Search results
- 1.0568179 - ÚOCHB 2023 GB eng A - Abstract
Brynda, Jiří - Kugler, Michael - Nekvinda, Jan - Holub, Josef - El Anwar, Suzan - Das, V. - Šícha, Václav - Pospíšilová, Klára - Fábry, Milan - Král, Vlastimil - Pachl, Petr - Hajdúch, M. - Grüner, Bohumír - Řezáčová, Pavlína
Structure-assisted design of inhibitors of CA IX enzyme based on polyhedral boron compounds.
Acta Crystallographica Section A-Foundation and Advances. Oxford Blackwell. Roč. 77 (2021), C864-C864. ISSN 2053-2733. E-ISSN 2053-2733
Institutional support: RVO:61388963 ; RVO:61388980 ; RVO:68378050
Keywords : carborane * cobal bis(dicarbollide) * carbonic anhydrase * enzyme inhibition * SAR study
https://journals.iucr.org/a/issues/2021/a2/00/a60441/a60441.pdf
Permanent Link: https://hdl.handle.net/11104/0339514 - 2.0521902 - ÚACH 2020 FR eng A - Abstract
Olejniczak, A. B. - Rózycka, D. - Rykowski, S. - Nekvinda, Jan - Grüner, Bohumír - Lesnikowski, Z. J. - Wyszko, E. - Fedoruk-Wyszomirska, A. - Gurda, D. - Orlicka Plocka, M. - Giel-Pietraszuk, M. - Kiliszek, A. - Rypniewski, W. - Kolodziej, P. - Ziaja-Soltys, M. - Bogucka-Kocka, A.
Compounds with carborane and matallacarborane components with antibacterial, anticancer, and antihelmintic activity.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "IL5".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
Institutional support: RVO:61388980
Keywords : metallacarborane
OECD category: Inorganic and nuclear chemistry
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306448 - 3.0521900 - ÚACH 2020 FR eng A - Abstract
El Anwar, Suzan - Assaf, K. - Begaj, B. - Gabel, D. - Grüner, Bohumír
N-alkylations of nonahalogenated 2-ammoniodecaborate anion and their complexation with gamma Cyclodextrin.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "P4".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
R&D Projects: GA ČR(CZ) GA19-04630S
Grant - others:AV ČR(CZ) DAAD-17-22
Program: Bilaterální spolupráce
Institutional support: RVO:61388980
Keywords : dodecaborate
OECD category: Inorganic and nuclear chemistry
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306834 - 4.0521898 - ÚACH 2020 FR eng A - Abstract
Nekvinda, Jan - Holub, Josef - Brynda, Jiří - Pospíšilová, Klára - Řezáčová, Pavlína - Grüner, Bohumír
Alkylsulfonamido carboranes: the isomer dependence observed in inhibitory activity towards Carbonic Anhydrase IX.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "O48".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
R&D Projects: GA ČR(CZ) GA15-05677S; GA ČR(CZ) GA18-27648S
Institutional support: RVO:61388980 ; RVO:68378050
Keywords : Carbonic Anhydrase
OECD category: Inorganic and nuclear chemistry; Biochemistry and molecular biology (UMG-J)
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306442 - 5.0521897 - ÚACH 2020 FR eng A - Abstract
Bednarska-Szczepaniak, K. - Przelazly, E. - Grüner, Bohumír - Lesnikowski, Z. J.
Metallacarborane-modified adenine nucleosides. Synthesis and effect on chemo-resistance of cancer cells against cisplatin.
EuroBoron 8 : program and abstracts. Montpellier: IEM, 2019. "P36".
[European Conference on Boron Chemistry /8./. 24.06.2019-27.06.2019, Montpellier]
Institutional support: RVO:61388980
Keywords : metallacarborane
OECD category: Inorganic and nuclear chemistry
http://euroboron8.org/WP/program/
Permanent Link: http://hdl.handle.net/11104/0306441 - 6.0520890 - ÚOCHB 2020 GB eng A - Abstract
Řezáčová, Pavlína - Kugler, Michael - Brynda, Jiří - Grüner, Bohumír - Hajdúch, M. - Nekvinda, Jan - Pospíšilová, Klára - Das, V. - Holub, Josef
Structure-assisted design of Carborane inhibitors of human Carbonic anhydrase IX.
Acta Crystallographica Section A-Foundation and Advances. Oxford Blackwell. Roč. 74, Suppl (2018), „e197“. ISSN 2053-2733. E-ISSN 2053-2733.
[European Crystallography Meeting /31./. 22.08.2018-27.08.2018, Oviedo]
R&D Projects: GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LO1304; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : anti-tumor agents * carborane inhibitors * Carbonic anhydrase IX
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Permanent Link: http://hdl.handle.net/11104/0305557 - 7.0501881 - ÚOCHB 2019 GB eng A - Abstract
Brynda, Jiří - Řezáčová, Pavlína - Fábry, Milan - Štěpánková, J. - Král, Vlastimil - Hajdúch, M. - Holub, Josef - Nekvinda, Jan - Pospíšilová, Klára - Kugler, Michael - Grüner, Bohumír
Carborane and metallacarborane inhibitors of carbonic anhydrase IX, promising compounds for cancer therapy.
FEBS Open Bio. Wiley. Roč. 8, Suppl 1 (2018), s. 438. ISSN 2211-5463. E-ISSN 2211-5463.
[FEBS Congress /43./ Biochemistry Forever. 07.07.2018-12.07.2018, Prague]
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : carbonic anhydrase IX * inhibitors
OECD category: Biochemistry and molecular biology
Permanent Link: http://hdl.handle.net/11104/0293863 - 8.0501879 - ÚOCHB 2019 GB eng A - Abstract
Kugler, Michael - Brynda, Jiří - Řezáčová, Pavlína - Fábry, Milan - Král, Vlastimil - Pospíšilová, Klára - Holub, Josef - Šícha, Václav - Nekvinda, Jan - Grüner, Bohumír
Structure-based design of human carbonic anhydrase XII inhibitors.
FEBS Open Bio. Wiley. Roč. 8, Suppl 1 (2018), s. 426-427. ISSN 2211-5463. E-ISSN 2211-5463.
[FEBS Congress /43./ Biochemistry Forever. 07.07.2018-12.07.2018, Prague]
Institutional support: RVO:61388963 ; RVO:68378050 ; RVO:61388980
Keywords : carbonic anhydrase XII * inhibitors
OECD category: Biochemistry and molecular biology
Permanent Link: http://hdl.handle.net/11104/0293860 - 9.0493641 - ÚOCHB 2019 SK eng A - Abstract
Šolínová, Veronika - Holub, Josef - Grüner, Bohumír - Kašička, Václav
Determination of acidity constants and ionic mobilities of polyhalogenated 2-ammonium-decaborate and 1-ammonium-dodecaborate anions by capillary electrophoresis.
24th International Symposium on Separation Sciences (ISSS 2018) and 21st International Conference Analytical Methods and Human Health (AMHH 2018). Bratislava: Comenius University in Bratislava, 2018 - (Hutta, M.; Bodor, R.; Halko, R.). s. 143. ISBN 978-80-971179-8-6.
[International Symposium on Separation Sciences (ISSS 2018) /24./ and International Conference Analytical Methods and Human Health (AMHH 2018) /21./. 17.06.2018-20.06.2018, Jasná]
R&D Projects: GA ČR(CZ) GA17-10832S; GA ČR(CZ) GA18-02597S
Institutional support: RVO:61388963 ; RVO:61388980
Keywords : capillary electrophoresis * acidity constant * polyhalogenated 2-ammonium-decaborate
OECD category: Analytical chemistry
Permanent Link: http://hdl.handle.net/11104/0286972 - 10.0491273 - ÚOCHB 2019 CZ eng A - Abstract
Srb, Pavel - Svoboda, Michal - Benda, L. - Lepšík, Martin - Tarábek, Ján - Šícha, Václav - Grüner, Bohumír - Grantz Šašková, Klára - Brynda, Jiří - Řezáčová, Pavlína - Konvalinka, Jan - Veverka, Václav
Capturing dynamically interacting inhibitor by paramagnetic NMR spectroscopy.
Prague Protein Spring Meeting 2018: Proteins at Work. Praha: Ústav organické chemie a biochemie AV ČR, 2018 - (Votrubová, T.; Pergl Šustková, H.; Vondrášek, J.). s. 70. ISBN 978-80-86241-58-6.
[Prague Protein Spring Meeting 2018: Proteins at Work. 03.05.2018-06.05.2018, Praha]
Institutional support: RVO:61388963 ; RVO:61388980
Keywords : paramagnetic ligands * intermolecular interactions * HIV-1 protease
OECD category: Biochemistry and molecular biology
Permanent Link: http://hdl.handle.net/11104/0285577