Search results
- 1.0494693 - ÚMG 2019 RIV GB eng J - Journal Article
Jurasek, M. - Černohorská, Markéta - Řehulka, J. - Spiwok, V. - Sulimenko, Tetyana - Dráberová, Eduarda - Darmostuk, M. - Gurska, S. - Frydrych, I. - Burianova, R. - Ruml, T. - Hajduch, M. - Bartůněk, Petr - Dráber, Pavel - Dzubak, P. - Drašar, P. B. - Sedlák, David
Estradiol dimer inhibits tubulin polymerization and microtubule dynamics.
Journal of Steroid Biochemistry and Molecular Biology. Roč. 183, Říjen (2018), s. 68-79. ISSN 0960-0760
R&D Projects: GA MŠMT LO1220; GA MŠMT(CZ) LO1304; GA MŠMT LM2015063; GA ČR GA15-22194S; GA ČR GA16-25159S
Institutional support: RVO:68378050
Keywords : Steroid dimer * Steroid receptor * Luciferase reporter assay * Microtubules * Microtubule dynamics * Tubulin assembly * Molecular dynamics simulation * Antimitotic activity
OECD category: Cell biology
Impact factor: 3.785, year: 2018
Permanent Link: http://hdl.handle.net/11104/0287788 - 2.0473082 - ÚMG 2017 RIV US eng J - Journal Article
Jurášek, M. - Džubák, P. - Rimpelová, S. - Sedlák, David - Konečný, P. - Frydrych, I. - Gurska, S. - Hajdúch, M. - Bogdanová, K. - Kolář, M. - Muller, Tomáš - Kmoníčková, Eva - Ruml, T. - Harmatha, Juraj - Drašar, P. B.
Trilobolide-steroid hybrids: Synthesis, cytotoxic and antimycobacterial activity.
Steroids. Roč. 117, JAN (2017), s. 97-104. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA MŠMT(CZ) LO1304; GA MŠMT LO1220; GA MŠMT LM2015063
Grant - others:GA ČR(CZ) GA14-04329S
Institutional support: RVO:68378050 ; RVO:68378041 ; RVO:61388963
Keywords : Trilobolide * Steroids * Click chemistry * Cytotoxicity * sar * Steroid receptor
OECD category: Biochemistry and molecular biology; Organic chemistry (UOCHB-X)
Impact factor: 2.523, year: 2017
Permanent Link: http://hdl.handle.net/11104/0270248 - 3.0423021 - ÚMG 2014 RIV US eng J - Journal Article
Jurášek, M. - Džubák, P. - Sedlák, David - Dvořáková, H. - Hajduch, M. - Bartůněk, Petr - Drasar, P.
Preparation, preliminary screening of new types of steroid conjugates and their activities on steroid receptors.
Steroids. Roč. 78, č. 3 (2013), s. 356-361. ISSN 0039-128X. E-ISSN 1878-5867
R&D Projects: GA MŠMT(CZ) LC06077; GA ČR(CZ) GAP503/11/0616; GA ČR(CZ) GAP304/10/1951
Institutional support: RVO:68378050
Keywords : click chemistry * steroid ribbons * cytotoxic activity * steroid receptor reporter assay * 2,6-bis((1H-1,2,3-triazol-1-yl)methyl)pyridine
Subject RIV: EB - Genetics ; Molecular Biology
Impact factor: 2.716, year: 2013
Permanent Link: http://hdl.handle.net/11104/0229188 - 4.0365123 - ÚMG 2012 RIV NL eng J - Journal Article
Sedlák, David - Paguio, A. - Bartůněk, Petr
Two panels of steroid receptor luciferase reporter cell lines for compound profiling.
Combinatorial Chemistry & High Throughput Screening. Roč. 14, č. 2 (2011), s. 248-266. ISSN 1386-2073. E-ISSN 1875-5402
R&D Projects: GA MŠMT(CZ) LC06077
Institutional research plan: CEZ:AV0Z50520514
Keywords : nuclear hormone receptor * steroid receptor * cell-based luciferase reporter assay
Subject RIV: EB - Genetics ; Molecular Biology
Impact factor: 1.785, year: 2011
Permanent Link: http://hdl.handle.net/11104/0200439