Search results
- 1.0534773 - ÚVGZ 2021 RIV US eng J - Journal Article
Campos, L. E. - Garibotto, F. - Angelina, E. - Kos, J. - Gonec, T. - Marvanová, P. - Vettorazzi, M. - Oravec, Michal - Jendrzejewska, I. - Jampílek, J. - Alvarez, S. E. - Enriz, R. D.
Hydroxynaphthalenecarboxamides and substituted piperazinylpropandiols, two new series of BRAF inhibitors. A theoretical and experimental study.
Bioorganic Chemistry. Roč. 103, OCT (2020), č. článku 104145. ISSN 0045-2068. E-ISSN 1090-2120
R&D Projects: GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : raf inhibitors * mapk pathway * BRAF inhibitors * Melanoma * Molecular modeling * Cell viability * ERK phosphorylation
OECD category: Biochemistry and molecular biology
Impact factor: 5.275, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0045206820314425?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0312945 - 2.0483037 - ÚVGZ 2019 RIV CH eng J - Journal Article
Padrtova, T. - Marvanová, P. - Odehnalová, K. - Kubínová, R. - Parravicini, V. - Garro, A. - Enriz, R. D. - Humpa, O. - Oravec, Michal - Mokrý, P.
Synthesis, analysis, cholinesterase-inhibiting activity and molecular modelling studies of 3-(dialkylamino)-2-hydroxypropyl 4-[(alkoxy-carbonyl)amino]benzoates and their quaternary ammonium salts.
Molecules. Roč. 22, č. 12 (2017), č. článku 2048. E-ISSN 1420-3049
R&D Projects: GA MŠMT(CZ) LM2015061; GA MŠMT(CZ) LO1415; GA MŠMT(CZ) EF16_013/0001609
Research Infrastructure: CzeCOS II - 90061
Institutional support: RVO:86652079
Keywords : Acetylcholinesterase * Arylcarbonyloxyaminopropanols * Butyrylcholinesterase * Quaternary ammonium salts * Tertiary amines
OECD category: Biochemistry and molecular biology
Impact factor: 3.098, year: 2017
Permanent Link: http://hdl.handle.net/11104/0278463 - 3.0477421 - ÚIACH 2018 RIV FR eng J - Journal Article
Vettorazzi, M. - Angelina, E. - Lima, S. - Goněc, T. - Otevřel, J. - Marvanová, P. - Padrtová, T. - Mokrý, P. - Bobáľ, P. - Acosta, L. M. - Palma, A. - Cobo, J. - Bobálová, Janette - Csollei, J. - Malik, I. - Alvarez, S. - Spiegel, S. - Jampílek, J. - Enriz, R. D.
An integrative study to identify novel scaffolds for sphingosine kinase 1 inhibitors.
European Journal of Medicinal Chemistry. Roč. 139, OCT (2017), s. 461-481. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:68081715
Keywords : sphingosine kinase 1 inhibitors * bioassays * molecular modelling * virtual screening
OECD category: Analytical chemistry
Impact factor: 4.816, year: 2017
Permanent Link: http://hdl.handle.net/11104/0273776File Download Size Commentary Version Access 0477421_IR.pdf 1 4.9 MB Other require