Search results
- 1.0456441 - ÚOCHB 2016 RIV FR eng J - Journal Article
Buemi, M. R. - De Luca, L. - Ferro, S. - Bruno, E. - Ceruso, M. - Supuran, C. T. - Pospíšilová, K. - Brynda, Jiří - Řezáčová, Pavlína - Gitto, R.
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms.
European Journal of Medicinal Chemistry. Roč. 102, Sep 18 (2015), s. 223-232. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:61388963
Keywords : human carbonic anhydrase * isoquinoline * quinoline * X-ray * molecular docking
Subject RIV: CE - Biochemistry
Impact factor: 3.902, year: 2015
Permanent Link: http://hdl.handle.net/11104/0256969 - 2.0455782 - ÚMG 2016 RIV FR eng J - Journal Article
Buemi, M. R. - De Luca, L. - Ferro, S. - Bruno, E. - Ceruso, M. - Supuran, C. T. - Pospíšilová, K. - Brynda, Jiří - Řezáčová, Pavlína - Gitto, R.
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms.
European Journal of Medicinal Chemistry. Roč. 102, SEP 18 (2015), s. 223-232. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR GA15-05677S
Grant - others:Fondo di Ateneo per la Ricerca (PRA)(IT) ORME09SPNC
Institutional support: RVO:68378050
Keywords : Human carbonic anhydrase * Isoquinoline * Quinoline * X-ray * Molecular docking
Subject RIV: EB - Genetics ; Molecular Biology
Impact factor: 3.902, year: 2015
Permanent Link: http://hdl.handle.net/11104/0256405 - 3.0378892 - ÚMG 2013 RIV US eng J - Journal Article
Gitto, R. - Damiano, F. - Mader, Pavel - De Luca, L. - Ferro, S. - Supuran, C. T. - Vullo, D. - Brynda, Jiří - Řezáčová, Pavlína - Chimirri, A.
Synthesis, structure-activity relationship studies, and X-ray crystallographic analysis of arylsulfonamides as potent carbonic anhydrase inhibitors.
Journal of Medicinal Chemistry. Roč. 55, č. 8 (2012), s. 3891-3899. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR GA203/09/0820
Grant - others:MiUR(IT) 20085HR5JK_002; EK(XE) 222741
Institutional research plan: CEZ:AV0Z50520514; CEZ:AV0Z40550506
Keywords : carbonic anhydrase * inhibitors * arylsulfonamides
Subject RIV: EB - Genetics ; Molecular Biology
Impact factor: 5.614, year: 2012
Permanent Link: http://hdl.handle.net/11104/0216412 - 4.0343450 - ÚOCHB 2011 RIV US eng J - Journal Article
Gitto, R. - Agnello, S. - Ferro, S. - De Luca, L. - Vullo, D. - Brynda, Jiří - Mader, Pavel - Supuran, C. T. - Chimirri, A.
Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic AnhydraseInhibitors: Synthesis, Biological Evaluation, and Enzyme-Ligand X-ray Studies.
Journal of Medicinal Chemistry. Roč. 53, č. 6 (2010), s. 2401-2408. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR GA203/09/0820
Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50520514
Keywords : inhibitor design * crystal structure * X-ray analysis * dehalogenase
Subject RIV: CC - Organic Chemistry
Impact factor: 5.207, year: 2010
Permanent Link: http://hdl.handle.net/11104/0185928