Search results
- 1.0544791 - ÚOCHB 2022 RIV FR eng J - Journal Article
Šimková, Adéla - Ormsby, Tereza - Sidej, Natan - Poštová Slavětínská, Lenka - Brynda, Jiří - Beranová, Jana - Šácha, Pavel - Majer, Pavel - Konvalinka, Jan
Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with α-ketoamide warheads.
European Journal of Medicinal Chemistry. Roč. 224, Nov 15 (2021), č. článku 113717. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA ČR(CZ) GA19-10280S; GA MZd(CZ) NV15-31379A; GA MŠMT(CZ) EF16_019/0000729; GA MŠMT(CZ) LM2015064
Institutional support: RVO:61388963
Keywords : fibroblast activation protein * seprase * FAP inhibitor * serine protease inhibition * prolyl endopeptidase * α-Ketoamide inhibitor
OECD category: Medicinal chemistry
Impact factor: 7.088, year: 2021
Method of publishing: Open access
https://doi.org/10.1016/j.ejmech.2021.113717
Permanent Link: http://hdl.handle.net/11104/0321598 - 2.0544017 - ÚI 2022 RIV CH eng J - Journal Article
Balážiová, E. - Výmola, P. - Hrabal, P. - Mateu, R. - Zubal, M. - Tomáš, R. - Netuka, D. - Kramář, F. - Zemanová, Z. - Svobodová, K. - Brabec, Marek - Šedo, A. - Bušek, P.
Fibroblast Activation Protein Expressing Mesenchymal Cells Promote Glioblastoma Angiogenesis.
Cancers (Basel). Roč. 13, č. 13 (2021), č. článku 3304. E-ISSN 2072-6694
R&D Projects: GA MZd NU21-04-00100
Institutional support: RVO:67985807
Keywords : glioblastoma * angiogenesis * microenvironment * fibroblast activation protein * seprase * angiopoietin * vessel destabilisation
OECD category: Statistics and probability
Impact factor: 6.575, year: 2021
Method of publishing: Open access
http://dx.doi.org/10.3390/cancers13133304
Permanent Link: http://hdl.handle.net/11104/0321082File Download Size Commentary Version Access 0544017-aoa.pdf 1 2 MB OA CC BY 4.0 Publisher’s postprint open-access - 3.0523934 - ÚOCHB 2021 RIV NL eng J - Journal Article
Šimková, Adéla - Bušek, P. - Šedo, A. - Konvalinka, Jan
Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications.
Biochimica Et Biophysica Acta-Proteins and Proteomics. Roč. 1868, č. 7 (2020), č. článku 140409. ISSN 1570-9639. E-ISSN 1878-1454
R&D Projects: GA MZd(CZ) NV15-31379A; GA MŠMT(CZ) LM2015064; GA MŠMT(CZ) EF16_019/0000729
Institutional support: RVO:61388963
Keywords : fibroblast activation protein * FAP inhibitors * FAP substrates * cancer tissue targeting * activity-based probes
OECD category: Biochemistry and molecular biology
Impact factor: 3.036, year: 2020
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/abs/pii/S1570963920300546
Permanent Link: http://hdl.handle.net/11104/0308229 - 4.0460195 - ÚI 2017 RIV CH eng J - Journal Article
Bušek, P. - Vaníčková, Z. - Hrabal, P. - Brabec, Marek - Frič, P. - Zavoral, M. - Škrha, J. - Kmochová, K. - Laclav, M. - Bunganič, B. - Augustyns, K. - Van Der Veken, P. - Šedo, A.
Increased Tissue and Circulating Levels of Dipeptidyl Peptidase-IV Enzymatic Activity in Patients with Pancreatic Ductal Adenocarcinoma.
Pancreatology. Roč. 16, č. 5 (2016), s. 829-838. ISSN 1424-3903. E-ISSN 1424-3911
Grant - others:GA MZd(CZ) NT14254
Institutional support: RVO:67985807
Keywords : Diabetes mellitus * Fibroblast activation protein alpha * Peptide hydrolases * Plasma * Stromal cells
Subject RIV: FD - Oncology ; Hematology
Impact factor: 2.580, year: 2016
Permanent Link: http://hdl.handle.net/11104/0260315