Search results
- 1.0568179 - ÚOCHB 2023 GB eng A - Abstract
Brynda, Jiří - Kugler, Michael - Nekvinda, Jan - Holub, Josef - El Anwar, Suzan - Das, V. - Šícha, Václav - Pospíšilová, Klára - Fábry, Milan - Král, Vlastimil - Pachl, Petr - Hajdúch, M. - Grüner, Bohumír - Řezáčová, Pavlína
Structure-assisted design of inhibitors of CA IX enzyme based on polyhedral boron compounds.
Acta Crystallographica Section A-Foundation and Advances. Oxford Blackwell. Roč. 77 (2021), C864-C864. ISSN 2053-2733. E-ISSN 2053-2733
Institutional support: RVO:61388963 ; RVO:61388980 ; RVO:68378050
Keywords : carborane * cobal bis(dicarbollide) * carbonic anhydrase * enzyme inhibition * SAR study
https://journals.iucr.org/a/issues/2021/a2/00/a60441/a60441.pdf
Permanent Link: https://hdl.handle.net/11104/0339514 - 2.0521902 - ÚACH 2020 FR eng A - Abstract
Olejniczak, A. B. - Rózycka, D. - Rykowski, S. - Nekvinda, Jan - Grüner, Bohumír - Lesnikowski, Z. J. - Wyszko, E. - Fedoruk-Wyszomirska, A. - Gurda, D. - Orlicka Plocka, M. - Giel-Pietraszuk, M. - Kiliszek, A. - Rypniewski, W. - Kolodziej, P. - Ziaja-Soltys, M. - Bogucka-Kocka, A.
Compounds with carborane and matallacarborane components with antibacterial, anticancer, and antihelmintic activity.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "IL5".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
Institutional support: RVO:61388980
Keywords : metallacarborane
OECD category: Inorganic and nuclear chemistry
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306448 - 3.0521898 - ÚACH 2020 FR eng A - Abstract
Nekvinda, Jan - Holub, Josef - Brynda, Jiří - Pospíšilová, Klára - Řezáčová, Pavlína - Grüner, Bohumír
Alkylsulfonamido carboranes: the isomer dependence observed in inhibitory activity towards Carbonic Anhydrase IX.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "O48".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
R&D Projects: GA ČR(CZ) GA15-05677S; GA ČR(CZ) GA18-27648S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : Carbonic Anhydrase
OECD category: Inorganic and nuclear chemistry; Biochemistry and molecular biology (UMG-J)
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306442 - 4.0520890 - ÚOCHB 2020 GB eng A - Abstract
Řezáčová, Pavlína - Kugler, Michael - Brynda, Jiří - Grüner, Bohumír - Hajdúch, M. - Nekvinda, Jan - Pospíšilová, Klára - Das, V. - Holub, Josef
Structure-assisted design of Carborane inhibitors of human Carbonic anhydrase IX.
Acta Crystallographica Section A-Foundation and Advances. Oxford Blackwell. Roč. 74, Suppl (2018), „e197“. ISSN 2053-2733. E-ISSN 2053-2733.
[European Crystallography Meeting /31./. 22.08.2018-27.08.2018, Oviedo]
R&D Projects: GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LO1304; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : anti-tumor agents * carborane inhibitors * Carbonic anhydrase IX
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Permanent Link: http://hdl.handle.net/11104/0305557 - 5.0501881 - ÚOCHB 2019 GB eng A - Abstract
Brynda, Jiří - Řezáčová, Pavlína - Fábry, Milan - Štěpánková, J. - Král, Vlastimil - Hajdúch, M. - Holub, Josef - Nekvinda, Jan - Pospíšilová, Klára - Kugler, Michael - Grüner, Bohumír
Carborane and metallacarborane inhibitors of carbonic anhydrase IX, promising compounds for cancer therapy.
FEBS Open Bio. Wiley. Roč. 8, Suppl 1 (2018), s. 438. ISSN 2211-5463. E-ISSN 2211-5463.
[FEBS Congress /43./ Biochemistry Forever. 07.07.2018-12.07.2018, Prague]
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : carbonic anhydrase IX * inhibitors
OECD category: Biochemistry and molecular biology
Permanent Link: http://hdl.handle.net/11104/0293863 - 6.0501879 - ÚOCHB 2019 GB eng A - Abstract
Kugler, Michael - Brynda, Jiří - Řezáčová, Pavlína - Fábry, Milan - Král, Vlastimil - Pospíšilová, Klára - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Grüner, Bohumír
Structure-based design of human carbonic anhydrase XII inhibitors.
FEBS Open Bio. Wiley. Roč. 8, Suppl 1 (2018), s. 426-427. ISSN 2211-5463. E-ISSN 2211-5463.
[FEBS Congress /43./ Biochemistry Forever. 07.07.2018-12.07.2018, Prague]
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : carbonic anhydrase XII * inhibitors
OECD category: Biochemistry and molecular biology
Permanent Link: http://hdl.handle.net/11104/0293860 - 7.0484846 - ÚACH 2018 CN eng A - Abstract
Nekvinda, Jan - Grüner, Bohumír
Synthesis of Medicinally Relevant Carborane Cluster Derivatives.
IMEBORON 16 Programme. Hong Kong: Chinese University of Hong Kong, 2017. s. 187.
[IMEBORON: International Meeting on Boron Chemistry /16./. 09.07.2017-13.07.2017, Hong Kong]
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:61388980
Keywords : carborane cluster
Subject RIV: CA - Inorganic Chemistry
Permanent Link: http://hdl.handle.net/11104/0279970 - 8.0484844 - ÚACH 2018 CN eng A - Abstract
Grüner, Bohumír - Holub, Josef - Nekvinda, Jan - Šícha, Václav - Štěpánková, J. - Hajdúch, M. - Pospíšilová, K. - Řezáčová, Pavlína - Brynda, Jiří
Rational Design and Synthesis of Carborane and Metallacarborane Sulfonamides as Inhibitors of Carbonic AnhydraseIX.
IMEBORON 16 Programme. Hong Kong: Chinese University of Hong Kong, 2017.
[IMEBORON: International Meeting on Boron Chemistry /16./. 09.07.2017-13.07.2017, Hong Kong]
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : carboranes
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UMG-J)
Permanent Link: http://hdl.handle.net/11104/0279972 - 9.0469489 - ÚACH 2017 RU eng A - Abstract
Grüner, Bohumír - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Štěpánková, J. - Hajdúch, M. - Řezáčová, Pavlína - Brynda, Jiří
Metallacarborane chemistry: Site-directed substitutions designed for specific inhibition activity towards CA-IX.
EuroBoron 7 : Book of Abstracts. Moscow: Federal Agency for Scientific Organisations, 2016. s. 20.
[International Congress on Neutron Capture Theraphy /17./. 02.10.2016-07.10.2016, Columbia]
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:61388980 ; RVO:61388963 ; RVO:68378050
Keywords : metallacarborane inhibitors
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UOCHB-X); FR - Pharmacology ; Medidal Chemistry (UMG-J)
http://icnct17.org/AbstractBook17.pdf
Permanent Link: http://hdl.handle.net/11104/0267272 - 10.0469464 - ÚACH 2017 US eng A - Abstract
Grüner, Bohumír - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Štěpánková, J. - Hajdúch, M. - Řezáčová, Pavlína - Brynda, Jiří
Carborane and metallacarborane inhibitors of Carbonic Anhydrase IX, compounds with possible double action.
The 17th International Congress on Neutron Capture Theraphy : Abstracts for presentation. Columbia: University of Missouri, 2016. s. 89.
[International Congress on Neutron Capture Theraphy /17./. 02.10.2016-07.10.2016, Columbia]
R&D Projects: GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028
Institutional support: RVO:61388980 ; RVO:61388963 ; RVO:68378050
Keywords : metallacarborane inhibitors
Subject RIV: CA - Inorganic Chemistry; CE - Biochemistry (UOCHB-X); FR - Pharmacology ; Medidal Chemistry (UMG-J)
http://icnct17.org/AbstractBook17.pdf
Permanent Link: http://hdl.handle.net/11104/0267255