Search results
- 1.0579099 - ÚMG 2024 RIV US eng J - Journal Article
Kutil, Z. - Mikešová, J. - Zessin, M. - Meleshin, M. - Nováková, Z. - Alquicer, Glenda - Kozikowski, A. - Sippl, W. - Bařinka, C. - Schutkowski, M.
Continuous Activity Assay for HDAC11 Enabling Reevaluation of HDAC Inhibitors.
ACS Omega. Roč. 4, č. 22 (2019), s. 19895-19904. ISSN 2470-1343. E-ISSN 2470-1343
R&D Projects: GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:68378050
Keywords : histone deacetylase inhibitors * sir2 family * posttranslational modifications * fluorescent-probe * peptide arrays * in-vitro * substrate-specificity * metabolic-regulation * fluorogenic probe * activity profiles
OECD category: Biochemistry and molecular biology
Impact factor: 2.870, year: 2019
Method of publishing: Open access
https://pubs.acs.org/doi/10.1021/acsomega.9b02808
Permanent Link: https://hdl.handle.net/11104/0347965 - 2.0571923 - BTÚ 2024 RIV CH eng J - Journal Article
Zessin, M. - Meleshin, M. - Hilscher, S. - Schiene-Fischer, C. - Bařinka, Cyril - Jung, M. - Schutkowski, M.
Continuous Fluorescent Sirtuin Activity Assay Based on Fatty Acylated Lysines.
International Journal of Molecular Sciences. Roč. 24, č. 8 (2023), č. článku 7416. E-ISSN 1422-0067
R&D Projects: GA ČR(CZ) GA21-31806S
Institutional support: RVO:86652036
Keywords : histone deacetylases * sirtuins * fluorescence quenching * sirtuin inhibitors
OECD category: Biochemistry and molecular biology
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1422-0067/24/8/7416
Permanent Link: https://hdl.handle.net/11104/0342895 - 3.0558797 - BTÚ 2023 RIV US eng J - Journal Article
Zessin, M. - Meleshin, M. - Praetorius, L. - Sippl, W. - Bařinka, Cyril - Schutkowski, M.
Uncovering Robust Delactoylase and Depyruvoylase Activities of HDAC Isoforms.
ACS Chemical Biology. Roč. 17, č. 6 (2022), s. 1364-1375. ISSN 1554-8929. E-ISSN 1554-8937
R&D Projects: GA ČR(CZ) GA21-31806S
Institutional support: RVO:86652036
Keywords : histone crotonylation * lysine * inhibitor * substrate
OECD category: Biochemistry and molecular biology
Impact factor: 4, year: 2022
Method of publishing: Limited access
https://pubs.acs.org/doi/10.1021/acschembio.1c00863
Permanent Link: https://hdl.handle.net/11104/0332584 - 4.0555060 - BTÚ 2023 RIV CH eng J - Journal Article
Ibrahim, H. - Abdelsalam, M. - Zeyn, Y. - Zessin, M. - Mustafa, A. - Fischer, M. - Zeyen, P. - Sun, P. - Buelbuel, E. - Vecchio, A. - Erdmann, F. - Schmidt, M. - Robaa, D. - Bařinka, Cyril - Romier, C. - Schutkowski, M. - Kraemer, O. - Sippl, W.
Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic Activity.
International Journal of Molecular Sciences. Roč. 23, č. 1 (2022), č. článku 369. E-ISSN 1422-0067
R&D Projects: GA ČR(CZ) GA21-31806S
Institutional support: RVO:86652036
Keywords : EFFICIENT GENERATION * EPIGENETIC THERAPY * AM1-BCC MODEL
OECD category: Biochemistry and molecular biology
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1422-0067/23/1/369
Permanent Link: http://hdl.handle.net/11104/0332121 - 5.0548916 - BTÚ 2022 RIV NL eng J - Journal Article
Zessin, M. - Meleshin, M. - Simic, Z. - Kalbas, D. - Arbach, M. - Gebhardt, P. - Melesina, J. - Liebscher, S. - Bordusa, F. - Sippl, W. - Bařinka, Cyril - Schutkowski, M.
Continuous Sirtuin/HDAC (histone deacetylase) activity assay using thioamides as PET (Photoinduced Electron Transfer)-based fluorescence quencher.
Bioorganic Chemistry. Roč. 117, DEC 2021 (2021). ISSN 0045-2068. E-ISSN 1090-2120
Institutional support: RVO:86652036
Keywords : Sirtuin assay * HDAC11 assay * Thioamide
OECD category: Organic chemistry
Impact factor: 5.307, year: 2021
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S0045206821008026?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0324965 - 6.0519605 - BTÚ 2020 RIV US eng J - Journal Article
Kutil, Zsofia - Mikesova, Jana - Zessin, M. - Meleshin, M. - Nováková, Zora - Alquicer, Glenda - Kozikowski, A. - Sippl, W. - Bařinka, Cyril - Schutkowski, M.
Continuous Activity Assay for HDAC11 Enabling Reevaluation of HDAC Inhibitors.
ACS Omega. Roč. 4, č. 22 (2019), s. 19895-19904. ISSN 2470-1343. E-ISSN 2470-1343
R&D Projects: GA ČR GA15-19640S; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:86652036
Keywords : histone deacetylase inhibitors * sir2 family * POSTTRANSLATIONAL MODIFICATIONS
OECD category: Biochemistry and molecular biology
Impact factor: 2.870, year: 2019
Method of publishing: Open access
https://pubs.acs.org/doi/10.1021/acsomega.9b02808
Permanent Link: http://hdl.handle.net/11104/0305194 - 7.0519596 - BTÚ 2020 RIV US eng J - Journal Article
Zessin, M. - Kutil, Zsofia - Meleshin, M. - Nováková, Zora - Ghazy, E. - Kalbas, D. - Marek, M. - Romier, Ch. - Sippl, W. - Bařinka, Cyril - Schutkowski, M.
One-Atom Substitution Enables Direct and Continuous Monitoring of Histone Deacylase Activity.
Biochemistry. Roč. 58, č. 48 (2019), s. 4777-4789. ISSN 0006-2960
R&D Projects: GA ČR GA15-19640S; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:86652036
Keywords : fluorescence quenching probes * epsilon-thioacetyl-lysine * deacetylase assay * sir2 family
OECD category: Biochemistry and molecular biology
Impact factor: 2.865, year: 2019
Method of publishing: Open access
https://pubs.acs.org/doi/10.1021/acs.biochem.9b00786
Permanent Link: http://hdl.handle.net/11104/0304590