Search results
- 1.0587109 - ÚEM 2025 RIV NL eng J - Journal Article
Chvojková, M. - Kolář, D. - Kováčová, K. - Čejková, L. - Misiachna, Anna - Hakenová, K. - Gorecki, L. - Horák, Martin - Korabecný, J. - Soukup, O. - Valeš, K.
Pro-cognitive effects of dual tacrine derivatives acting as cholinesterase inhibitors and NMDA receptor antagonists.
Biomedicine & Pharmacotherapy. Roč. 176, July (2024), č. článku 116821. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA MŠMT(CZ) LX22NPO5107; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
Keywords : acetylcholinesterase * alzheimer disease * cognition * polypharmacology * receptors * N-Methyl-D-Aspartate * tacrine
OECD category: Neurosciences (including psychophysiology
Impact factor: 7.5, year: 2022
https://www.sciencedirect.com/science/article/pii/S0753332224007054?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0354401File Download Size Commentary Version Access Chvojková 2024.pdf 0 1.8 MB Publisher’s postprint open-access - 2.0582133 - ÚEM 2025 RIV NL eng J - Journal Article
Misiachna, Anna - Svobodová, B. - Netolický, Jakub - Chvojková, M. - Kletečková, L. - Prchal, L. - Novák, M. - Hrabinová, M. - Kučera, T. - Mucková, L. - Moravcová, Z. - Karasová-Ždárová, J. - Pejchal, J. - Blažek, F. - Maliňák, D. - Hakenová, K. - Hrčka Krausová, Barbora - Kolcheva, Marharyta - Ladislav, Marek - Korábečný, J. - Pahnke, J. - Valeš, K. - Horák, Martin - Soukup, O.
Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition.
European Journal of Medicinal Chemistry. Roč. 266, feb. (2024), č. článku 116130. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA TA ČR(CZ) TO01000078; GA MŠMT(CZ) EH22_008/0004562
Institutional support: RVO:68378041
OECD category: Neurosciences (including psychophysiology
Impact factor: 6.7, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S0223523424000102?via%3Dihub https://doi.org/10.5281/zenodo.10949371 https://doi.org/10.2139/ssrn.4658299
Permanent Link: https://hdl.handle.net/11104/0350209File Download Size Commentary Version Access Misiachna příloha 2024.pdf 1 9.8 MB Other open-access Misiachna 2024.pdf 4 5 MB Publisher’s postprint open-access - 3.0579544 - FGÚ 2024 RIV GB eng J - Journal Article
Kolář, D. - Krajčovič, Branislav - Kletečková, L. - Kunčická, Daniela - Valeš, K. - Brožka, Hana
Review: Genes Involved in Mitochondrial Physiology Within 22q11.2 Deleted Region and Their Relevance to Schizophrenia.
Schizophrenia Bulletin. Roč. 49, č. 6 (2023), s. 1637-1653. ISSN 0586-7614. E-ISSN 1745-1701
R&D Projects: GA ČR(CZ) GA22-15096S; GA MZd(CZ) NU22J-04-00061
Institutional support: RVO:67985823
Keywords : energy metabolism * 22q11.2DS * schizophrenia * mitochondria
OECD category: Neurosciences (including psychophysiology
Impact factor: 6.6, year: 2022
Method of publishing: Limited access
https://doi.org/10.1093/schbul/sbad066
Permanent Link: https://hdl.handle.net/11104/0348361 - 4.0578778 - ÚMG 2024 RIV NL eng J - Journal Article
Chrienová, Z. - Ryšánek, David - Novák, Josef - Vašicová, Pavla - Oleksak, P. - Andrýs, R. - Skarka, A. - Dumanovic, J. - Milovanovic, Z. - Jacevic, V. - Chvojková, M. - Holubová, K. - Valeš, K. - Skoupilová, V. - Valko, M. - Jomová, K. - Alomar, S. Y. - Botelho, F. D. - Franca, T. C. C. - Kuča, K. - Hodný, Zdeněk - Nepovimova, E.
Frentizole derivatives with mTOR inhibiting and senomorphic properties.
Biomedicine & Pharmacotherapy. Roč. 167, Nov (2023), č. článku 115600. ISSN 0753-3322. E-ISSN 1950-6007
R&D Projects: GA MŠMT LX22NPO5102
Institutional support: RVO:68378050
Keywords : cellular senescence * life-span * alzheimers-disease * mitochondrial dysfunction * rapamycin * cells * growth * expression * longevity * apoptosis * Frentizole * abad * mtor * Cellular senescence * Aging
OECD category: Biochemistry and molecular biology
Impact factor: 7.5, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S0753332223013987?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0347694File Download Size Commentary Version Access Chrienova_2023_CC BY.pdf 3 992.3 KB Publisher’s postprint open-access - 5.0551558 - ÚEM 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
Institutional support: RVO:68378041
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
OECD category: Medicinal chemistry
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0326821 - 6.0545470 - FGÚ 2022 RIV IE eng J - Journal Article
Kolář, D. - Kletečková, L. - Brožka, Hana - Valeš, K.
Mini-review: Brain energy metabolism and its role in animal models of depression, bipolar disorder, schizophrenia and autism.
Neuroscience Letters. Roč. 760, Aug 24 (2021), č. článku 136003. ISSN 0304-3940. E-ISSN 1872-7972
R&D Projects: GA MZd(CZ) EF16_025/0007444; GA ČR(CZ) GA18-09296S
Institutional support: RVO:67985823
Keywords : schizophrenia * autism * depression * bipolar * mitochondria * metabolism
OECD category: Neurosciences (including psychophysiology
Impact factor: 3.197, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.neulet.2021.136003
Permanent Link: http://hdl.handle.net/11104/0322157 - 7.0543492 - ÚEM 2022 RIV US eng J - Journal Article
Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
R&D Projects: GA ČR(CZ) GA20-12047S
Institutional support: RVO:68378041
Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
OECD category: Pharmacology and pharmacy
Impact factor: 6.100, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bcp.2021.114460
Permanent Link: http://hdl.handle.net/11104/0320802 - 8.0542659 - FGÚ 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
OECD category: Pharmacology and pharmacy
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0320032 - 9.0524502 - ÚFE 2021 RIV US eng J - Journal Article
Krištofíková, Z. - Špringer, Tomáš - Gedeonová, Erika - Hofmannová, A. - Říčný, J. - Hromádková, L. - Vyhnálek, M. - Laczó, J. - Nikolai, T. - Hort, J. - Petrásek, Tomáš - Stuchlík, Aleš - Valeš, K. - Klaschka, Jan - Homola, Jiří
Interactions of 17β-Hydroxysteroid Dehydrogenase Type 10 and Cyclophilin D in Alzheimer's Disease.
Neurochemical Research. Roč. 45, č. 4 (2020), s. 915-927. ISSN 0364-3190. E-ISSN 1573-6903
R&D Projects: GA MZd(CZ) NV16-27611A
Institutional support: RVO:67985882 ; RVO:67985823 ; RVO:67985807
Keywords : Cerebrospinal fluid * Mitochondrial matrix proteins * Amyloid β * Transgenic rat model * Alzheimer's disease * Frontotemporal lobar degeneration
OECD category: Biochemistry and molecular biology; Biochemistry and molecular biology (FGU-C); Biochemistry and molecular biology (UIVT-O)
Impact factor: 3.996, year: 2020
Method of publishing: Open access
https://link.springer.com/content/pdf/10.1007/s11064-020-02970-y.pdf
Permanent Link: http://hdl.handle.net/11104/0308856File Download Size Commentary Version Access UFE 0524502.pdf 5 1.4 MB Other require - 10.0518489 - ÚEM 2020 RIV NL eng J - Journal Article
Kaniaková, Martina - Nepovímová, E. - Kletečková, L. - Skřenková, Kristýna - Holubová, K. - Chrienová, Z. - Hepnarová, V. - Kučera, T. - Kobrlová, T. - Valeš, K. - Korábečný, J. - Soukup, O. - Horák, Martin
Combination of Memantine and 6-Chlorotacrine as Novel Multi-Target Compound against Alzheimer's Disease.
Current Alzheimer Research. Roč. 16, č. 9 (2019), s. 821-833. ISSN 1567-2050. E-ISSN 1875-5828
Institutional support: RVO:68378041
Keywords : 6-Chlorotacrine * memantine * acetylcholinesterase
OECD category: Neurosciences (including psychophysiology
Impact factor: 3.047, year: 2019
Method of publishing: Limited access
http://www.eurekaselect.com/170309/article
Permanent Link: http://hdl.handle.net/11104/0303623