Search results
- 1.0586203 - ÚOCHB 2025 RIV DE eng J - Journal Article
Tóth, Luca Julianna - Krejčová, Kateřina - Dejmek, Milan - Žilecká, Eva - Klepetářová, Blanka - Poštová Slavětínská, Lenka - Bouřa, Evžen - Nencka, Radim
Novel analogues of a nonnucleoside SARS-CoV-2 RdRp inhibitor as potential antivirotics.
Beilstein Journal of Organic Chemistry. Roč. 20, May (2024), s. 1029-1036. ISSN 1860-5397. E-ISSN 1860-5397
R&D Projects: GA MŠMT(CZ) LX22NPO5103
Institutional support: RVO:61388963
Keywords : antivirotics * nonnucleotide inhibitor * RNA-dependent RNA polymerase * SARS-CoV-2
Impact factor: 2.7, year: 2022
Method of publishing: Open access
https://doi.org/10.3762/bjoc.20.91
Permanent Link: https://hdl.handle.net/11104/0353790File Download Size Commentary Version Access 10.3762bjoc.20.91.pdf 0 914.3 KB Publisher’s postprint open-access - 2.0586002 - ÚOCHB 2025 RIV US eng J - Journal Article
Spiwoková, Petra - Horn, Martin - Fanfrlík, Jindřich - Jílková, Adéla - Fajtová, Pavla - Leontovyč, Adrian - Houštecká, Radka - Bieliková, Lucia - Brynda, Jiří - Chanová, M. - Mertlíková-Kaiserová, Helena - Diaz-Caro, E. J. E. - Almaliti, J. - El Sakkary, N. - Gerwick, W. H. - Caffrey, C. R. - Mareš, Michael
Nature-Inspired Gallinamides Are Potent Antischistosomal Agents: Inhibition of the Cathepsin B1 Protease Target and Binding Mode Analysis.
ACS Infectious Diseases. (2024). ISSN 2373-8227
R&D Projects: GA MŠMT(CZ) LTAUSA19109; GA MŠMT(CZ) LUAUS23050; GA MZd(CZ) NV18-05-00345
Institutional support: RVO:61388963
Keywords : cathepsin B * cysteine protease * drug target * parasite * Schistosoma mansoni * acrylamide inhibitor
Impact factor: 5.3, year: 2022
Method of publishing: Open access
https://doi.org/10.1021/acsinfecdis.3c00589
Permanent Link: https://hdl.handle.net/11104/0353623 - 3.0584422 - BFÚ 2025 RIV GB eng J - Journal Article
Figueiredo, J. - Mergny, Jean-Louis - Cruz, C.
G-quadruplex ligands in cancer therapy: Progress, challenges, and clinical perspectives.
Life Sciences. Roč. 340, MAR 1 2024 (2024), č. článku 122481. ISSN 0024-3205. E-ISSN 1879-0631
Institutional support: RVO:68081707
Keywords : telomeric g-quadruplex * structure-based design * growth in-vitro * quindoline derivatives * cell-proliferation * pancreatic-cancer * dna structures * inhibitor
OECD category: Pharmacology and pharmacy
Impact factor: 6.1, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S0024320524000705?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0353658 - 4.0583605 - BFÚ 2024 RIV NL eng J - Journal Article
Daďová, Petra - Mikulová, Antónia - Jaroušek, Radim - Chorvátová, Michaela - Uldrijan, S. - Kubala, Lukáš
A forskolin-mediated increase in cAMP promotes T helper cell differentiation into the Th1 and Th2 subsets rather than into the Th17 subset.
International Immunopharmacology. Roč. 125, DEC 2023 (2023), č. článku 111166. ISSN 1567-5769. E-ISSN 1878-1705
Institutional support: RVO:68081707
Keywords : dependent protein-kinase * cyclic-amp * genetic architecture * pde4 inhibitor * responses * memory * naive * lymphocytes * expression * modulators
OECD category: Immunology
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S1567576923014923?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0351615 - 5.0583159 - ÚOCHB 2025 RIV US eng J - Journal Article
Kriegelstein, Michal - Nováková, Gabriela - Marek, Aleš
Synthesis of [3H]Org24598 using in-house prepared [3H]MeI.
Journal of Labelled Compounds and Radiopharmaceuticals. Roč. 67, č. 3 (2024), s. 91-103. ISSN 0362-4803. E-ISSN 1099-1344
Institutional support: RVO:61388963
Keywords : [H-3]fluoxetine * [H-3]methylation * [H-3]methyl iodide preparation * [H-3]Org24598 * [H-3]thioanisol * COware gas reactor * GlyT1 inhibitor
Impact factor: 1.8, year: 2022
Method of publishing: Limited access
https://doi.org/10.1002/jlcr.4084
Permanent Link: https://hdl.handle.net/11104/0351151 - 6.0582851 - ÚOCHB 2025 RIV CH eng J - Journal Article
Matoušková, Zuzana - Orsághová, Katarína - Srb, Pavel - Pytelková, Jana - Kukačka, Zdeněk - Buša, Michal - Hajdušek, Ondřej - Šíma, Radek - Fábry, Milan - Novák, Petr - Horn, Martin - Kopáček, Petr - Mareš, Michael
An Unusual Two-Domain Thyropin from Tick Saliva: NMR Solution Structure and Highly Selective Inhibition of Cysteine Cathepsins Modulated by Glycosaminoglycans.
International Journal of Molecular Sciences. Roč. 25, č. 4 (2024), č. článku 2240. ISSN 1661-6596
R&D Projects: GA ČR(CZ) GA21-08826S; GA ČR(CZ) GA22-27695S; GA MŠMT(CZ) EF16_019/0000759; GA ČR(CZ) GA22-30920S; GA MŠMT(CZ) LUC23037
Institutional support: RVO:61388963 ; RVO:61388971 ; RVO:60077344
Keywords : cathepsin * cysteine protease * tick * parasite * saliva * thyropin * protease inhibitor * protein structure
Impact factor: 5.6, year: 2022
Method of publishing: Open access
https://doi.org/10.3390/ijms25042240
Permanent Link: https://hdl.handle.net/11104/0350903 - 7.0582665 - ÚOCHB 2025 RIV eng J - Journal Article
Galkin, Maksym - Priss, Anastasiia - Kyriukha, Y. - Shvadchak, V.
Navigating α-Synuclein Aggregation Inhibition: Methods, Mechanisms, and Molecular Targets.
Chemical Record. Roč. 24, č. 2 (2024), č. článku e202300282. ISSN 1527-8999. E-ISSN 1528-0691
Institutional support: RVO:61388963
Keywords : amyloid * inhibitor * alpha-synuclein * Parkinson's disease * protein misfolding
Impact factor: 6.6, year: 2022
Method of publishing: Limited access
https://doi.org/10.1002/tcr.202300282
Permanent Link: https://hdl.handle.net/11104/0350744 - 8.0580702 - MBÚ 2025 RIV NL eng J - Journal Article
Kovář, Marek - Šubr, Vladimír - Běhalová, Kateřina - Studenovský, Martin - Starenko, Daniil - Kovářová, Jiřina - Procházková, Petra - Etrych, Tomáš - Kostka, Libor
Chemosensitization of tumors via simultaneous delivery of STAT3 inhibitor and doxorubicin through HPMA copolymer-based nanotherapeutics with pH-sensitive activation.
Nanomedicine: Nanotechnology, Biology and Medicine. Roč. 56, February 2024 (2024), s. 102730. ISSN 1549-9634. E-ISSN 1549-9642
R&D Projects: GA MZd(CZ) NU21-03-00273; GA MŠMT LX22NPO5102
Institutional support: RVO:61388971 ; RVO:61389013
Keywords : STAT3 inhibitor * Doxorubicin * HPMA copolymer carrier * pH-sensitive drug * release
OECD category: Pharmacology and pharmacy; Medicinal chemistry (UMCH-V)
Impact factor: 5.4, year: 2022
Method of publishing: Open access
https://www.sciencedirect.com/science/article/pii/S1549963423000813
Permanent Link: https://hdl.handle.net/11104/0349459File Download Size Commentary Version Access 0580702.pdf 1 5 MB CC BY license Publisher’s postprint open-access Kovar et al_Nanomedicine.pdf 0 5 MB Publisher’s postprint open-access - 9.0579447 - ÚOCHB 2025 RIV GB eng J - Journal Article
Misehe, Mbilo - Šála, Michal - Matoušová, Marika - Hercík, Kamil - Kocek, Hugo - Chalupská, Dominika - Chaloupecká, Ema - Hájek, Miroslav - Bouřa, Evžen - Mertlíková-Kaiserová, Helena - Nencka, Radim
Design, synthesis and evaluation of novel thieno[2,3d]pyrimidine derivatives as potent and specific RIPK2 inhibitors.
Bioorganic & Medicinal Chemistry. Roč. 97, January (2024), č. článku 129567. ISSN 0968-0896. E-ISSN 1464-3391
R&D Projects: GA MZd(CZ) NU20-05-00472; GA MŠMT(CZ) LX22NPO5103
Institutional support: RVO:61388963
Keywords : kinase inhibitor * thieno [2,3d] pyrimidine derivative * receptor-interacting protein kinase 2 * RIPK2 * NOD
Impact factor: 3.5, year: 2022
Method of publishing: Open access
https://doi.org/10.1016/j.bmcl.2023.129567
Permanent Link: https://hdl.handle.net/11104/0348249File Download Size Commentary Version Access 10.1016j.bmcl.2023.129567.pdf 0 1.6 MB Publisher’s postprint open-access - 10.0578414 - MBÚ 2024 RIV NL eng J - Journal Article
Sun, Daquan - Kotianová, Michala - Rozmoš, Martin - Hršelová, Hana - Bukovská, Petra - Jansa, Jan
Arbuscular mycorrhizal hyphae selectively suppress soil ammonia oxidizers but probably not by production of biological nitrification inhibitors.
Plant and Soil. Roč. 491, č. 1-2 (2023), s. 627-643. ISSN 0032-079X. E-ISSN 1573-5036
R&D Projects: GA ČR(CZ) GA21-07247S; GA ČR(CZ) GA23-04690S
Institutional support: RVO:61388971
Keywords : nitrogen * plant * archaea * fungi * ecosystems * diversity * community * transport * growth * pcr * Ammonia-oxidizing (AO) microorganisms * Biological nitrification inhibitor (BNI) * Microbial community profiling * Nitrogen (N) * N-15 isotopic labelling and tracing * Quantitative real-time PCR (qPCR)
OECD category: Microbiology
Impact factor: 4.9, year: 2022
Method of publishing: Limited access
https://link.springer.com/article/10.1007/s11104-023-06144-x
Permanent Link: https://hdl.handle.net/11104/0347410