Search results
- 1.0379112 - FGÚ 2013 RIV GB eng J - Journal Article
Borovská, Jiřina - Vyklický, Vojtěch - Šťastná, Eva - Kapras, Vojtěch - Slavíková, Barbora - Horák, Martin - Chodounská, Hana - Vyklický ml., Ladislav
Access of inhibitory neurosteroids to the NMDA receptor.
British Journal of Pharmacology. Roč. 166, č. 3 (2012), s. 1069-1083. ISSN 0007-1188. E-ISSN 1476-5381
R&D Projects: GA ČR(CZ) GA309/07/0271; GA ČR(CZ) GA203/08/1498; GA MŠMT(CZ) 1M0517; GA MŠMT(CZ) LC554; GA ČR(CZ) GAP303/11/0075; GA ČR(CZ) GAP303/12/1464
Grant - others:GA ČR(CZ) GD309/08/H079; GA MŠk(CZ) ED0007/01/01
Program: ED
Institutional research plan: CEZ:AV0Z50110509; CEZ:AV0Z40550506
Keywords : neurosteroids * NMDA receptor * patch-clamp
Subject RIV: ED - Physiology
Impact factor: 5.067, year: 2012
Permanent Link: http://hdl.handle.net/11104/0210378 - 2.0364480 - FGÚ 2012 RIV NL eng J - Journal Article
Rambousek, Lukáš - Bubeníková-Valešová, V. - Kačer, P. - Syslová, K. - Kenney, Jana - Holubová, Kristína - Najmanová, V. - Zach, P. - Svoboda, Jan - Stuchlík, Aleš - Chodounská, Hana - Kapras, Vojtěch - Adamusová, Eva - Borovská, Jiřina - Vyklický ml., Ladislav - Valeš, Karel
Cellular and behavioural effects of a new steroidal inhibitor of the N-methyl-d-aspartate receptor 3α5β-pregnanolone glutamate.
Neuropharmacology. Roč. 61, 1-2 (2011), s. 61-68. ISSN 0028-3908. E-ISSN 1873-7064
R&D Projects: GA MZd(CZ) NS10365; GA MZd(CZ) NR9180; GA ČR(CZ) GA309/07/0271; GA ČR(CZ) GA203/08/1498; GA ČR(CZ) GA309/09/0286; GA MŠMT(CZ) 1M0517; GA MŠMT(CZ) LC554
Grant - others:EC(XE) LSMH-CT-2007-037765
Institutional research plan: CEZ:AV0Z50110509; CEZ:AV0Z40550506
Keywords : neuroactive steroid * NMDA * neuroprotectivity
Subject RIV: FH - Neurology
Impact factor: 4.814, year: 2011
Permanent Link: http://hdl.handle.net/11104/0199958 - 3.0363595 - ÚOCHB 2012 RIV CZ eng J - Journal Article
Šťastná, Eva - Chodounská, Hana - Pouzar, Vladimír - Borovská, Jiřina - Vyklický ml., Ladislav
Synthesis of pregnane 3-carboxylic acids via Pd-catalyzed alkoxycarbonylation and their effect on NMDA receptor activity.
Collection of Czechoslovak Chemical Communications. Roč. 76, č. 9 (2011), s. 1141-1161. ISSN 0010-0765
R&D Projects: GA ČR(CZ) GA203/08/1498; GA ČR(CZ) GA309/07/0271
Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50110509
Keywords : neurosteroids * carboxylic acid * alkoxycarbonylation * steroids * NMDA receptor activity
Subject RIV: CC - Organic Chemistry
Impact factor: 1.283, year: 2011
Permanent Link: http://hdl.handle.net/11104/0199354 - 4.0361126 - ÚOCHB 2012 RIV US eng J - Journal Article
Vidrna, Lukáš - Černý, Ivan - Pouzar, Vladimír - Borovská, Jiřina - Vyklický, Vojtěch - Vyklický ml., Ladislav - Chodounská, Hana
Azido analogs of neuroactive steroids.
Steroids. Roč. 76, 10/11 (2011), s. 1043-1050. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA MŠMT(CZ) LC06077; GA MŠMT(CZ) LC554; GA ČR(CZ) GA203/08/1498; GA ČR(CZ) GA309/07/0271
Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50110509
Keywords : neuroactive steroids * synthesis * azides * NMDA receptor
Subject RIV: CC - Organic Chemistry
Impact factor: 2.829, year: 2011
Permanent Link: http://hdl.handle.net/11104/0198523 - 5.0352522 - FGÚ 2011 RIV CZ cze J - Journal Article
Valeš, Karel - Rambousek, Lukáš - Stuchlík, Aleš - Chodounská, Hana - Vyklický ml., Ladislav
Srovnání vlivu systémové aplikace non-kompetitivních a use-dependentních NMDA antagonistů na lokomoční aktivitu a kognitivní funkce u laboratorního potkana.
[Comparison of effects of systemic application of non-competitive and use-dependent NMDA antagonists on the locomotor aktivity and cognitive function in the laboratory rat.]
Psychiatrie. Roč. 14, Suppl.2 (2010), s. 26-30. ISSN 1211-7579
R&D Projects: GA MŠMT(CZ) 1M0517; GA MZd(CZ) NR9180; GA MZd(CZ) NS10365; GA ČR(CZ) GA203/08/1498
Institutional research plan: CEZ:AV0Z50110509; CEZ:AV0Z40550506
Keywords : NMDA receptor * glutamate excitotoxicity * NMDA antagonists
Subject RIV: FH - Neurology
Permanent Link: http://hdl.handle.net/11104/0192013 - 6.0346335 - ÚOCHB 2011 RIV FR eng J - Journal Article
Dansey, M. V. - Di Chenna, P. - Valeiro, A. S. - Krištofíková, Z. - Chodounská, Hana - Kasal, Alexander - Burton, G.
Synthesis and GABAA receptor activity of A-homo analogues of neuroactive steroids.
European Journal of Medicinal Chemistry. Roč. 45, č. 7 (2010), s. 3063-3069. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA203/08/1498
Institutional research plan: CEZ:AV0Z40550506
Keywords : A-homopregnane * neurosteroid * gamma-aminobutyric acid * GABAA receptor
Subject RIV: CC - Organic Chemistry
Impact factor: 3.193, year: 2010
Permanent Link: http://hdl.handle.net/11104/0187392 - 7.0345044 - ÚOCHB 2011 RIV US eng J - Journal Article
Šťastná, Eva - Černý, Ivan - Pouzar, Vladimír - Chodounská, Hana
Stereoselectivity of sodium borohydride reduction of saturated steroidal ketones utilizing conditions of Luche reduction.
Steroids. Roč. 75, č. 10 (2010), s. 721-725. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA ČR(CZ) GA203/08/1498; GA MŠMT(CZ) LC06077
Institutional research plan: CEZ:AV0Z40550506
Keywords : steroid * synthesis * stereoselectivity
Subject RIV: CC - Organic Chemistry
Impact factor: 3.106, year: 2010
Permanent Link: http://hdl.handle.net/11104/0186411 - 8.0328948 - FGÚ 2010 RIV GB eng J - Journal Article
Petrovič, Miloš - Sedláček, Miloslav - Cais, Ondřej - Horák, Martin - Chodounská, Hana - Vyklický ml., Ladislav
Pregnenolone sulfate modulation of N-methyl-d-aspartate receptors is phosphorylation dependent.
[Modulace N-methyl-D-aspartátových receptorů pregnenolonsulfátem je závislá na fosforylaci.]
Neuroscience. Roč. 160, č. 3 (2009), s. 616-628. ISSN 0306-4522. E-ISSN 1873-7544
R&D Projects: GA ČR(CZ) GA309/07/0271; GA ČR(CZ) GA203/08/1498; GA MŠMT(CZ) LC554; GA MŠMT(CZ) 1M0517
Grant - others:EC(XE) LSHM-CT-2007-037765
Institutional research plan: CEZ:AV0Z50110509; CEZ:AV0Z40550506
Keywords : NMDA * patch-clamp * phosphorylation
Subject RIV: ED - Physiology
Impact factor: 3.292, year: 2009
Permanent Link: http://hdl.handle.net/11104/0175120 - 9.0324227 - ÚOCHB 2009 RIV CZ eng J - Journal Article
Kapras, Vojtěch - Šťastná, Eva - Chodounská, Hana - Pouzar, Vladimír - Krištofíková, Zdena
Preparation of steroid sulfamates and their interaction with GABAA receptor.
[Příprava steroidních sulfamátů a jejich interakce s MNDA receptory.]
Collection of Czechoslovak Chemical Communications. Roč. 74, č. 4 (2009), s. 643-650. ISSN 0010-0765
R&D Projects: GA ČR(CZ) GA203/08/1498
Institutional research plan: CEZ:AV0Z40550506
Keywords : sulfamates * neurosteroids * GABAA receptors * pregnane
Subject RIV: CC - Organic Chemistry
Impact factor: 0.856, year: 2009
Permanent Link: http://hdl.handle.net/11104/0171978 - 10.0323768 - ÚOCHB 2009 RIV US eng J - Journal Article
Šťastná, Eva - Chodounská, Hana - Pouzar, Vladimír - Kapras, Vojtěch - Borovská, Jiřina - Cais, Ondřej - Vyklický ml., Ladislav
Synthesis of C3, C5, and C7 pregnane derivatives and their effect on NMDA receptor responses in cultured rat hippocampal neurons.
[Syntéza C3, C5 a C7 pregnanových derivátů a jejich vliv na NMDA receptory v kultuře krysích hipokampálních neuronů.]
Steroids. Roč. 74, č. 2 (2009), s. 256-263. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA ČR(CZ) GA309/07/0271; GA ČR(CZ) GA203/08/1498
Grant - others:GA MŠk(CZ) LC554; FP6 Photolysis(XE) LSHM-CT-2007-037765
Program: LC
Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50110509
Keywords : pregnane derivatives * NMDA receptor * structure-activity relationship * patch-clamp recording
Subject RIV: CC - Organic Chemistry
Impact factor: 2.905, year: 2009
Permanent Link: http://hdl.handle.net/11104/0171628