, L. - Mecava, M. - Prchal, L. - Mezeiová, E. - Musílek, K. - Soukup, O. - Korábečný, J.
    Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D-2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
    Biomolecules. Roč. 11, č. 9 (2021), č. článku 1262. E-ISSN 2218-273X
    Institutional support: RVO:67985823
    Keywords : aripiprazole * dopamine receptor * blood–brain barrier * molecular modeling studies * schizophrenia
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/9/1262
    Permanent Link: http://hdl.handle.net/11104/0322976
     
     
  2. 2.
    0541833 - ÚEM 2022 RIV CH eng J - Journal Article
    Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
    Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
    Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
    R&D Projects: GA MZd(CZ) NU20-08-00296
    Research Infrastructure: e-INFRA CZ - 90140
    Institutional support: RVO:68378041
    Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/1/3
    Permanent Link: http://hdl.handle.net/11104/0319349
     
     
  3. 3.
    0541685 - FGÚ 2022 RIV CH eng J - Journal Article
    Konečný, J. - Misiachna, Anna - Hrabinová, M. - Pulkrábková, L. - Benková, M. - Prchal, L. - Kučera, T. - Kobrlová, T. - Finger, V. - Kolcheva, Marharyta - Kortus, Štěpán - Jun, D. - Valko, M. - Horák, Martin - Soukup, O. - Korábečný, J.
    Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists.
    Biomolecules. Roč. 11, č. 1 (2021), č. článku 3. E-ISSN 2218-273X
    Research Infrastructure: e-INFRA CZ - 90140
    Institutional support: RVO:67985823
    Keywords : acetylcholinesterase * Alzheimer´s disease * butyrylcholinesterase * fluorene * in vitro * in silico * multi-target directed ligands * N-methyl-d-aspartate receptor
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/1/3
    Permanent Link: http://hdl.handle.net/11104/0319216
     
     


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