Search results

  1. 1.
    0584241 - ÚEM 2025 RIV NL eng J - Journal Article
    Mezeiová, E. - Prchal, L. - Hrabinová, M. - Mucková, L. - Pulkrabková, L. - Soukup, O. - Misiachna, Anna - Janoušek, J. - Fibigar, J. - Kučera, T. - Horák, Martin - Makhaeva, G.F. - Korabecný, J.
    Morphing cholinesterase inhibitor amiridine into multipotent drugs for the
    treatment of Alzheimer’s disease.
    Biomedicine & Pharmacotherapy. Roč. 173, april. (2024), č. článku 116399. ISSN 0753-3322. E-ISSN 1950-6007
    R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) EH22_008/0004562
    Institutional support: RVO:68378041
    Keywords : amiridine * acetylcholinesterase * antioxidant capacity * butyrylcholinesterase * multi-target directed ligands * NMDA receptors
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 7.5, year: 2022
    Method of publishing: Open access
    https://www.sciencedirect.com/science/article/pii/S075333222400283X?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0352201
    FileDownloadSizeCommentaryVersionAccess
    Mezeirová 2024.pdf31.7 MBPublisher’s postprintopen-access
     
     
  2. 2.
    0556370 - FGÚ 2023 RIV FR eng J - Journal Article
    Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
    Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
    European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
    Institutional support: RVO:67985823
    Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.7, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1016/j.ejmech.2022.114193
    Permanent Link: http://hdl.handle.net/11104/0330742
     
     
  3. 3.
    0546462 - FGÚ 2022 RIV CH eng J - Journal Article
    Jůza, R. - Štefková, K. - Dehaen, W. - Randáková, Alena - Petrásek, T. - Vojtěchová, I. - Kobrlová, T. - Pulkrábková, L. - Mucková, L. - Mecava, M. - Prchal, L. - Mezeiová, E. - Musílek, K. - Soukup, O. - Korábečný, J.
    Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D-2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
    Biomolecules. Roč. 11, č. 9 (2021), č. článku 1262. E-ISSN 2218-273X
    Institutional support: RVO:67985823
    Keywords : aripiprazole * dopamine receptor * blood–brain barrier * molecular modeling studies * schizophrenia
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/9/1262
    Permanent Link: http://hdl.handle.net/11104/0322976
     
     
  4. 4.
    0504524 - FGÚ 2020 RIV FR eng J - Journal Article
    Chalupová, K. - Korábečný, J. - Bartolini, M. - Monti, B. - Lamba, D. - Caliandro, R. - Pesaresi, A. - Brazzolotto, X. - Gastellier, A.-J. - Nachon, F. - Pejchal, J. - Jarošová, M. - Hepnarová, V. - Jun, D. - Hrabinová, M. - Doležal, R. - Zdarová Karasová, J. - Mžik, M. - Krištofíková, Z. - Misík, J. - Mucková, L. - Jošt, P. - Soukup, O. - Benková, M. - Setnička, V. - Habartová, L. - Chvojková, Markéta - Kletečková, Lenka - Valeš, Karel - Mezeiová, E. - Uliassi, E. - Vališ, M. - Nepovímová, E. - Bolognesi, M. L. - Kuča, K.
    Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease.
    European Journal of Medicinal Chemistry. Roč. 168, Apr 15 (2019), s. 491-514. ISSN 0223-5234. E-ISSN 1768-3254
    Institutional support: RVO:67985823
    Keywords : multi-target directed ligands * Alzheimer's disease * tacrine-tryptophan hybrids * acetylcholinesterase
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 5.573, year: 2019
    Method of publishing: Limited access
    https://doi.org/10.1016/j.ejmech.2019.02.021
    Permanent Link: http://hdl.handle.net/11104/0296178
     
     
  5. 5.
    0504272 - FGÚ 2020 RIV US eng J - Journal Article
    Nepovímová, E. - Janočková, J. - Misík, J. - Kubík, Štěpán - Stuchlík, Aleš - Valeš, Karel - Korábečný, J. - Mezeiová, E. - Doležal, R. - Soukup, O. - Kobrlová, T. - Pham, N. L. - Nguyen, T. D. - Konečný, J. - Kuča, K.
    Orexin supplementation in narcolepsy treatment: A review.
    Medicinal Research Reviews. Roč. 39, č. 3 (2019), s. 961-975. ISSN 0198-6325. E-ISSN 1098-1128
    R&D Projects: GA ČR(CZ) GA17-08596S
    Institutional support: RVO:67985823
    Keywords : cell transplantation * gene therapy * hypocretin * narcolepsy * orexin * orexin agonists
    OECD category: Pharmacology and pharmacy
    Impact factor: 9.300, year: 2019
    Method of publishing: Limited access
    https://doi.org/10.1002/med.21550
    Permanent Link: http://hdl.handle.net/11104/0295940
     
     


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