Search results
- 1.0518499 - ÚOCHB 2020 TH eng A - Abstract
Břehová, Petra - Šmídková, Markéta - Skácel, Jan - Dračínský, Martin - Mertlíková-Kaiserová, Helena - Velasquez, M. P. S. - Watts, W. J. - Janeba, Zlatko
Synthesis of acyclic nucleoside phosphonates derived from 2-aminothiazoles and their evaluation as inhibitors of bacterial and human adenylate cyclases.
20th Tetrahedron Symposium. Bangkok: Elsevier, 2019. P1.005, „P1004“.
[Tetrahedron Symposium /20./. 18.06.2019-21.06.2019, Bangkok]
Institutional support: RVO:61388963
Keywords : nucleoside analogues * adenylate cyclases * aminothiazoles
OECD category: Organic chemistry
Permanent Link: http://hdl.handle.net/11104/0303890 - 2.0490582 - ÚOCHB 2019 CZ eng A - Abstract
Adla, Santosh Kumar - Slavíková, Barbora - Chodounská, Hana - Vyklický, Vojtěch - Ladislav, Marek - Hubálková, Pavla - Krausová, Barbora - Nekardová, Michaela - Šmídková, Markéta - Monincová, Lenka - Souček, Radko - Majer, Pavel - Vyklický ml., Ladislav - Kudová, Eva
Steroidal inhibitors of N‐methyl‐D‐aspartate receptors with C‐3 amide structural motif: Evaluation of their inhibitory effect, cytotoxicity and plasma stability.
Sborník příspěvků 6. České lipidomické konference. Praha: Ústav organické chemie a biochemie AV ČR, 2018 - (Kuda, O.). P5. ISBN 978-80-86241-59-3.
[Česká lipidomická konference /6./. 14.06.2018-15.06.2018, Praha]
Institutional support: RVO:61388963 ; RVO:67985823 ; RVO:86652036
Keywords : steroidal inhibitor * NMDA * PAG
OECD category: Organic chemistry
http://lipidomics.uochb.cas.cz/6CLK_sbornik2018.pdf
Permanent Link: http://hdl.handle.net/11104/0284793File Download Size Commentary Version Access 6CLK_sbornik2018.pdf 1 666.7 KB Publisher’s postprint open-access - 3.0481195 - ÚOCHB 2018 CZ eng A - Abstract
Česnek, Michal - Dračínský, Martin - Šmídková, Markéta - Mertlíková-Kaiserová, Helena - Velasquez, M. P. S. - Watts, V. J. - Janeba, Zlatko
Synthesis and evaluation of novel acyclic nucleoside phosphonates with unnatural nucleobases as potent inhibitors of Bordetella pertussis adenylate cyclase toxin.
SCNAC 2017. 17th Symposium on Chemistry of Nucleic Acid Components. Praha: Confis Conference, 2017. s. 128.
[SCNAC 2017. Symposium on Chemistry of Nucleic Acid Components /17./. 04.06.2017-09.06.2017, Český Krumlov]
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates (ANPs) * adenylate cyclase toxin (ACT) * Bordetella pertussis
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0276795 - 4.0481189 - ÚOCHB 2018 CZ eng A - Abstract
Břehová, Petra - Šmídková, Markéta - Skácel, Jan - Dračínský, Martin - Mertlíková-Kaiserová, Helena - Velasquez, M. P. S. - Watts, V. J. - Janeba, Zlatko
Synthesis of acyclic nucleoside phosphonates with unnatural heterocyclic bases bearing aryl substituents and their inhibitory activity towards bacterial and human adenylate cyclases.
SCNAC 2017. 17th Symposium on Chemistry of Nucleic Acid Components. Praha: Confis Conference, 2017. s. 125.
[SCNAC 2017. Symposium on Chemistry of Nucleic Acid Components /17./. 04.06.2017-09.06.2017, Český Krumlov]
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates (ANPs) * adenylate cyclase toxin (ACT) * Bordetella pertussis
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0276789 - 5.0465007 - ÚOCHB 2017 NL eng A - Abstract
Frydrych, Jan - Dračínský, Martin - Gnanasekaran, Ramachandran - Lepšík, Martin - Šmídková, Markéta - Tloušťová, Eva - Mertlíková-Kaiserová, Helena - Janeba, Zlatko
Novel adenine acyclic nucleoside phosphonates and their derivatives as potent inhibitors of bacterial adenylate cyclases.
ECHC 2016. 27th European Colloquium on Heterocyclic Chemistry. Amsterdam: -, 2016.
[ECHC 2016. European Colloquium on Heterocyclic Chemistry /27./. 03.07.2016-06.07.2016, Amsterdam]
R&D Projects: GA MV VG20102015046; GA ČR(CZ) GBP208/12/G016; GA MŠMT LO1302
Institutional support: RVO:61388963
Keywords : acyclic nuceloside phosphonates * bacterial adenylate cyclases
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0263730 - 6.0464964 - ÚOCHB 2017 ES eng A - Abstract
Česnek, Michal - Šmídková, Markéta - Dračínský, Martin - Janeba, Zlatko
Novel acyclic nucleoside phosphonates containing unnatural nucleobases as potent inhibitors of Bordetella pertussis adenylyl cyclase toxin.
17th Tetrahedron Symposium. Challenges in Biological, Bioorganic, Organic and Medicinal Chemistry. Sitges: Elsevier, 2016.
[Tetrahedron Symposium. Challenges in Biological, Bioorganic, Organic and Medicinal Chemistry /17./. 28.06.2016-01.07.2016, Sitges]
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates (ANPs) * adenylate cyclase toxin (ACT) * Bordetella pertussis
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0263704 - 7.0464963 - ÚOCHB 2017 ES eng A - Abstract
Břehová, Petra - Šmídková, Markéta - Mertlíková-Kaiserová, Helena - Skácel, Jan - Dračínský, Martin - Janeba, Zlatko
Synthesis of acyclic nucleoside phosphonates bearing aryl substituent at the acyclic linker as potential inhibitors of adenylate cyclase toxin from Bordetella pertussis.
17th Tetrahedron Symposium. Challenges in Biological, Bioorganic, Organic and Medicinal Chemistry. Sitges: Elsevier, 2016.
[Tetrahedron Symposium. Challenges in Biological, Bioorganic, Organic and Medicinal Chemistry /17./. 28.06.2016-01.07.2016, Sitges]
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates (ANPs) * adenylate cyclase toxin (ACT) * Bordetella pertussis
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0263697 - 8.0459819 - ÚOCHB 2017 CZ eng A - Abstract
Kudová, Eva - Vyklický ml., Ladislav - Šmídková, Markéta - Nekardová, Michaela - Zborníková, Eva - Balaštík, Martin - Valeš, Karel - Mareš, Pavel - Paleček, Jiří
SMART Steroids.
Sborník příspěvků 5. České lipidomické konference. Praha: Ústav organické chemie a biochemie AV ČR, 2016 - (Kuda, O.). s. 16-17. ISBN 978-80-86241-54-8.
[Česká lipidomická konference /5./. 21.04.2016-22.04.2016, Praha]
R&D Projects: GA TA ČR(CZ) TE01020028; GA ČR(CZ) GAP303/12/1464
Institutional support: RVO:61388963 ; RVO:67985823
Keywords : NMDA receptor * neurosteroids
Subject RIV: ED - Physiology
Permanent Link: http://hdl.handle.net/11104/0259975File Download Size Commentary Version Access 5CLK-sbornik_2016.pdf 0 1 MB Publisher’s postprint open-access - 9.0454279 - ÚOCHB 2016 CZ eng A - Abstract
Břehová, Petra - Šmídková, Markéta - Mertlíková-Kaiserová, Helena - Dračínský, Martin - Janeba, Zlatko
Synthesis of acyclic nucleoside phosphonates bearing (N-methyl)anthraniloyl substituent as potential inhibitors of adenylate cyclase toxin from Bordetella Pertussis.
Liblice 2015. 50th Advances in Organic, Bioorganic and Pharmaceutical Chemistry. Praha: Czech Chemical Society, 2015. s. 61.
[Liblice 2015. Advances in Organic, Bioorganic and Pharmaceutical Chemistry /50./. 06.11.2015-08.11.2015, Olomouc]
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates * adenylate cyclase toxin * prodrugs
Subject RIV: CC - Organic Chemistry
Permanent Link: http://hdl.handle.net/11104/0256230 - 10.0442824 - ÚOCHB 2016 CZ cze A - Abstract
Hájek, Miroslav - Kužmová, Erika - Šmídková, Markéta - Kolman, Viktor - Zídek, Zdeněk - Jansa, P.
Studium vlivu polysubstituovaných pyrimidinů na expresi genů spojených se zánětlivou reakcí.
[Effects of polysubstituted pyrimidines on expression of inflammation-related genes.]
ENBIK 2014. Konferenční sborník. Praha: Vysoká škola chemicko-technologická v Praze, 2014 - (Čech, P.; Svozil, D.). s. 78. ISBN 978-80-7080-883-2.
[ENBIK 2014. 09.06.2014-11.06.2014, Kouty na Vysočině]
Institutional support: RVO:61388963 ; RVO:68378041
Keywords : inflammation * gene expression * substituted pyrimidines
Subject RIV: CE - Biochemistry
Permanent Link: http://hdl.handle.net/11104/0245646