Search results
- 1.0558879 - ÚVGZ 2023 RIV CH eng J - Journal Article
Gonec, T. - Pindjakova, D. - Vrablova, L. - Strharsky, T. - Michnova, H. - Kauerová, T. - Kollár, P. - Oravec, Michal - Jendrzejewska, I. - Čížek, A. - Jampílek, J.
Antistaphylococcal Activities and ADME-Related Properties of Chlorinated Arylcarbamoylnaphthalenylcarbamates.
Pharmaceuticals. Roč. 15, č. 6 (2022), č. článku 715. E-ISSN 1424-8247
R&D Projects: GA MŠMT(CZ) LM2018123; GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : antimicrobial activity * staphylococcus-aureus * biological-activity * resistance * derivatives * permeability * mechanisms * spectrum * design * oxides * hydroxynaphthalenes * carbamates * antistaphylococcal activity * cytotoxicity * lipophilicity * structure-activity relationships
OECD category: Pharmacology and pharmacy
Impact factor: 4.6, year: 2022
Method of publishing: Open access
https://www.mdpi.com/1424-8247/15/6/715
Permanent Link: http://hdl.handle.net/11104/0332380 - 2.0536266 - ÚVGZ 2021 RIV CH eng J - Journal Article
Kos, J. - Bak, A. - Kozik, V. - Jankech, T. - Strharsky, T. - Swietlicka, A. - Michnova, H. - Hošek, J. - Smolinski, A. - Oravec, Michal - Devinsky, F. - Hutta, M. - Jampílek, J.
Biological Activities and ADMET-Related Properties of Novel Set of Cinnamanilides dagger.
Molecules. Roč. 25, č. 18 (2020), č. článku 4121. E-ISSN 1420-3049
R&D Projects: GA MŠMT(CZ) EF16_019/0000797
Institutional support: RVO:86652079
Keywords : molecular lipophilicity * drug discovery * log-p * som-4d-qsar * prediction * hybrids * agents * pk(a) * dye * cinnamamides * synthesis * antistaphylococcal activity * MTT assay * cytotoxicity * lipophilicity * pca * ive-pls * quantitative structure-property relationships
OECD category: Demography
Impact factor: 4.412, year: 2020
Method of publishing: Open access
https://www.mdpi.com/1420-3049/25/18/4121
Permanent Link: http://hdl.handle.net/11104/0314080 - 3.0492117 - ÚVGZ 2019 RIV CH eng J - Journal Article
Pospíšilová, Š. - Kos, J. - Michnova, H. - Kapustíková, I. - Strhanský, T. - Oravec, Michal - Moricz, A. M. - Bakonyi, J. - Kauerová, T. - Kollár, P. - Čížek, A. - Jampílek, J.
Synthesis and Spectrum of Biological Activities of Novel N-arylcinnamamides.
International Journal of Molecular Sciences. Roč. 19, č. 8 (2018), č. článku E2318. E-ISSN 1422-0067
R&D Projects: GA MŠMT(CZ) LO1415; GA MŠMT(CZ) EF16_013/0001609
Institutional support: RVO:86652079
Keywords : MTT assay * PET inhibition * antifungal activity * antistaphylococcal activity * biofilm * cinnamamides * structure–activity relationship * time-kill assay * toxicity
OECD category: Biochemistry and molecular biology
Impact factor: 4.183, year: 2018
Permanent Link: http://hdl.handle.net/11104/0285679