Search results
- 1.0544791 - ÚOCHB 2022 RIV FR eng J - Journal Article
Šimková, Adéla - Ormsby, Tereza - Sidej, Natan - Poštová Slavětínská, Lenka - Brynda, Jiří - Beranová, Jana - Šácha, Pavel - Majer, Pavel - Konvalinka, Jan
Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with α-ketoamide warheads.
European Journal of Medicinal Chemistry. Roč. 224, Nov 15 (2021), č. článku 113717. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA19-10280S; GA MZd(CZ) NV15-31379A; GA MŠMT(CZ) EF16_019/0000729; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963
Keywords : fibroblast activation protein * seprase * FAP inhibitor * serine protease inhibition * prolyl endopeptidase * α-Ketoamide inhibitor
OECD category: Medicinal chemistry
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113717
Permanent Link: http://hdl.handle.net/11104/0321598 - 2.0523934 - ÚOCHB 2021 RIV NL eng J - Journal Article
Šimková, Adéla - Bušek, P. - Šedo, A. - Konvalinka, Jan
Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications.
Biochimica Et Biophysica Acta-Proteins and Proteomics. Roč. 1868, č. 7 (2020), č. článku 140409. ISSN 1570-9639. E-ISSN 1878-1454
R&D Projects: GA MZd(CZ) NV15-31379A; GA MŠMT(CZ) LM2015064; GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : fibroblast activation protein * FAP inhibitors * FAP substrates * cancer tissue targeting * activity-based probes
OECD category: Biochemistry and molecular biology
Impact factor: 3.036, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/abs/pii/S1570963920300546
Permanent Link: http://hdl.handle.net/11104/0308229 - 3.0519252 - ÚOCHB 2020 RIV CH eng J - Journal Article
Beranová, Jana - Knedlík, Tomáš - Šimková, Adéla - Šubr, Vladimír - Kostka, Libor - Etrych, Tomáš - Šácha, Pavel - Konvalinka, Jan
Tris-(Nitrilotriacetic Acid)-Decorated Polymer Conjugates as Tools for Immobilization and Visualization of His-Tagged Proteins.
Catalysts. Roč. 9, č. 12 (2019), č. článku 1011. E-ISSN 2073-4344
R&D Projects: GA MŠMT(CZ) EF16_019/0000729; GA MPO(CZ) FV10490; GA MPO(CZ) FV10370; GA ČR(CZ) GA19-10280S; GA MŠMT(CZ) LQ1604; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61388963 ; RVO:61389013
Keywords : antibody mimetics * protein immobilization * His-tag * tris-nitrilotriacetic acid (tris-NTA) * iBodies * biocompatible polymers * N-(2-hydroxypropyl) methacrylamide (HPMA)
OECD category: Biochemistry and molecular biology; Polymer science (UMCH-V)
Impact factor: 3.520, year: 2019
Method of publishing: Open access
https://www.mdpi.com/2073-4344/9/12/1011
Permanent Link: http://hdl.handle.net/11104/0304263File Download Size Commentary Version Access 0519252.pdf 10 1.6 MB Publisher’s postprint open-access