Search results

  1. 1.
    0492895 - ÚOCHB 2019 RIV US eng J - Journal Article
    Neburková, Jitka - Sedlák, František - Žáčková Suchanová, J. - Kostka, Libor - Šácha, Pavel - Šubr, Vladimír - Etrych, Tomáš - Šimon, Petr - Bařinková, Jitka - Kryštůfek, Robin - Španielová, Hana - Forstová, J. - Konvalinka, Jan - Cígler, Petr
    Inhibitor-GCPII Interaction: Selective and Robust System for Targeting Cancer Cells with Structurally Diverse Nanoparticles.
    Molecular Pharmaceutics. Roč. 15, č. 8 (2018), s. 2932-2945. ISSN 1543-8384. E-ISSN 1543-8392
    R&D Projects: GA ČR(CZ) GA16-16336S; GA ČR(CZ) GA16-02938S; GA MŠMT LO1302
    Institutional support: RVO:61388963 ; RVO:61389013
    Keywords : GCPII * PSMA * inhibitor * click chemistry * targeting * cell * nanodiamond
    OECD category: Biochemistry and molecular biology; Polymer science (UMCH-V)
    Impact factor: 4.396, year: 2018
    Permanent Link: http://hdl.handle.net/11104/0286398
     
     
  2. 2.
    0445391 - ÚOCHB 2016 RIV US eng J - Journal Article
    Tykvart, Jan - Schimer, Jiří - Jančařík, Andrej - Bařinková, Jitka - Navrátil, Václav - Starková, Jana - Šrámková, Karolína - Konvalinka, Jan - Majer, Pavel - Šácha, Pavel
    Design of Highly Potent Urea-Based, Exosite-Binding Inhibitors Selective for Glutamate Carboxypeptidase II.
    Journal of Medicinal Chemistry. Roč. 58, č. 10 (2015), s. 4357-4363. ISSN 0022-2623. E-ISSN 1520-4804
    R&D Projects: GA ČR GBP208/12/G016; GA MŠMT LO1302
    Institutional support: RVO:61388963
    Keywords : GCPII selective inhibitors * GCPIII * GCPII
    Subject RIV: CE - Biochemistry
    Impact factor: 5.589, year: 2015
    Permanent Link: http://hdl.handle.net/11104/0247685
     
     
  3. 3.
    0431499 - ÚOCHB 2015 RIV GB eng J - Journal Article
    Tykvart, Jan - Schimer, Jiří - Bařinková, Jitka - Pachl, Petr - Poštová Slavětínská, Lenka - Majer, Pavel - Konvalinka, Jan - Šácha, Pavel
    Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery.
    Bioorganic & Medicinal Chemistry. Roč. 22, č. 15 (2014), s. 4099-4108. ISSN 0968-0896. E-ISSN 1464-3391
    R&D Projects: GA ČR GBP208/12/G016
    Grant - others:OPPK(CZ) CZ.2.16/3.1.00/24016
    Institutional support: RVO:61388963
    Keywords : GCPII * PSMA * structure-aided drug design * specific drug targeting
    Subject RIV: CE - Biochemistry
    Impact factor: 2.793, year: 2014
    Permanent Link: http://hdl.handle.net/11104/0236131
     
     


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