Search results
- 1.0570624 - ÚEM 2024 RIV GB eng J - Journal Article
Kolcheva, Marharyta - Ladislav, Marek - Netolický, Jakub - Kortus, Štěpán - Řeháková, Kristýna - Hrčka Krausová, Barbora - Hemeliková, Katarina - Misiachna, Anna - Kádková, Anna - Klíma, M. - Chalupská, D. - Horák, Martin
The pathogenic N650K variant in the GluN1 subunit regulates the trafficking, conductance, and pharmacological properties of NMDA receptors.
Neuropharmacology. Roč. 222, jan. (2023), č. článku 109297. ISSN 0028-3908. E-ISSN 1873-7064
R&D Projects: GA MŠMT(CZ) LX22NPO5107; GA ČR(CZ) GA20-12420S
Institutional support: RVO:68378041
Keywords : glutamate receptor * hippocampal neuron * neurodegeneration * ion channel * ketamine * memantine
OECD category: Neurosciences (including psychophysiology
Impact factor: 4.7, year: 2022
Method of publishing: Open access
https://doi.org/10.1016/j.neuropharm.2022.109297
Permanent Link: https://hdl.handle.net/11104/0341931Review Download Size Commentary Version Access Kolcheva 2023.pdf 8 7.8 MB Publisher’s postprint open-access - 2.0566214 - FGÚ 2024 RIV GB eng J - Journal Article
Kolcheva, Marharyta - Ladislav, M. - Netolický, J. - Kortus, Š. - Řeháková, K. - Hrčka Krausová, B. - Hemelíková, K. - Misiachna, A. - Kádková, A. - Klíma, Martin - Chalupská, Dominika - Horák, M.
The pathogenic N650K variant in the GluN1 subunit regulates the trafficking, conductance, and pharmacological properties of NMDA receptors.
Neuropharmacology. Roč. 222, 1 January (2023), č. článku 109297. ISSN 0028-3908. E-ISSN 1873-7064
R&D Projects: GA ČR(CZ) GA20-12420S; GA MŠMT(CZ) LX22NPO5107
Institutional support: RVO:67985823 ; RVO:61388963
Keywords : glutamate receptor * hippocampal neuron * neurodegeneration * ion channel * ketamine * memantine
OECD category: Neurosciences (including psychophysiology
Impact factor: 4.7, year: 2022
Method of publishing: Open access
https://doi.org/10.1016/j.neuropharm.2022.109297
Permanent Link: https://hdl.handle.net/11104/0341691 - 3.0564838 - ÚOCHB 2023 RIV GB eng J - Journal Article
Mustafa, E. R. - Gambeta, E. - Stringer, Robin Nicholas - Souza, I. A. - Zamponi, G. W. - Weiss, N.
Electrophysiological and computational analysis of Cav3.2 channel variants associated with familial trigeminal neuralgia.
Molecular Brain. Roč. 15, č. 1 (2022), č. článku 91. E-ISSN 1756-6606
Institutional support: RVO:61388963
Keywords : trigeminal neuralgia * ion channel * calcium channel * CACNA1H * Cav3 * 2 channel * channelopathy
OECD category: Biochemistry and molecular biology
Impact factor: 3.6, year: 2022
Method of publishing: Open access
https://doi.org/10.1186/s13041-022-00978-9
Permanent Link: https://hdl.handle.net/11104/0336462File Download Size Commentary Version Access 10.1186s13041-022-00978-9.pdf 3 4.7 MB Publisher’s postprint open-access - 4.0556683 - ÚOCHB 2023 RIV NL eng J - Journal Article
Tempra, Carmelo - Scollo, Federica - Pannuzzo, M. - Lolicato, F. - La Rosa, C.
A unifying framework for amyloid-mediated membrane damage: The lipid-chaperone hypothesis.
Biochimica Et Biophysica Acta-Proteins and Proteomics. Roč. 1870, č. 4 (2022), č. článku 140767. ISSN 1570-9639. E-ISSN 1878-1454
R&D Projects: GA ČR(CZ) GX19-26854X
Institutional support: RVO:61388963 ; RVO:61388955
Keywords : amyloid * aggregation * ion channel-like * model membrane * lipid-chaperone * toxic oligomer
OECD category: Physical chemistry
Impact factor: 3.2, year: 2022
Method of publishing: Limited access
https://doi.org/10.1016/j.bbapap.2022.140767
Permanent Link: http://hdl.handle.net/11104/0330806File Download Size Commentary Version Access 0556683.pdf 3 4.4 MB Publisher’s postprint require - 5.0556398 - ÚOCHB 2023 RIV US eng J - Journal Article
Boušová, Kristýna - Zouharová, Monika - Heřman, P. - Vymětal, Jiří - Vetýšková, Veronika - Jirásková, Kateřina - Vondrášek, Jiří
TRPM5 Channel Binds Calcium-Binding Proteins Calmodulin and S100A1.
Biochemistry. Roč. 61, č. 6 (2022), s. 413-423. ISSN 0006-2960
Institutional support: RVO:61388963
Keywords : ion channel * ryanodine receptor * N-terminus
OECD category: Biochemistry and molecular biology
Impact factor: 2.9, year: 2022
Method of publishing: Limited access
https://doi.org/10.1021/acs.biochem.1c00647
Permanent Link: http://hdl.handle.net/11104/0331043 - 6.0551558 - ÚEM 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
Institutional support: RVO:68378041
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
OECD category: Medicinal chemistry
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0326821 - 7.0543492 - ÚEM 2022 RIV US eng J - Journal Article
Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
R&D Projects: GA ČR(CZ) GA20-12047S
Institutional support: RVO:68378041
Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
OECD category: Pharmacology and pharmacy
Impact factor: 6.100, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bcp.2021.114460
Permanent Link: http://hdl.handle.net/11104/0320802 - 8.0543350 - FGÚ 2022 RIV US eng J - Journal Article
Kaniaková, Martina - Korábečný, J. - Holubová, Kristína - Kletečková, Lenka - Chvojková, Markéta - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Krausová, B. - Horák, Martin - Valeš, Karel - Soukup, O.
7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
Biochemical Pharmacology. Roč. 186, Apr (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
OECD category: Pharmacology and pharmacy
Impact factor: 6.100, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.bcp.2021.114460
Permanent Link: http://hdl.handle.net/11104/0320571 - 9.0542659 - FGÚ 2022 RIV FR eng J - Journal Article
Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA MZd(CZ) EF16_025/0007444
Institutional support: RVO:67985823
Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
OECD category: Pharmacology and pharmacy
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113434
Permanent Link: http://hdl.handle.net/11104/0320032 - 10.0542632 - FGÚ 2022 RIV NL eng J - Journal Article
Kolcheva, Marharyta - Kortus, Š. - Hrčka Krausová, B. - Baráčková, P. - Misiachna, A. - Danačíková, Šárka - Kaniaková, M. - Hemelíková, K. - Hotovec, M. - Řeháková, K. - Horák, M.
Specific pathogenic mutations in the M3 domain of the GluN1 subunit regulate the surface delivery and pharmacological sensitivity of NMDA receptors.
Neuropharmacology. Roč. 189, 15 May (2021), č. článku 108528. ISSN 0028-3908. E-ISSN 1873-7064
R&D Projects: GA ČR(CZ) GA20-12420S
Institutional support: RVO:67985823
Keywords : electrophysiology * glutamate receptor * hippocampal neuron * ion channel * memantine * membrane domain
OECD category: Neurosciences (including psychophysiology
Impact factor: 5.273, year: 2021
Method of publishing: Limited access
https://doi.org/10.1016/j.neuropharm.2021.108528
Permanent Link: http://hdl.handle.net/11104/0320020