Search results

  1. 1.
    0584241 - ÚEM 2025 RIV NL eng J - Journal Article
    Mezeiová, E. - Prchal, L. - Hrabinová, M. - Mucková, L. - Pulkrabková, L. - Soukup, O. - Misiachna, Anna - Janoušek, J. - Fibigar, J. - Kučera, T. - Horák, Martin - Makhaeva, G.F. - Korabecný, J.
    Morphing cholinesterase inhibitor amiridine into multipotent drugs for the
    treatment of Alzheimer’s disease.
    Biomedicine & Pharmacotherapy. Roč. 173, april. (2024), č. článku 116399. ISSN 0753-3322. E-ISSN 1950-6007
    R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) EH22_008/0004562
    Institutional support: RVO:68378041
    Keywords : amiridine * acetylcholinesterase * antioxidant capacity * butyrylcholinesterase * multi-target directed ligands * NMDA receptors
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 7.5, year: 2022
    Method of publishing: Open access
    https://www.sciencedirect.com/science/article/pii/S075333222400283X?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0352201
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    Mezeirová 2024.pdf31.7 MBPublisher’s postprintopen-access
     
     
  2. 2.
    0584110 - ÚMCH 2025 RIV GB eng J - Journal Article
    Hoang, Stéphane - Zhukouskaya, Hanna - Ivanko, Iryna - Svoboda, Jan - Hympánová, M. - Marek, J. - Soukup, O. - Šlouf, Miroslav - Kotek, J. - Doris, E. - Gravel, E. - Tomšík, Elena - Hrubý, Martin
    Improved electro-destruction of bacterial biofilms by coating conductive surfaces with polymers.
    European Polymer Journal. Roč. 209, 15 April (2024), č. článku 112910. ISSN 0014-3057. E-ISSN 1873-1945
    R&D Projects: GA ČR(CZ) GA21-01090S; GA MŠMT(CZ) LUAUS24272; GA MŠMT(CZ) EH22_008/0004607
    Institutional support: RVO:61389013
    Keywords : bacteria * biofilm * polymer
    OECD category: Polymer science
    Impact factor: 6, year: 2022
    Method of publishing: Limited access
    https://www.sciencedirect.com/science/article/pii/S001430572400171X?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0352482
     
     
  3. 3.
    0582133 - ÚEM 2025 RIV NL eng J - Journal Article
    Misiachna, Anna - Svobodová, B. - Netolický, Jakub - Chvojková, M. - Kletečková, L. - Prchal, L. - Novák, M. - Hrabinová, M. - Kučera, T. - Mucková, L. - Moravcová, Z. - Karasová-Ždárová, J. - Pejchal, J. - Blažek, F. - Maliňák, D. - Hakenová, K. - Hrčka Krausová, Barbora - Kolcheva, Marharyta - Ladislav, Marek - Korábečný, J. - Pahnke, J. - Valeš, K. - Horák, Martin - Soukup, O.
    Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition.
    European Journal of Medicinal Chemistry. Roč. 266, feb. (2024), č. článku 116130. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA TA ČR(CZ) TO01000078; GA MŠMT(CZ) EH22_008/0004562
    Institutional support: RVO:68378041
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 6.7, year: 2022
    Method of publishing: Open access
    https://www.sciencedirect.com/science/article/pii/S0223523424000102?via%3Dihub https://doi.org/10.5281/zenodo.10949371 https://doi.org/10.2139/ssrn.4658299
    Permanent Link: https://hdl.handle.net/11104/0350209
    FileDownloadSizeCommentaryVersionAccess
    Misiachna příloha 2024.pdf19.8 MBOtheropen-access
    Misiachna 2024.pdf45 MBPublisher’s postprintopen-access
     
     
  4. 4.
    0573825 - FGÚ 2024 RIV GB eng J - Journal Article
    Vojtěchová, Iveta - Tučková, K. - Jůza, R. - Stuchlík, Aleš - Kelemen, E. - Korábečný, J. - Soukup, O. - Petrásek, Tomáš
    Dopaminergic and glutamatergic models of psychosis show differential sensitivity to aripiprazole and a novel experimental compound modulating D2/5-HT receptor activity.
    Progress in Neuro-Psychopharmacology & Biological Psychiatry. Roč. 127, 20 Dec (2023), č. článku 110819. ISSN 0278-5846. E-ISSN 1878-4216
    R&D Projects: GA MZd(CZ) NU22-04-00526
    Institutional support: RVO:67985823
    Keywords : schizophrenia * dizocilpine * amphetamine * antipsychotic * aripiprazole
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 5.6, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1016/j.pnpbp.2023.110819
    Permanent Link: https://hdl.handle.net/11104/0344177
     
     
  5. 5.
    0572189 - ÚEM 2024 RIV CH eng J - Journal Article
    Svobodová, B. - Pulkrabová, L. - Pánek, D. - Misiachna, Anna - Kolcheva, Marharyta - Andrýs, R. - Handl, J. - Čapek, J. - Nývltová, P. - Roušar, T. - Prchal, L. - Hepnarová, V. - Hrabinová, M. - Mucková, L. - Tosnerová, D. - Karabanovich, G. - Finger, V. - Soukup, O. - Horák, Martin - Korabecný, J.
    Structure-Guided Design of N-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer’s Disease.
    International Journal of Molecular Sciences. Roč. 24, č. 11 (2023), č. článku 9124. ISSN 1661-6596
    R&D Projects: GA ČR(CZ) GA22-24384S; GA MŠMT(CZ) LX22NPO5107
    Institutional support: RVO:68378041
    Keywords : Alzheimer’s disease * acetylcholinesterase * enzyme inhibition * N-methyl-d-aspartate receptor * multi-target directed ligands * monoamine oxidase A/B
    OECD category: Pharmacology and pharmacy
    Impact factor: 5.6, year: 2022
    Method of publishing: Open access
    https://doi.org/10.3390/ijms24119124
    Permanent Link: https://hdl.handle.net/11104/0342960
    FileDownloadSizeCommentaryVersionAccess
    Svobodová 2023.pdf23.8 MBPublisher’s postprintopen-access
     
     
  6. 6.
    0559439 - ÚMG 2023 RIV FR eng J - Journal Article
    Gorecki, L. - Muthna, D. - Merdita, S. - Andrš, Martin - Kučera, T. - Havelek, R. - Mucková, L. - Kobrlová, T. - Soukup, J. - Krupa, P. - Prchal, L. - Soukup, O. - Roh, J. - Řezáčová, M. - Korábečný, J.
    7-Azaindole, 2,7-diazaindole, and 1H-pyrazole as core structures for novel anticancer agents with potential chemosensitizing properties.
    European Journal of Medicinal Chemistry. Roč. 240, June (2022), č. článku 114580. ISSN 0223-5234. E-ISSN 1768-3254
    Institutional support: RVO:68378050
    Keywords : ATR inhibition * Berzosertib * Cancer * Chemosensitization * Cytotoxicity * Glioblastoma
    OECD category: Cell biology
    Impact factor: 6.7, year: 2022
    Method of publishing: Limited access
    https://www.sciencedirect.com/science/article/abs/pii/S0223523422004822?via%3Dihub
    Permanent Link: https://hdl.handle.net/11104/0332860
     
     
  7. 7.
    0556370 - FGÚ 2023 RIV FR eng J - Journal Article
    Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
    Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
    European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
    Institutional support: RVO:67985823
    Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.7, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1016/j.ejmech.2022.114193
    Permanent Link: http://hdl.handle.net/11104/0330742
     
     
  8. 8.
    0551558 - ÚEM 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
    Institutional support: RVO:68378041
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
    OECD category: Medicinal chemistry
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0326821
     
     
  9. 9.
    0546462 - FGÚ 2022 RIV CH eng J - Journal Article
    Jůza, R. - Štefková, K. - Dehaen, W. - Randáková, Alena - Petrásek, T. - Vojtěchová, I. - Kobrlová, T. - Pulkrábková, L. - Mucková, L. - Mecava, M. - Prchal, L. - Mezeiová, E. - Musílek, K. - Soukup, O. - Korábečný, J.
    Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D-2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
    Biomolecules. Roč. 11, č. 9 (2021), č. článku 1262. E-ISSN 2218-273X
    Institutional support: RVO:67985823
    Keywords : aripiprazole * dopamine receptor * blood–brain barrier * molecular modeling studies * schizophrenia
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.064, year: 2021
    Method of publishing: Open access
    https://www.mdpi.com/2218-273X/11/9/1262
    Permanent Link: http://hdl.handle.net/11104/0322976
     
     
  10. 10.
    0544878 - ÚMG 2022 RIV NZ eng J - Journal Article
    Salajková, Šárka - Havel, Filip - Šrámek, Michal - Novotný, Filip - Malinak, D. - Doležal, R. - Prchal, L. - Benková, M. - Soukup, O. - Musílek, K. - Kuca, K. - Bártek, Jiří - Proska, J. - Žárská, Monika - Hodný, Zdeněk
    The Effect of Chemical Structure of OEG Ligand Shells with Quaternary Ammonium Moiety on the Colloidal Stabilization, Cellular Uptake and Photothermal Stability of Gold Nanorods.
    International Journal of Nanomedicine. Roč. 16, May (2021), s. 3407-3427. E-ISSN 1178-2013
    R&D Projects: GA ČR GA16-13967S; GA MZd NV19-08-00523; GA MŠMT(CZ) LM2015062; GA MŠMT(CZ) LM2015062; GA MŠMT(CZ) EF16_013/0001775
    Institutional support: RVO:68378050
    Keywords : gold nanorods * quaternary ammonium salts * oligoethylene glycol * cellular uptake * photothermal stability
    OECD category: Pharmacology and pharmacy
    Impact factor: 7.033, year: 2021
    Method of publishing: Open access
    https://www.dovepress.com/the-effect-of-chemical-structure-of-oeg-ligand-shells-with-quaternary--peer-reviewed-fulltext-article-IJN
    Permanent Link: http://hdl.handle.net/11104/0321676
     
     

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