Search results

  1. 1.
    0570624 - ÚEM 2024 RIV GB eng J - Journal Article
    Kolcheva, Marharyta - Ladislav, Marek - Netolický, Jakub - Kortus, Štěpán - Řeháková, Kristýna - Hrčka Krausová, Barbora - Hemeliková, Katarina - Misiachna, Anna - Kádková, Anna - Klíma, M. - Chalupská, D. - Horák, Martin
    The pathogenic N650K variant in the GluN1 subunit regulates the trafficking, conductance, and pharmacological properties of NMDA receptors.
    Neuropharmacology. Roč. 222, jan. (2023), č. článku 109297. ISSN 0028-3908. E-ISSN 1873-7064
    R&D Projects: GA MŠMT(CZ) LX22NPO5107; GA ČR(CZ) GA20-12420S
    Institutional support: RVO:68378041
    Keywords : glutamate receptor * hippocampal neuron * neurodegeneration * ion channel * ketamine * memantine
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 4.7, year: 2022
    Method of publishing: Open access
    https://doi.org/10.1016/j.neuropharm.2022.109297
    Permanent Link: https://hdl.handle.net/11104/0341931
     
    Review DownloadSizeCommentaryVersionAccess
    Kolcheva 2023.pdf87.8 MBPublisher’s postprintopen-access
     
  2. 2.
    0566214 - FGÚ 2024 RIV GB eng J - Journal Article
    Kolcheva, Marharyta - Ladislav, M. - Netolický, J. - Kortus, Š. - Řeháková, K. - Hrčka Krausová, B. - Hemelíková, K. - Misiachna, A. - Kádková, A. - Klíma, Martin - Chalupská, Dominika - Horák, M.
    The pathogenic N650K variant in the GluN1 subunit regulates the trafficking, conductance, and pharmacological properties of NMDA receptors.
    Neuropharmacology. Roč. 222, 1 January (2023), č. článku 109297. ISSN 0028-3908. E-ISSN 1873-7064
    R&D Projects: GA ČR(CZ) GA20-12420S; GA MŠMT(CZ) LX22NPO5107
    Institutional support: RVO:67985823 ; RVO:61388963
    Keywords : glutamate receptor * hippocampal neuron * neurodegeneration * ion channel * ketamine * memantine
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 4.7, year: 2022
    Method of publishing: Open access
    https://doi.org/10.1016/j.neuropharm.2022.109297
    Permanent Link: https://hdl.handle.net/11104/0341691
     
     
  3. 3.
    0564838 - ÚOCHB 2023 RIV GB eng J - Journal Article
    Mustafa, E. R. - Gambeta, E. - Stringer, Robin Nicholas - Souza, I. A. - Zamponi, G. W. - Weiss, N.
    Electrophysiological and computational analysis of Cav3.2 channel variants associated with familial trigeminal neuralgia.
    Molecular Brain. Roč. 15, č. 1 (2022), č. článku 91. E-ISSN 1756-6606
    Institutional support: RVO:61388963
    Keywords : trigeminal neuralgia * ion channel * calcium channel * CACNA1H * Cav3 * 2 channel * channelopathy
    OECD category: Biochemistry and molecular biology
    Impact factor: 3.6, year: 2022
    Method of publishing: Open access
    https://doi.org/10.1186/s13041-022-00978-9
    Permanent Link: https://hdl.handle.net/11104/0336462
    FileDownloadSizeCommentaryVersionAccess
    10.1186s13041-022-00978-9.pdf34.7 MBPublisher’s postprintopen-access
     
     
  4. 4.
    0556683 - ÚOCHB 2023 RIV NL eng J - Journal Article
    Tempra, Carmelo - Scollo, Federica - Pannuzzo, M. - Lolicato, F. - La Rosa, C.
    A unifying framework for amyloid-mediated membrane damage: The lipid-chaperone hypothesis.
    Biochimica Et Biophysica Acta-Proteins and Proteomics. Roč. 1870, č. 4 (2022), č. článku 140767. ISSN 1570-9639. E-ISSN 1878-1454
    R&D Projects: GA ČR(CZ) GX19-26854X
    Institutional support: RVO:61388963 ; RVO:61388955
    Keywords : amyloid * aggregation * ion channel-like * model membrane * lipid-chaperone * toxic oligomer
    OECD category: Physical chemistry
    Impact factor: 3.2, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bbapap.2022.140767
    Permanent Link: http://hdl.handle.net/11104/0330806
    FileDownloadSizeCommentaryVersionAccess
    0556683.pdf34.4 MBPublisher’s postprintrequire
     
     
  5. 5.
    0556398 - ÚOCHB 2023 RIV US eng J - Journal Article
    Boušová, Kristýna - Zouharová, Monika - Heřman, P. - Vymětal, Jiří - Vetýšková, Veronika - Jirásková, Kateřina - Vondrášek, Jiří
    TRPM5 Channel Binds Calcium-Binding Proteins Calmodulin and S100A1.
    Biochemistry. Roč. 61, č. 6 (2022), s. 413-423. ISSN 0006-2960
    Institutional support: RVO:61388963
    Keywords : ion channel * ryanodine receptor * N-terminus
    OECD category: Biochemistry and molecular biology
    Impact factor: 2.9, year: 2022
    Method of publishing: Limited access
    https://doi.org/10.1021/acs.biochem.1c00647
    Permanent Link: http://hdl.handle.net/11104/0331043
     
     
  6. 6.
    0551558 - ÚEM 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 july (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA ČR(CZ) GA20-12047S; GA TA ČR(CZ) TO01000078
    Institutional support: RVO:68378041
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacologyin vivo * tacrine
    OECD category: Medicinal chemistry
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0326821
     
     
  7. 7.
    0543492 - ÚEM 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, K. - Kletečková, L. - Chvojková, M. - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Hrčka Krausová, Barbora - Horák, Martin - Valeš, K. - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, apr. (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA ČR(CZ) GA20-12047S
    Institutional support: RVO:68378041
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320802
     
     
  8. 8.
    0543350 - FGÚ 2022 RIV US eng J - Journal Article
    Kaniaková, Martina - Korábečný, J. - Holubová, Kristína - Kletečková, Lenka - Chvojková, Markéta - Hakenová, K. - Prchal, L. - Novák, M. - Doležal, R. - Hepnarová, V. - Svobodová, B. - Kučera, T. - Lichnerová, Katarina - Krausová, B. - Horák, Martin - Valeš, Karel - Soukup, O.
    7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo.
    Biochemical Pharmacology. Roč. 186, Apr (2021), č. článku 114460. ISSN 0006-2952. E-ISSN 1873-2968
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : behavioral experiment * electrophysiology * glutamate receptor * mutation * ion channel * acetylcholinesterase
    OECD category: Pharmacology and pharmacy
    Impact factor: 6.100, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.bcp.2021.114460
    Permanent Link: http://hdl.handle.net/11104/0320571
     
     
  9. 9.
    0542659 - FGÚ 2022 RIV FR eng J - Journal Article
    Gorecki, L. - Misiachna, Anna - Damborský, J. - Doležal, R. - Korábečný, J. - Čejková, L. - Hakenová, K. - Chvojková, M. - Zdarová Karasová, J. - Prchal, L. - Novák, M. - Kolcheva, Marharyta - Kortus, Štěpán - Valeš, K. - Horák, Martin - Soukup, O.
    Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors.
    European Journal of Medicinal Chemistry. Roč. 219, 5 July (2021), č. článku 113434. ISSN 0223-5234. E-ISSN 1768-3254
    R&D Projects: GA MZd(CZ) EF16_025/0007444
    Institutional support: RVO:67985823
    Keywords : QSAR * acetylcholinesterase * electrophysiology * glutamate receptor * ion channel * pharmacology * in vivo * tacrine
    OECD category: Pharmacology and pharmacy
    Impact factor: 7.088, year: 2021
    Method of publishing: Open access
    https://doi.org/10.1016/j.ejmech.2021.113434
    Permanent Link: http://hdl.handle.net/11104/0320032
     
     
  10. 10.
    0542632 - FGÚ 2022 RIV NL eng J - Journal Article
    Kolcheva, Marharyta - Kortus, Š. - Hrčka Krausová, B. - Baráčková, P. - Misiachna, A. - Danačíková, Šárka - Kaniaková, M. - Hemelíková, K. - Hotovec, M. - Řeháková, K. - Horák, M.
    Specific pathogenic mutations in the M3 domain of the GluN1 subunit regulate the surface delivery and pharmacological sensitivity of NMDA receptors.
    Neuropharmacology. Roč. 189, 15 May (2021), č. článku 108528. ISSN 0028-3908. E-ISSN 1873-7064
    R&D Projects: GA ČR(CZ) GA20-12420S
    Institutional support: RVO:67985823
    Keywords : electrophysiology * glutamate receptor * hippocampal neuron * ion channel * memantine * membrane domain
    OECD category: Neurosciences (including psychophysiology
    Impact factor: 5.273, year: 2021
    Method of publishing: Limited access
    https://doi.org/10.1016/j.neuropharm.2021.108528
    Permanent Link: http://hdl.handle.net/11104/0320020
     
     

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