Search results
- 1.0567440 - ÚVGZ 2023 RIV CH eng J - Journal Article
Gonec, T. - Vráblová, L. - Pidnjaková, D. - Strhanský, T. - Oravec, Michal - Jampílek, J.
Preparation and Hydro-Lipophilic Properties of Monosubstituted N-Aryl-4-hydroxyquinoline-3-carboxanilides †.
Chemistry Proceedings. Roč. 2022, č. 12 (2022), č. článku 28. E-ISSN 2673-4583
R&D Projects: GA MŠMT(CZ) LM2018123; GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : hydroxyquinoline-carboxanilides * synthesis * lipophilicity
OECD category: Organic chemistry
Method of publishing: Open access
https://www.mdpi.com/2673-4583/12/1/28
Permanent Link: https://hdl.handle.net/11104/0338695File Download Size Commentary Version Access chemproc-12-00028.pdf 2 1.4 MB Publisher’s postprint open-access - 2.0566362 - ÚVGZ 2023 RIV CH eng J - Journal Article
Strharsky, T. - Pindjakova, D. - Kos, J. - Vrablova, L. - Smak, P. - Michnová, H. - Gonec, T. - Hošek, J. - Oravec, Michal - Jendrzejewska, I. - Čížek, A. - Jampílek, J.
Trifluoromethylcinnamanilide Michael Acceptors for Treatment of Resistant Bacterial Infections.
International Journal of Molecular Sciences. Roč. 23, č. 23 (2022), č. článku 15090. E-ISSN 1422-0067
R&D Projects: GA MŠMT(CZ) LM2018123; GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : cinnamamides * Michael acceptors * antimicrobial activity * cytotoxicity * lipophilicity * structure-activity relationships * docking study
OECD category: Biochemistry and molecular biology
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1422-0067/23/23/15090
Permanent Link: https://hdl.handle.net/11104/0337705File Download Size Commentary Version Access ijms-23-15090.pdf 3 4.8 MB Publisher’s postprint open-access - 3.0558879 - ÚVGZ 2023 RIV CH eng J - Journal Article
Gonec, T. - Pindjakova, D. - Vrablova, L. - Strharsky, T. - Michnova, H. - Kauerová, T. - Kollár, P. - Oravec, Michal - Jendrzejewska, I. - Čížek, A. - Jampílek, J.
Antistaphylococcal Activities and ADME-Related Properties of Chlorinated Arylcarbamoylnaphthalenylcarbamates.
Pharmaceuticals. Roč. 15, č. 6 (2022), č. článku 715. E-ISSN 1424-8247
R&D Projects: GA MŠMT(CZ) LM2018123; GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : antimicrobial activity * staphylococcus-aureus * biological-activity * resistance * derivatives * permeability * mechanisms * spectrum * design * oxides * hydroxynaphthalenes * carbamates * antistaphylococcal activity * cytotoxicity * lipophilicity * structure-activity relationships
OECD category: Pharmacology and pharmacy
Impact factor: 4.6, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1424-8247/15/6/715
Permanent Link: http://hdl.handle.net/11104/0332380 - 4.0546621 - BFÚ 2022 RIV CH eng J - Journal Article
Gajdar, J. - Kos, J. - Gonec, T. - Brázdová, Marie - Soldanová, Zuzana - Fojta, Miroslav - Jampílek, J. - Barek, J. - Fischer, J.
Substituent effect of ring-substituted 3-hydroxynaphthalene-2-carboxanilides and 2-hydroxynaphthalene-1-carboxanilides in relation to their electrochemical and biological activity.
Journal of Electroanalytical Chemistry. Roč. 899, OCT 15 2021 (2021), č. článku 115667. ISSN 1572-6657. E-ISSN 1873-2569
Institutional support: RVO:68081707
Keywords : herbicidal activity * antioxidant activity * antimycobacterial * antibacterial * agents
OECD category: Electrochemistry (dry cells, batteries, fuel cells, corrosion metals, electrolysis)
Impact factor: 4.598, year: 2021
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S1572665721006937?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0323067 - 5.0534773 - ÚVGZ 2021 RIV US eng J - Journal Article
Campos, L. E. - Garibotto, F. - Angelina, E. - Kos, J. - Gonec, T. - Marvanová, P. - Vettorazzi, M. - Oravec, Michal - Jendrzejewska, I. - Jampílek, J. - Alvarez, S. E. - Enriz, R. D.
Hydroxynaphthalenecarboxamides and substituted piperazinylpropandiols, two new series of BRAF inhibitors. A theoretical and experimental study.
Bioorganic Chemistry. Roč. 103, OCT (2020), č. článku 104145. ISSN 0045-2068. E-ISSN 1090-2120
R&D Projects: GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : raf inhibitors * mapk pathway * BRAF inhibitors * Melanoma * Molecular modeling * Cell viability * ERK phosphorylation
OECD category: Biochemistry and molecular biology
Impact factor: 5.275, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0045206820314425?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0312945 - 6.0524255 - BFÚ 2021 RIV GB eng J - Journal Article
Gajdar, J. - Tsami, K. - Michnova, H. - Gonec, T. - Brázdová, Marie - Soldanová, Zuzana - Fojta, Miroslav - Jampílek, J. - Barek, J. - Fischer, J.
Electrochemistry of ring-substituted 1-hydroxynaphthalene-2-carboxanilides: Relation to structure and biological activity.
Electrochimica acta. Roč. 332, FEB 1 2020 (2020), č. článku 135485. ISSN 0013-4686. E-ISSN 1873-3859
Institutional support: RVO:68081707
Keywords : herbicidal activity * mycobacterium-tuberculosis * ANTIMYCOBACTERIAL
OECD category: Electrochemistry (dry cells, batteries, fuel cells, corrosion metals, electrolysis)
Impact factor: 6.901, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0013468619323576?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0308637 - 7.0446420 - ÚVGZ 2016 RIV GB eng J - Journal Article
Kos, J. - Zadražilová, I. - Nevin, E. - Soral, M. - Gonec, T. - Kollár, P. - Oravec, Michal - Coffey, A. - O'Mahony, J. - Liptaj, T. - Kralova, K. - Jampílek, J.
Ring-substituted 8-hydroxyquinoline-2-carboxanilides as potential antimycobacterial agents.
Bioorganic & Medicinal Chemistry. Roč. 23, č. 15 (2015), s. 4188-4196. ISSN 0968-0896. E-ISSN 1464-3391
Institutional support: RVO:67179843
Keywords : 8-Hydroxyquinolines * in vitro antimycobacterial activity * in vitro cytotoxicity * MTT assay * Structure–activity relationships
Subject RIV: CE - Biochemistry
Impact factor: 2.923, year: 2015
Permanent Link: http://hdl.handle.net/11104/0248413