Search results
- 1.0584241 - ÚEM 2025 RIV NL eng J - Journal Article
Mezeiová, E. - Prchal, L. - Hrabinová, M. - Mucková, L. - Pulkrabková, L. - Soukup, O. - Misiachna, Anna - Janoušek, J. - Fibigar, J. - Kučera, T. - Horák, Martin - Makhaeva, G.F. - Korabecný, J.
Morphing cholinesterase inhibitor amiridine into multipotent drugs for the
treatment of Alzheimer’s disease.
Biomedicine & Pharmacotherapy. Roč. 173, april. (2024), č. článku 116399. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
Keywords : amiridine * acetylcholinesterase * antioxidant capacity * butyrylcholinesterase * multi-target directed ligands * NMDA receptors
OECD category: Neurosciences (including psychophysiology
Impact factor: 7.5, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S075333222400283X?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0352201File Download Size Commentary Version Access Mezeirová 2024.pdf 3 1.7 MB Publisher’s postprint open-access - 2.0556370 - FGÚ 2023 RIV FR eng J - Journal Article
Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
OECD category: Pharmacology and pharmacy
Impact factor: 6.7, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2022.114193
Permanent Link: http://hdl.handle.net/11104/0330742 - 3.0546462 - FGÚ 2022 RIV CH eng J - Journal Article
Jůza, R. - Štefková, K. - Dehaen, W. - Randáková, Alena - Petrásek, T. - Vojtěchová, I. - Kobrlová, T. - Pulkrábková, L. - Mucková, L. - Mecava, M. - Prchal, L. - Mezeiová, E. - Musílek, K. - Soukup, O. - Korábečný, J.
Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D-2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
Biomolecules. Roč. 11, č. 9 (2021), č. článku 1262. E-ISSN 2218-273X
Institutional support: RVO:67985823
Keywords : aripiprazole * dopamine receptor * blood–brain barrier * molecular modeling studies * schizophrenia
OECD category: Pharmacology and pharmacy
Impact factor: 6.064, year: 2021
Method of publishing: Open access
https://www.mdpi.com/2218-273X/11/9/1262
Permanent Link: http://hdl.handle.net/11104/0322976 - 4.0504524 - FGÚ 2020 RIV FR eng J - Journal Article
Chalupová, K. - Korábečný, J. - Bartolini, M. - Monti, B. - Lamba, D. - Caliandro, R. - Pesaresi, A. - Brazzolotto, X. - Gastellier, A.-J. - Nachon, F. - Pejchal, J. - Jarošová, M. - Hepnarová, V. - Jun, D. - Hrabinová, M. - Doležal, R. - Zdarová Karasová, J. - Mžik, M. - Krištofíková, Z. - Misík, J. - Mucková, L. - Jošt, P. - Soukup, O. - Benková, M. - Setnička, V. - Habartová, L. - Chvojková, Markéta - Kletečková, Lenka - Valeš, Karel - Mezeiová, E. - Uliassi, E. - Vališ, M. - Nepovímová, E. - Bolognesi, M. L. - Kuča, K.
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease.
European Journal of Medicinal Chemistry. Roč. 168, Apr 15 (2019), s. 491-514. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : multi-target directed ligands * Alzheimer's disease * tacrine-tryptophan hybrids * acetylcholinesterase
OECD category: Neurosciences (including psychophysiology
Impact factor: 5.573, year: 2019
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2019.02.021
Permanent Link: http://hdl.handle.net/11104/0296178 - 5.0504272 - FGÚ 2020 RIV US eng J - Journal Article
Nepovímová, E. - Janočková, J. - Misík, J. - Kubík, Štěpán - Stuchlík, Aleš - Valeš, Karel - Korábečný, J. - Mezeiová, E. - Doležal, R. - Soukup, O. - Kobrlová, T. - Pham, N. L. - Nguyen, T. D. - Konečný, J. - Kuča, K.
Orexin supplementation in narcolepsy treatment: A review.
Medicinal Research Reviews. Roč. 39, č. 3 (2019), s. 961-975. ISSN 0198-6325. E-ISSN 1098-1128
R&D Projects: GA ČR(CZ) GA17-08596S
Institutional support: RVO:67985823
Keywords : cell transplantation * gene therapy * hypocretin * narcolepsy * orexin * orexin agonists
OECD category: Pharmacology and pharmacy
Impact factor: 9.300, year: 2019
Method of publishing: Limited access
https://doi.org/10.1002/med.21550
Permanent Link: http://hdl.handle.net/11104/0295940