Search results
- 1.0539170 - ÚMG 2021 RIV GB eng J - Journal Article
Kugler, Michael - Holub, J. - Brynda, Jiří - Pospíšilová, K. - El Anwar, S. - Bavol, D. - Havránek, M. - Král, Vlastimil - Fábry, Milan - Gruner, B. - Řezáčová, Pavlína
The structural basis for the selectivity of sulfonamido dicarbaboranes toward cancer-associated carbonic anhydrase IX.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 35, č. 1 (2020), s. 1800-1810. ISSN 1475-6366. E-ISSN 1475-6374
Institutional support: RVO:68378050
Keywords : tumor hypoxia * medicinal chemistry * drug discovery * binding-sites * inhibition * boron * pharmacophores * opportunities * conjugation * metastasis * Carbonic anhydrase IX * carborane * enzyme inhibitors * structure-activity relationship
OECD category: Biochemistry and molecular biology
Impact factor: 5.051, year: 2020
Method of publishing: Open access
https://www.tandfonline.com/doi/full/10.1080/14756366.2020.1816996
Permanent Link: http://hdl.handle.net/11104/0316870 - 2.0538151 - ÚFP 2021 RIV GB eng J - Journal Article
Novotný, L. - Čeřovský, Jaroslav - Dhyani, P. - Ficker, O. - Havránek, M. - Hejtmánek, M. - Janoška, Z. - Kafka, V. - Kulkov, S. - Marčišovská, M. - Marcisovský, M. - Neue, G. - Svihra, P. - Svoboda, V. - Tomášek, L. - Tunkl, M. - Vrba, V.
Runaway electron diagnostics using silicon strip detector.
Journal of Instrumentation. Roč. 15, č. 7 (2020), č. článku C07015. ISSN 1748-0221. E-ISSN 1748-0221
R&D Projects: GA ČR(CZ) GA18-02482S
Institutional support: RVO:61389021
Keywords : Runaway electrons * silicon strip detector
OECD category: Fluids and plasma physics (including surface physics)
Impact factor: 1.415, year: 2020
Method of publishing: Limited access
https://iopscience.iop.org/article/10.1088/1748-0221/15/07/C07015/pdf
Permanent Link: http://hdl.handle.net/11104/0315973 - 3.0538009 - FZÚ 2021 RIV GB eng J - Journal Article
Marčišovská, M. - Dudas, D. - Havránek, M. - Kabátová, A. - Kafka, V. - Kostina, A. - Macková, A. - Marcisovský, M. - Mitrofanov, S. V. - Popule, Jiří - Romanenko, Oleksandr V. - Tomášek, L. - Vrba, V.
TID and SEU testing of the novel X-CHIP-03 monolithic pixel detector.
Journal of Instrumentation. Roč. 15, č. 1 (2020), s. 1-11, č. článku C01043. ISSN 1748-0221. E-ISSN 1748-0221
R&D Projects: GA MŠMT EF16_013/0001812
Institutional support: RVO:68378271 ; RVO:61389005
Keywords : radiation damage to detector materials (solid state) * radiation damage to electronic components * radiation-hard detectors * radiation-hard electronics
OECD category: Particles and field physics; Nuclear physics (UJF-V)
Impact factor: 1.415, year: 2020
Method of publishing: Limited access
https://doi.org/10.1088/1748-0221/15/01/C01043
Permanent Link: http://hdl.handle.net/11104/0315849 - 4.0533528 - ÚOCHB 2021 RIV US eng J - Journal Article
Dosoudil, P. - Kotek, V. - Kolman, Viktor - Baszczyňski, Ondřej - Kaiser, Martin Maxmilian - Janeba, Zlatko - Havránek, M.
Development of Scalable Synthesis of 5-Butyl-4-(4-methoxyphenyl)-6-phenylpyrimidin-2-amine (WQE-134), a Dual Inhibitor of Nitric Oxide and Prostaglandin E2 Production.
Organic Process Research & Development. Roč. 24, č. 9 (2020), s. 1718-1724. ISSN 1083-6160. E-ISSN 1520-586X
R&D Projects: GA TA ČR(CZ) TE01020028
Institutional support: RVO:61388963
Keywords : pyrimidines * Eaton’s reagent * upscale * C-acylation
OECD category: Organic chemistry
Impact factor: 3.317, year: 2020
Method of publishing: Limited access
https://doi.org/10.1021/acs.oprd.0c00324
Permanent Link: http://hdl.handle.net/11104/0312366 - 5.0532715 - ÚOCHB 2021 RIV GB eng J - Journal Article
Kugler, Michael - Holub, Josef - Brynda, Jiří - Pospíšilová, Klára - El Anwar, Suzan - Bavol, Dmytro - Havránek, M. - Král, V. - Fábry, M. - Grüner, Bohumír - Řezáčová, Pavlína
The structural basis for the selectivity of sulfonamido dicarbaboranes toward cancer-associated carbonic anhydrase IX.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 35, č. 1 (2020), s. 1800-1810. ISSN 1475-6366. E-ISSN 1475-6374
R&D Projects: GA ČR(CZ) GA18-27648S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) EF16_019/0000729
Grant - others:AV ČR(CZ) L200321851
Program: Program podpory perspektivníchlidských zdrojů - postdoktorandů
Institutional support: RVO:61388963 ; RVO:61388980
Keywords : carbonic anhydrase IX * carbone * enzyme inhibitors * sulfonamide * structure-activity relationship
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Impact factor: 5.051, year: 2020
Method of publishing: Open access
https://doi.org/10.1080/14756366.2020.1816996
Permanent Link: http://hdl.handle.net/11104/0311123File Download Size Commentary Version Access The structural basis for the selectivity of sulfonamido dicarbaboranes toward cancer associated carbonic anhydrase IX.pdf 2 3.7 MB Publisher’s postprint open-access - 6.0531266 - ÚMG 2021 RIV FR eng J - Journal Article
Dvořanová, J. - Kugler, Michael - Holub, J. - Šícha, V. - Das, V. - Nekvinda, J. - El Anwar, S. - Havránek, M. - Pospíšilová, K. - Fábry, Milan - Král, Vlastimil - Medvědiková, M. - Matějková, S. - Lišková, B. - Gurská, S. - Dzubak, P. - Brynda, Jiří - Hajduch, M. - Gruner, B. - Řezáčová, P.
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
European Journal of Medicinal Chemistry. Roč. 200, August (2020), č. článku 112460. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA15-05677S
Institutional support: RVO:68378050
Keywords : Anti-tumor agents * Carbonic anhydrase IX * Carboranes * Dicarbollide * Enzyme inhibitors * Drug penetration * Multicellular spheroids
OECD category: Medicinal chemistry
Impact factor: 6.514, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/abs/pii/S0223523420304311?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0309958 - 7.0524603 - ÚOCHB 2021 RIV FR eng J - Journal Article
Dvořanová, J. - Kugler, Michael - Holub, Josef - Šícha, Václav - Das, V. - Nekvinda, Jan - El Anwar, Suzan - Havránek, M. - Pospíšilová, Klára - Fábry, M. - Král, V. - Medvedíková, M. - Matějková, Stanislava - Lišková, B. - Gurská, S. - Džubák, P. - Brynda, J. - Hajdúch, M. - Grüner, Bohumír - Řezáčová, Pavlína
Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX.
European Journal of Medicinal Chemistry. Roč. 200, Aug 15 (2020), č. článku 112460. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA18-27648S; GA ČR(CZ) GA15-05677S; GA TA ČR(CZ) TE01020028; GA MŠMT(CZ) LM2015064
Grant - others:AV ČR(CZ) L200321851
Program: Program podpory perspektivníchlidských zdrojů - postdoktorandů
Institutional support: RVO:61388963 ; RVO:61388980
Keywords : anti-tumor agents * carbonic anhydrase IX * carboranes * dicarbollide * enzyme inhibitors * drug penetration * multicellular spheroids
OECD category: Biochemistry and molecular biology; Inorganic and nuclear chemistry (UACH-T)
Impact factor: 6.514, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S0223523420304311?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0308946 - 8.0523138 - ÚACH 2021 RIV CH eng J - Journal Article
Havránek, M. - Samsonov, M. A. - Holub, Josef - Růžičková, Z. - Drož, L. - Růžička, A. - Fanfrlík, Jindřich - Hnyk, Drahomír
The influence of halogenated hypercarbon on crystal packing in the series of 1-Ph-2-X-1,2-dicarba-closo-dodecaboranes (X = F, Cl, Br, I).
Molecules. Roč. 25, č. 5 (2020), č. článku 1200. E-ISSN 1420-3049
R&D Projects: GA ČR(CZ) GA19-17156S
Institutional support: RVO:61388980 ; RVO:61388963
Keywords : Halogen bond * Icosahedral boron cluster * Sigma hole
OECD category: Inorganic and nuclear chemistry; Organic chemistry (UOCHB-X)
Impact factor: 4.412, year: 2020
Method of publishing: Open access
Permanent Link: http://hdl.handle.net/11104/0307530File Download Size Commentary Version Access 0523138.pdf 1 2.8 MB CC 4.0 licence Publisher’s postprint open-access - 9.0509566 - ÚFP 2020 RIV NL eng J - Journal Article
Svihra, P. - Břeň, D. - Casolari, Andrea - Čeřovský, Jaroslav - Dhyani, P. - Farník, Michal - Ficker, Ondřej - Havránek, M. - Hejtmanek, M. - Janoška, Z. - Kafka, V. - Kulhánek, Petr - Linhart, V. - Tomešová, Eva - Marčišovská, M. - Marcisovský, M. - Mlynář, Jan - Neue, G. - Novotný, L. - Svoboda, V. - Tomášek, L. - Urban, Jakub - Vančura, P. - Varju, Jozef - Vrba, V. - Weinzettl, Vladimír
Runaway electrons diagnostics using segmented semiconductor detectors.
Fusion Engineering and Design. Roč. 146, September (2019), s. 316-319. ISSN 0920-3796. E-ISSN 1873-7196
R&D Projects: GA ČR(CZ) GA18-02482S; GA MŠMT(CZ) LM2015045
Institutional support: RVO:61389021
Keywords : Runaway electrons * Semiconductor detectors * Tokamaks
OECD category: Fluids and plasma physics (including surface physics)
Impact factor: 1.692, year: 2019
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/abs/pii/S0920379618308196?via%3Dihub
Permanent Link: http://hdl.handle.net/11104/0300275 - 10.0501816 - FZÚ 2019 RIV GB eng J - Journal Article
Havránek, M. - Benka, T. - Hejtmanek, M. - Janoška, Z. - Kafka, Z. - Kopeček, Jaromír - Kuklová, M. - Marčišovská, M. - Marcisovský, M. - Neue, G. - Svihra, P. - Tomášek, L. - Vančura, P. - Vrba, V.
MAPS sensor for radiation imaging designed in 180 nm SOI CMOS technology.
Journal of Instrumentation. Roč. 13, č. 6 (2018), s. 1-10, č. článku C06004. ISSN 1748-0221. E-ISSN 1748-0221
R&D Projects: GA MŠMT LM2015058
Institutional support: RVO:68378271
Keywords : active pixel sensor * X-ray detectors
OECD category: Nuclear physics
Impact factor: 1.366, year: 2018
Permanent Link: http://hdl.handle.net/11104/0293800