Search results
- 1.0545890 - ÚEB 2022 RIV GB eng J - Journal Article
Maková, B. - Mik, V. - Lišková, B. - Gonzalez, G. - Vítek, D. - Medvedíková, M. - Monfort, B. - Ručilová, V. - Kadlecová, A. - Khirsariya, P. - Gándara Barreiro, Z. - Havlíček, Libor - Zatloukal, M. - Soural, M. - Paruch, K. - D'Autréaux, B. - Hajdúch, M. - Strnad, M. - Voller, Jiří
Cytoprotective activities of kinetin purine isosteres.
Bioorganic & Medicinal Chemistry. Roč. 33, MAR 1 (2021), č. článku 115993. ISSN 0968-0896. E-ISSN 1464-3391
Institutional support: RVO:61389030
Keywords : bioisostery – Friedreich́s ataxia * Cytokinin * Kinetin * Mitoprotection – familial dysautonomia * Neuroprotection
OECD category: Pharmacology and pharmacy
Impact factor: 3.461, year: 2021
Method of publishing: Open access
http://doi.org/10.1016/j.bmc.2021.115993
Permanent Link: http://hdl.handle.net/11104/0322516File Download Size Commentary Version Access 2021_Makova_BIOORGANIC & MEDICINAL CHEMISTRY_115993.pdf 1 1.1 MB Other open-access - 2.0541275 - MBÚ 2021 RIV CZ eng J - Journal Article
Jourová, L. - Lišková, B. - Lněničková, K. - Zemanová, N. - Anzenbacher, P. - Hermanová, Petra - Hudcovic, Tomáš - Kozáková, Hana - Anzenbacherová, E.
Presence or Absence of Microbiome Modulates the Response of Mice Organism to Administered Drug Nabumetone.
Physiological Research. Roč. 69, Suppl 4 (2020), s. 583-594. ISSN 0862-8408. E-ISSN 1802-9973
R&D Projects: GA ČR(CZ) GA19-08294S
Institutional support: RVO:61388971
Keywords : Gut microbiome * Cytochromes P450 * Germ-free mice * Nabumetone * Metabolism of drugs
OECD category: Immunology
Impact factor: 1.881, year: 2020
Method of publishing: Open access
https://www.biomed.cas.cz/physiolres/pdf/2020/69_S583.pdf
Permanent Link: http://hdl.handle.net/11104/0318861 - 3.0536679 - ÚMCH 2021 RIV US eng J - Journal Article
Švec, Pavel - Nový, Z. - Kučka, Jan - Petřík, M. - Sedláček, Ondřej - Kuchař, M. - Lišková, B. - Medvedíková, M. - Kolouchová, Kristýna - Groborz, Ondřej - Loukotová, Lenka - Konefal, Rafal - Hajdúch, M. - Hrubý, Martin
Iodinated choline transport-targeted tracers.
Journal of Medicinal Chemistry. Roč. 63, č. 24 (2020), s. 15960-15978. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GA19-01602S; GA MZd(CZ) NV16-30544A; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61389013
Keywords : choline transport * radioiodination * fluorocholine
OECD category: Polymer science
Impact factor: 7.446, year: 2020
Method of publishing: Limited access
https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01710
Permanent Link: http://hdl.handle.net/11104/0315705 - 4.0532766 - ÚOCHB 2021 RIV DE eng J - Journal Article
Veselovská, Lucia - Kudlová, N. - Gurská, S. - Lišková, B. - Medvedíková, M. - Hodek, Ondřej - Tloušťová, Eva - Milisavljevič, Nemanja - Tichý, Michal - Perlíková, Pavla - Mertlíková-Kaiserová, Helena - Trylčová, Jana - Pohl, Radek - Klepetářová, Blanka - Džubák, P. - Hajdúch, M. - Hocek, Michal
Synthesis and Cytotoxic and Antiviral Activity Profiling of All-Four Isomeric Series of Pyrido-Fused 7-Deazapurine Ribonucleosides.
Chemistry - A European Journal. Roč. 26, č. 57 (2020), s. 13002-13015. ISSN 0947-6539. E-ISSN 1521-3765
R&D Projects: GA ČR(CZ) GA19-08124S; GA MZd(CZ) NV15-31984A; GA MŠMT(CZ) LM2015064
Grant - others:AV ČR(CZ) AP1501
Program: Akademická prémie - Praemium Academiae
Institutional support: RVO:61388963
Keywords : antitumor agents * antiviral agents * drug discovery * phosphorylation * ribonucleosides
OECD category: Organic chemistry
Impact factor: 5.236, year: 2020
Method of publishing: Limited access
https://doi.org/10.1002/chem.202001124
Permanent Link: http://hdl.handle.net/11104/0311179 - 5.0531266 - ÚMG 2021 RIV FR eng J - Journal Article
Dvořanová, J. - Kugler, Michael - Holub, J. - Šícha, V. - Das, V. - Nekvinda, J. - El Anwar, S. - Havránek, M. - Pospíšilová, K. - Fábry, Milan - Král, Vlastimil - Medvědiková, M. - Matějková, S. - Lišková, B. - Gurská, S. - Dzubak, P. - Brynda, Jiří - Hajduch, M. - Gruner, B. - Řezáčová, P.
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
European Journal of Medicinal Chemistry. Roč. 200, August (2020), č. článku 112460. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:68378050
Keywords : Anti-tumor agents * Carbonic anhydrase IX * Carboranes * Dicarbollide * Enzyme inhibitors * Drug penetration * Multicellular spheroids
OECD category: Medicinal chemistry
Impact factor: 6.514, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/abs/pii/S0223523420304311?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0309958 - 6.0524603 - ÚOCHB 2021 RIV FR eng J - Journal Article
Dvořanová, J. - Kugler, Michael - Holub, Josef - Šícha, Václav - Das, V. - Nekvinda, Jan - El Anwar, Suzan - Havránek, M. - Pospíšilová, Klára - Fábry, M. - Král, V. - Medvedíková, M. - Matějková, Stanislava - Lišková, B. - Gurská, S. - Džubák, P. - Brynda, J. - Hajdúch, M. - Grüner, Bohumír - Řezáčová, Pavlína
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
European Journal of Medicinal Chemistry. Roč. 200, Aug 15 (2020), č. článku 112460. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA18-27648S; GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LM2015064
Grant - others:AV ČR(CZ) L200321851
Program: Program podpory perspektivníchlidských zdrojů - postdoktorandů
Institutional support: RVO:61388963 ; RVO:61388980
Keywords : anti-tumor agents * carbonic anhydrase IX * carboranes * dicarbollide * enzyme inhibitors * drug penetration * multicellular spheroids
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Impact factor: 6.514, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0223523420304311?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0308946 - 7.0511473 - ÚACH 2020 RIV US eng J - Journal Article
Grüner, Bohumír - Brynda, Jiří - Das, V. - Šícha, Václav - Štěpánková, J. - Nekvinda, Jan - Holub, Josef - Pospíšilová, B. - Fábry, Milan - Pachl, P. - Král, Vlastimil - Kugler, M. - Mašek, V. - Medvědiková, M. - Matějková, S. - Nová, A. - Lišková, B. - Gurská, S. - Džubák, P. - Hajdúch, M. - Řezáčová, Pavlína
Metallacarborane sulfamides: Unconventional, specific, and highly selective inhibitors of carbonic anhydrase IX.
Journal of Medicinal Chemistry. Roč. 62, č. 21 (2019), s. 9560-9575. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GA15-05677S; GA ČR(CZ) GA18-27648S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : Anti-tumor agents * Carbonic anhydrase IX * Cobaltacarborane inhibitors * Drug penetration * Multicellular spheroids
OECD category: Inorganic and nuclear chemistry; Medicinal chemistry (UMG-J)
Impact factor: 6.205, year: 2019
Method of publishing: Limited access
https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.9b00945
Permanent Link: http://hdl.handle.net/11104/0302697 - 8.0511423 - ÚOCHB 2020 RIV US eng J - Journal Article
Grüner, B. - Brynda, Jiří - Das, V. - Šícha, V. - Štěpánková, J. - Nekvinda, J. - Holub, J. - Pospíšilová, Klára - Fábry, M. - Pachl, Petr - Král, V. - Kugler, Michael - Mašek, V. - Medvedíková, M. - Matějková, Stanislava - Nová, A. - Lišková, B. - Gurská, S. - Džubák, P. - Hajdúch, M. - Řezáčová, Pavlína
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX.
Journal of Medicinal Chemistry. Roč. 62, č. 21 (2019), s. 9560-9575. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963
Keywords : cobalt bis(1,2-dicarbollide) * carborane complexes * medicinal chemistry
OECD category: Biochemistry and molecular biology
Impact factor: 6.205, year: 2019
Method of publishing: Limited access
https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.9b00945
Permanent Link: http://hdl.handle.net/11104/0301695 - 9.0498520 - ÚOCHB 2019 RIV US eng J - Journal Article
Tokarenko, Anna - Lišková, B. - Smolen, Sabina - Táborská, N. - Tichý, Michal - Gurská, S. - Perlíková, Pavla - Frydrych, I. - Tloušťová, Eva - Znojek, P. - Mertlíková-Kaiserová, Helena - Poštová Slavětínská, Lenka - Pohl, Radek - Klepetářová, Blanka - Khalid, N. U. A. - Wenren, Y. - Laposa, R. R. - Džubák, P. - Hajdúch, M. - Hocek, Michal
Synthesis and Cytotoxic and Antiviral Profiling of Pyrrolo- and Furo-Fused 7-Deazapurine Ribonucleosides.
Journal of Medicinal Chemistry. Roč. 61, č. 20 (2018), s. 9347-9359. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR(CZ) GA16-00178S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LO1304; GA MŠMT(CZ) LM2015064
Grant - others:AV ČR(CZ) AP1501
Program: Akademická prémie - Praemium Academiae
Institutional support: RVO:61388963
Keywords : hepatitis C virus * adenosine kinase inhibitors * mitochondrial RNA polymerase
OECD category: Organic chemistry
Impact factor: 6.054, year: 2018
https://pubs.acs.org/doi/full/10.1021/acs.jmedchem.8b01258
Permanent Link: http://hdl.handle.net/11104/0291128File Download Size Commentary Version Access 0498520.pdf 9 1.9 MB Publisher’s postprint open-access - 10.0480502 - MBÚ 2018 RIV NL eng J - Journal Article
Jourová, L. - Anzenbacher, P. - Lišková, B. - Matušková, Z. - Hermanová, Petra - Hudcovic, Tomáš - Kozáková, Hana - Hrnčířová, Lucia - Anzenbacherová, E.
Colonization by non-pathogenic bacteria alters mRNA expression of cytochromes P450 in originally germ-free mice.
Folia Microbiologica. Roč. 62, č. 6 (2017), s. 463-469. ISSN 0015-5632. E-ISSN 1874-9356
R&D Projects: GA ČR(CZ) GAP303/12/0535; GA ČR GA15-07268S
Institutional support: RVO:61388971
Keywords : HUMAN GUT MICROBIOTA * GENE-EXPRESSION * NISSLE 1917
OECD category: Microbiology
Impact factor: 1.311, year: 2017
Permanent Link: http://hdl.handle.net/11104/0276349