Search results
- 1.0587109 - ÚEM 2025 RIV NL eng J - Journal Article
Chvojková, M. - Kolář, D. - Kováčová, K. - Čejková, L. - Misiachna, Anna - Hakenová, K. - Gorecki, L. - Horák, Martin - Korabecný, J. - Soukup, O. - Valeš, K.
Pro-cognitive effects of dual tacrine derivatives acting as cholinesterase inhibitors and NMDA receptor antagonists.
Biomedicine & Pharmacotherapy. Roč. 176, July (2024), č. článku 116821. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA MŠMT(CZ) LX22NPO5107; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
Keywords : acetylcholinesterase * alzheimer disease * cognition * polypharmacology * receptors * N-Methyl-D-Aspartate * tacrine
OECD category: Neurosciences (including psychophysiology
Impact factor: 7.5, year: 2022
https://www.sciencedirect.com/science/article/pii/S0753332224007054?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0354401File Download Size Commentary Version Access Chvojková 2024.pdf 0 1.8 MB Publisher’s postprint open-access - 2.0584241 - ÚEM 2025 RIV NL eng J - Journal Article
Mezeiová, E. - Prchal, L. - Hrabinová, M. - Mucková, L. - Pulkrabková, L. - Soukup, O. - Misiachna, Anna - Janoušek, J. - Fibigar, J. - Kučera, T. - Horák, Martin - Makhaeva, G.F. - Korabecný, J.
Morphing cholinesterase inhibitor amiridine into multipotent drugs for the
treatment of Alzheimer’s disease.
Biomedicine & Pharmacotherapy. Roč. 173, april. (2024), č. článku 116399. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
Keywords : amiridine * acetylcholinesterase * antioxidant capacity * butyrylcholinesterase * multi-target directed ligands * NMDA receptors
OECD category: Neurosciences (including psychophysiology
Impact factor: 7.5, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S075333222400283X?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0352201File Download Size Commentary Version Access Mezeirová 2024.pdf 3 1.7 MB Publisher’s postprint open-access - 3.0572189 - ÚEM 2024 RIV CH eng J - Journal Article
Svobodová, B. - Pulkrabová, L. - Pánek, D. - Misiachna, Anna - Kolcheva, Marharyta - Andrýs, R. - Handl, J. - Čapek, J. - Nývltová, P. - Roušar, T. - Prchal, L. - Hepnarová, V. - Hrabinová, M. - Mucková, L. - Tosnerová, D. - Karabanovich, G. - Finger, V. - Soukup, O. - Horák, Martin - Korabecný, J.
Structure-Guided Design of N-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer’s Disease.
International Journal of Molecular Sciences. Roč. 24, č. 11 (2023), č. článku 9124. ISSN 1661-6596
R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) LX22NPO5107
Institutional support: RVO:68378041
Keywords : Alzheimer’s disease * acetylcholinesterase * enzyme inhibition * N-methyl-d-aspartate receptor * multi-target directed ligands * monoamine oxidase A/B
OECD category: Pharmacology and pharmacy
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://doi.org/10.3390/ijms24119124
Permanent Link: https://hdl.handle.net/11104/0342960File Download Size Commentary Version Access Svobodová 2023.pdf 2 3.8 MB Publisher’s postprint open-access - 4.0492869 - ÚEM 2019 RIV NL eng J - Journal Article
Kaniaková, Martina - Kletečková, L. - Lichnerová, Katarina - Holubová, K. - Skřenková, Kristýna - Kořínek, M. - Krůšek, J. - Smejkalová, T. - Korabecný, J. - Valeš, K. - Soukup, O. - Horák, Martin
7-Methoxyderivative of tacrine is a 'foot-in-the-door' open-channel blocker of GluN1/GluN2 and GluN1/GluN3 NMDA receptors with neuroprotective activity in vivo.
Neuropharmacology. Roč. 140, sep 15 (2018), s. 217-232. ISSN 0028-3908. E-ISSN 1873-7064
Institutional support: RVO:68378041
Keywords : behavioural experiment * electrophysiology * glutamate receptor * human pathogenic mutation * ion channel * pharmacology
OECD category: Neurosciences (including psychophysiology
Impact factor: 4.367, year: 2018
Permanent Link: http://hdl.handle.net/11104/0294014