Search results
- 1.0490659 - ÚOCHB 2019 RIV US eng J - Journal Article
Zimmermann, S. C. - Tichý, Tomáš - Vávra, Jan - Dash, R. P. - Slusher, C. E. - Gadiano, A. J. - Wu, Y. - Jančařík, Andrej - Tenora, Lukáš - Monincová, Lenka - Prchalová, E. - Riggins, G. J. - Majer, Pavel - Slusher, B. S. - Rais, R.
N-Substituted Prodrugs of Mebendazole Provide Improved Aqueous Solubility and Oral Bioavailability in Mice and Dogs.
Journal of Medicinal Chemistry. Roč. 61, č. 9 (2018), s. 3918-3929. ISSN 0022-2623. E-ISSN 1520-4804
Institutional support: RVO:61388963
Keywords : anthelmintic drug mebendazole * water soluble prodrugs * in vivo
OECD category: Organic chemistry
Impact factor: 6.054, year: 2018
Permanent Link: http://hdl.handle.net/11104/0284815 - 2.0480326 - ÚOCHB 2018 RIV US eng J - Journal Article
Rais, R. - Vávra, Jan - Tichý, Tomáš - Dash, R. P. - Gadiano, A. J. - Tenora, Lukáš - Monincová, Lenka - Bařinka, Cyril - Alt, J. - Zimmermann, S. C. - Slusher, C. E. - Wu, Y. - Wozniak, K. - Majer, Pavel - Tsukamoto, T. - Slusher, B. S.
Discovery of a para-Acetoxy-benzyl Ester Prodrug of a Hydroxamate-Based Glutamate Carboxypeptidase II Inhibitor as Oral Therapy for Neuropathic Pain.
Journal of Medicinal Chemistry. Roč. 60, č. 18 (2017), s. 7799-7809. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA MŠMT(CZ) LM2015043; GA MŠMT(CZ) ED1.1.00/02.0109
Institutional support: RVO:61388963 ; RVO:86652036
Keywords : linked acidic dipeptidase * peripheral mononeuropathy * biological activity
OECD category: Organic chemistry; Organic chemistry (BTO-N)
Impact factor: 6.253, year: 2017
Permanent Link: http://hdl.handle.net/11104/0276130 - 3.0427622 - ÚOCHB 2015 RIV US eng J - Journal Article
Ferraris, D. V. - Majer, Pavel - Ni, C. - Slusher, C. E. - Rais, R. - Wu, Y. - Wozniak, K. M. - Alt, J. - Rojas, C. - Slusher, B. S. - Tsukamoto, T.
delta-Thiolactones as Prodrugs of Thiol-Based Glutamate Carboxypeptidase II (GCPII) Inhibitors.
Journal of Medicinal Chemistry. Roč. 57, č. 1 (2014), s. 243-247. ISSN 0022-2623. E-ISSN 1520-4804
Institutional support: RVO:61388963
Keywords : pharmacokinetics * discovery * disorders * diagnosis * pain
Subject RIV: CC - Organic Chemistry
Impact factor: 5.447, year: 2014
Permanent Link: http://hdl.handle.net/11104/0233159