Search results
- 1.0574400 - ÚOCHB 2024 RIV GB eng J - Journal Article
Potalitsyn, Pavlo - Mrázková, Lucie - Selicharová, Irena - Tencerová, Michaela - Ferenčáková, Michaela - Chrudinová, Martina - Turnovská, Tereza - Brzozowski, A. M. - Marek, Aleš - Kaminský, Jakub - Jiráček, Jiří - Žáková, Lenka
Non-glycosylated IGF2 prohormones are more mitogenic than native IGF2.
Communications Biology. Roč. 6, č. 1 (2023), č. článku 863. E-ISSN 2399-3642
R&D Projects: GA ČR(CZ) GA19-14069S; GA MŠMT(CZ) EF16_019/0000729; GA MŠMT(CZ) LX22NPO5104
Institutional support: RVO:61388963 ; RVO:67985823
Keywords : hormone * prohormone * precursor * mitogenic * receptor * IGF
OECD category: Biochemistry and molecular biology
Impact factor: 5.9, year: 2022
Method of publishing: Open access
https://doi.org/10.1038/s42003-023-05239-6
Permanent Link: https://hdl.handle.net/11104/0344735File Download Size Commentary Version Access 10.1038s42003-023-05239-6.pdf 1 2.1 MB Publisher’s postprint open-access - 2.0546413 - ÚOCHB 2022 RIV US eng J - Journal Article
Páníková, Terezie - Mitrová, Katarína - Halamová, Tereza - Mrzílková, Karolína - Pícha, Jan - Chrudinová, Martina - Kurochka, Andrii - Selicharová, Irena - Žáková, Lenka - Jiráček, Jiří
Insulin Analogues with Altered Insulin Receptor Isoform Binding Specificities and Enhanced Aggregation Stabilities.
Journal of Medicinal Chemistry. Roč. 64, č. 19 (2021), s. 14848-14859. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : insulin * hepatoselective * stability
OECD category: Medicinal chemistry
Impact factor: 8.039, year: 2021
Method of publishing: Limited access
https://doi.org/10.1021/acs.jmedchem.1c01388
Permanent Link: http://hdl.handle.net/11104/0322932 - 3.0533335 - ÚOCHB 2021 RIV GB eng J - Journal Article
Dzianová, P. - Asai, Seiya - Chrudinová, Martina - Kosinová, L. - Potalitsyn, Pavlo - Šácha, Pavel - Hadravová, Romana - Selicharová, Irena - Kříž, J. - Turkenburg, J. P. - Brzozowski, A. M. - Jiráček, Jiří - Žáková, Lenka
The efficiency of insulin production and its content in insulin-expressing model β-cells correlate with their Zn2+ levels.
Open Biology. Roč. 10, č. 10 (2020), č. článku 200137. E-ISSN 2046-2441
R&D Projects: GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : insulin * zinc * beta cells * production ZnT8
OECD category: Biochemistry and molecular biology
Impact factor: 6.411, year: 2020
Method of publishing: Open access
https://doi.org/10.1098/rsob.200137
Permanent Link: http://hdl.handle.net/11104/0311840 - 4.0511146 - ÚOCHB 2020 RIV US eng J - Journal Article
Macháčková, Kateřina - Mlčochová, K. - Potalitsyn, Pavlo - Hanková, Kateřina - Socha, Ondřej - Buděšínský, Miloš - Muždalo, Anja - Lepšík, Martin - Černeková, Michaela - Radosavljević, Jelena - Fábry, Milan - Mitrová, Katarína - Chrudinová, Martina - Lin, Jingjing - Yurenko, Yevgen - Hobza, Pavel - Selicharová, Irena - Žáková, Lenka - Jiráček, Jiří
Mutations at hypothetical binding site 2 in insulin and insulin-like growth factors 1 and 2 result in receptor- and hormone-specific responses.
Journal of Biological Chemistry. Roč. 294, č. 46 (2019), s. 17371-17382. ISSN 0021-9258. E-ISSN 1083-351X
R&D Projects: GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963 ; RVO:68378050
Keywords : insulin * IGF * receptor
OECD category: Biochemistry and molecular biology
Impact factor: 4.238, year: 2019
Method of publishing: Open access
http://www.jbc.org/content/294/46/17371
Permanent Link: http://hdl.handle.net/11104/0301483File Download Size Commentary Version Access 0511146.pdf 2 2.2 MB Publisher’s postprint open-access - 5.0498264 - ÚOCHB 2019 RIV US eng J - Journal Article
Chrudinová, Martina - Žáková, Lenka - Marek, Aleš - Socha, Ondřej - Buděšínský, Miloš - Hubálek, Martin - Pícha, Jan - Macháčková, Kateřina - Jiráček, Jiří - Selicharová, Irena
A versatile insulin analog with high potency for both insulin and insulin-like growth factor 1 receptors: Structural implications for receptor binding.
Journal of Biological Chemistry. Roč. 293, č. 43 (2018), s. 16818-16829. ISSN 0021-9258. E-ISSN 1083-351X
R&D Projects: GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : insulin * insulin-like growth factor (IGF) * structure-function * insulin receptor * protein design * kinetics * binding * Site 1
OECD category: Biochemistry and molecular biology
Impact factor: 4.106, year: 2018
http://www.jbc.org/content/293/43/16818.full
Permanent Link: http://hdl.handle.net/11104/0291126File Download Size Commentary Version Access 0498264.pdf 2 2.3 MB Publisher’s postprint open-access - 6.0495744 - ÚOCHB 2019 RIV DE eng J - Journal Article
Fabre, Benjamin - Pícha, Jan - Selicharová, Irena - Žáková, Lenka - Chrudinová, Martina - Hajduch, Jan - Jiráček, Jiří
Probing Tripodal Peptide Scaffolds as Insulin and IGF-1 Receptor Ligands.
European Journal of Organic Chemistry. Roč. 2018, č. 37 (2018), s. 5193-5201. ISSN 1434-193X. E-ISSN 1099-0690
R&D Projects: GA ČR GA14-17305S; GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : insulin * peptidomimetics * insulin receptor * IGF-1
OECD category: Organic chemistry
Impact factor: 3.029, year: 2018
Permanent Link: http://hdl.handle.net/11104/0288670 - 7.0489708 - ÚOCHB 2019 RIV US eng J - Journal Article
Macháčková, Kateřina - Chrudinová, Martina - Radosavljević, Jelena - Potalitsyn, Pavlo - Křížková, Květoslava - Fábry, Milan - Selicharová, Irena - Collinsová, Michaela - Brzozowski, A. M. - Žáková, Lenka - Jiráček, Jiří
Converting Insulin-like Growth Factors 1 and 2 into High-Affinity Ligands for Insulin Receptor Isoform A by the Introduction of an Evolutionarily Divergent Mutation.
Biochemistry. Roč. 57, č. 16 (2018), s. 2373-2382. ISSN 0006-2960
R&D Projects: GA ČR GA15-19018S
Institutional support: RVO:61388963 ; RVO:68378050
Keywords : insulin-like growth factor * insulin * receptor * analog
OECD category: Biochemistry and molecular biology
Impact factor: 2.952, year: 2018
https://pubs.acs.org/doi/10.1021/acs.biochem.7b01260
Permanent Link: http://hdl.handle.net/11104/0284074File Download Size Commentary Version Access 0489708.pdf 5 3.3 MB Publisher’s postprint open-access - 8.0484559 - ÚOCHB 2018 RIV US eng J - Journal Article
Macháčková, Kateřina - Collinsová, Michaela - Chrudinová, Martina - Selicharová, Irena - Pícha, Jan - Buděšínský, Miloš - Vaněk, Václav - Žáková, Lenka - Brzozowski, A. M. - Jiráček, Jiří
Insulin-like Growth Factor 1 Analogs Clicked in the C Domain: Chemical Synthesis and Biological Activities.
Journal of Medicinal Chemistry. Roč. 60, č. 24 (2017), s. 10105-10117. ISSN 0022-2623. E-ISSN 1520-4804
Institutional support: RVO:61388963
Keywords : IGF-1 * receptor * synthesis * triazole
OECD category: Biochemistry and molecular biology
Impact factor: 6.253, year: 2017
http://pubs.acs.org/doi/full/10.1021/acs.jmedchem.7b01331
Permanent Link: http://hdl.handle.net/11104/0279723File Download Size Commentary Version Access 0484559.pdf 6 1.7 MB Publisher’s postprint open-access - 9.0469437 - ÚOCHB 2017 RIV US eng J - Journal Article
Fabre, Benjamin - Pícha, Jan - Vaněk, Václav - Selicharová, Irena - Chrudinová, Martina - Collinsová, Michaela - Žáková, Lenka - Buděšínský, Miloš - Jiráček, Jiří
Synthesis and Evaluation of a Library of Trifunctional Scaffold-Derived Compounds as Modulators of the Insulin Receptor.
ACS Combinatorial Science. Roč. 18, č. 12 (2016), s. 710-722. ISSN 2156-8952. E-ISSN 2156-8944
R&D Projects: GA ČR GA14-17305S
Institutional support: RVO:61388963
Keywords : insulin mimetics * insulin receptor * library * protein-protein interactions * scaffold * trifunctional
Subject RIV: CE - Biochemistry
Impact factor: 3.168, year: 2016
http://pubs.acs.org/doi/full/10.1021/acscombsci.6b00132
Permanent Link: http://hdl.handle.net/11104/0267220 - 10.0461800 - ÚOCHB 2017 RIV US eng J - Journal Article
Křížková, Květoslava - Chrudinová, Martina - Povalová, Anna - Selicharová, Irena - Collinsová, Michaela - Vaněk, Václav - Brzozowski, A. M. - Jiráček, Jiří - Žáková, Lenka
Insulin-Insulin-like Growth Factors Hybrids as Molecular Probes of Hormone:Receptor Binding Specificity.
Biochemistry. Roč. 55, č. 21 (2016), s. 2903-2913. ISSN 0006-2960
R&D Projects: GA ČR GA15-19018S
Institutional support: RVO:61388963
Keywords : alanine scanning mutagenesis * high-affinity binding * type 1 IGF receptor
Subject RIV: CE - Biochemistry
Impact factor: 2.938, year: 2016
http://pubs.acs.org/doi/pdf/10.1021/acs.biochem.6b00140
Permanent Link: http://hdl.handle.net/11104/0261380File Download Size Commentary Version Access 0461800.pdf 2 1.9 MB Publisher’s postprint open-access