Search results

  1. 1.
    0385940 - ÚOCHB 2013 RIV US eng J - Journal Article
    Schimer, Jiří - Cígler, Petr - Veselý, J. - Grantz Šašková, Klára - Lepšík, Martin - Brynda, Jiří - Řezáčová, Pavlína - Kožíšek, Milan - Císařová, I. - Oberwinkler, H. - Kraeusslich, H. G. - Konvalinka, Jan
    Structure-Aided Design of Novel Inhibitors of HIV Protease Based on a Benzodiazepine Scaffold.
    Journal of Medicinal Chemistry. Roč. 55, č. 22 (2012), s. 10130-10135. ISSN 0022-2623. E-ISSN 1520-4804
    R&D Projects: GA ČR GBP208/12/G016; GA ČR GAP207/11/1798
    Institutional research plan: CEZ:AV0Z40550506; CEZ:AV0Z50520514
    Keywords : HIV protease inhibitor * rational drug design * 1,4-benzodiazepines
    Subject RIV: CE - Biochemistry
    Impact factor: 5.614, year: 2012
    Permanent Link: http://hdl.handle.net/11104/0215861
     
     
  2. 2.
    0194573 - UOCHB-X 20020244 RIV GB eng J - Journal Article
    Weber, Jan - Mesters, J. R. - Lepšík, Martin - Prejdová, Jana - Švec, Martin - Šponarová, Jana - Mlčochová, Petra - Skalická, Kristina - Stříšovský, Kvido - Kondrová, Taťána - Souček, Milan - Machala, L. - Staňková, M. - Vondrášek, Jiří - Klimkait, T. - Kraeusslich, H. G. - Hilgenfeld, R. - Konvalinka, Jan
    Unusual binding mode of an HIV-1 protease inhibitor explains its potency against multi-grug-resistant virus strains.
    Journal of Molecular Biology. Roč. 324, - (2002), s. 739-754. ISSN 0022-2836. E-ISSN 1089-8638
    R&D Projects: GA ČR GA203/00/0828; GA MŠMT LN00A032; GA MZd NI6339
    Institutional research plan: CEZ:AV0Z4055905
    Keywords : HIV protease inhibitor
    Subject RIV: CE - Biochemistry
    Impact factor: 5.359, year: 2002
    Permanent Link: http://hdl.handle.net/11104/0090248
     
     
  3. 3.
    0192940 - UOCHB-X 970313 RIV US eng J - Journal Article
    Pichová, Iva - Weber, Jan - Litera, Jaroslav - Konvalinka, Jan - Vondrášek, Jiří - Souček, Milan - Štrop, Petr - Majer, Pavel - Heuser, A. E. - Kraeusslich, H. G.
    Peptide Inhibitors of HIV-2 Proteases: A Comparative Study.
    Leukemia. Roč. 11, č. 3 (1997), s. 120-122. ISSN 0887-6924. E-ISSN 1476-5551
    R&D Projects: GA ČR GA303/96/1235; GA AV ČR IAA4055503
    Impact factor: 1.046, year: 1997
    Permanent Link: http://hdl.handle.net/11104/0088659
     
     


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