Search results
- 1.0556370 - FGÚ 2023 RIV FR eng J - Journal Article
Jůza, R. - Vojtěchová, I. - Štefková-Mazochová, K. - Dehaen, W. - Petrásek, T. - Prchal, L. - Kobrlová, T. - Janoušek, J. - Vlček, P. - Mezeiová, E. - Svozil, D. - Zdarová Karasová, J. - Pejchal, J. - Stark, H. - Satala, G. - Bojarski, A. J. - Kubacka, M. - Mogilski, S. - Randáková, Alena - Musílek, K. - Soukup, O. - Korábečný, J.
Novel D-2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
European Journal of Medicinal Chemistry. Roč. 232, Mar 15 (2022), č. článku 114193. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : aripiprazole * cariprazine * dopamine type 2 receptor * drug development * serotonin receptor type 3 * schizophrenia * 1,4-Di-substituted aromatic piperazines * antipsychotic
OECD category: Pharmacology and pharmacy
Impact factor: 6.7, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2022.114193
Permanent Link: http://hdl.handle.net/11104/0330742 - 2.0551558 - ÚEM 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
Institutional support: RVO:68378041
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
OECD category: Medicinal chemistry
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0326821 - 3.0542659 - FGÚ 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
OECD category: Pharmacology and pharmacy
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0320032 - 4.0504524 - FGÚ 2020 RIV FR eng J - Journal Article
Chalupová, K. - Korábečný, J. - Bartolini, M. - Monti, B. - Lamba, D. - Caliandro, R. - Pesaresi, A. - Brazzolotto, X. - Gastellier, A.-J. - Nachon, F. - Pejchal, J. - Jarošová, M. - Hepnarová, V. - Jun, D. - Hrabinová, M. - Doležal, R. - Zdarová Karasová, J. - Mžik, M. - Krištofíková, Z. - Misík, J. - Mucková, L. - Jošt, P. - Soukup, O. - Benková, M. - Setnička, V. - Habartová, L. - Chvojková, Markéta - Kletečková, Lenka - Valeš, Karel - Mezeiová, E. - Uliassi, E. - Vališ, M. - Nepovímová, E. - Bolognesi, M. L. - Kuča, K.
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease.
European Journal of Medicinal Chemistry. Roč. 168, Apr 15 (2019), s. 491-514. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:67985823
Keywords : multi-target directed ligands * Alzheimer's disease * tacrine-tryptophan hybrids * acetylcholinesterase
OECD category: Neurosciences (including psychophysiology
Impact factor: 5.573, year: 2019
Method of publishing: Limited access
https://doi.org/10.1016/j.ejmech.2019.02.021
Permanent Link: http://hdl.handle.net/11104/0296178 - 5.0440989 - FGÚ 2015 RIV CZ eng J - Journal Article
Šepsová, V. - Krůšek, Jan - Zdarová Karasová, J. - Zemek, F. - Musílek, K. - Kuča, K. - Soukup, O.
The interaction of quaternary reversible acetylcholinesterase inhibitors with the nicotinic receptor.
Physiological Research. Roč. 63, č. 6 (2014), s. 771-777. ISSN 0862-8408. E-ISSN 1802-9973
R&D Projects: GA ČR(CZ) GBP304/12/G069
Institutional support: RVO:67985823
Keywords : acetylcholinesterase inhibitor * nicotin receptor
Subject RIV: ED - Physiology
Impact factor: 1.293, year: 2014
Permanent Link: http://hdl.handle.net/11104/0244064 - 6.0397542 - FGÚ 2014 RIV NL eng J - Journal Article
Soukup, O. - Jun, D. - Zdarová Karasová, J. - Patočka, J. - Musílek, K. - Korábečný, J. - Krůšek, Jan - Kaniaková, Martina - Šepsová, V. - Mandíková, J. - Trejtnar, F. - Pohanka, M. - Drtinová, L. - Pavlík, M. - Tobin, G. - Kuča, K.
A Resurrection of 7-MEOTA:a comparison with Tacrine.
Current Alzheimer Research. Roč. 10, č. 8 (2013), s. 893-906. ISSN 1567-2050. E-ISSN 1875-5828
R&D Projects: GA ČR(CZ) GA202/09/0806; GA ČR(CZ) GBP304/12/G069
Institutional research plan: CEZ:AV0Z50110509
Institutional support: RVO:67985823
Keywords : 7-Methoxytacrine * acetylcholinesterase inhibitor
Subject RIV: ED - Physiology
Impact factor: 3.796, year: 2013
Permanent Link: http://hdl.handle.net/11104/0225180 - 7.0333208 - ÚCHP 2011 RIV CH eng J - Journal Article
Kuča, K. - Musilová, L. - Paleček, J. - Církva, Vladimír - Paar, M. - Musílek, K. - Hrabinová, M. - Pohanka, M. - Zdarová Karasová, J. - Jun, D.
Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon.
Molecules. Roč. 14, č. 12 (2009), s. 4915-4921. E-ISSN 1420-3049
Grant - others:MO0(CZ) FZV0000604
Institutional research plan: CEZ:AV0Z40720504
Keywords : acetylcholinesterase * reactivator * oxime
Subject RIV: CC - Organic Chemistry
Impact factor: 1.738, year: 2009
Permanent Link: http://hdl.handle.net/11104/0178252