Search results
- 1.0584812 - BTÚ 2025 RIV US eng J - Journal Article
Sychra, T. - Spalenkova, A. - Balatka, S. - Václavíková, R. - Šeborová, K. - Ehrlichová, M. - Truksa, Jaroslav - Sandoval-Acuna, Cristian - Němcová, V. - Szabo, A. - Kočí, K. - Tesarova, T. - Chen, L. - Ojima, I. - Oliverius, M. - Souček, P.
Third-generation taxanes SB-T-121605 and SB-T-121606 are effective in pancreatic ductal adenocarcinoma.
iScience. Roč. 27, č. 2 (2024), č. článku 109044. E-ISSN 2589-0042
R&D Projects: GA ČR(CZ) GA21-14082S
Institutional support: RVO:86652036
Keywords : biological evaluation * cancer * microenvironment * cytotoxicity * transport * design
OECD category: Biochemistry and molecular biology
Impact factor: 5.8, year: 2022
Method of publishing: Limited access
https://www.sciencedirect.com/science/article/pii/S2589004224002657?via%3Dihub
Permanent Link: https://hdl.handle.net/11104/0352753 - 2.0546168 - ÚSMH 2022 RIV CH eng J - Journal Article
Chocholatá, P. - Kulda, V. - Dvořáková, J. - Šupová, Monika - Žaloudková, Margit - Babuška, V.
In situ hydroxyapatite synthesis enhances biocompatibility of pva/ha hydrogels.
International Journal of Molecular Sciences. Roč. 22, č. 17 (2021), č. článku 9335. E-ISSN 1422-0067
Institutional support: RVO:67985891
Keywords : In situ synthesis * Hydrogel * Scaffold * Polyvinyl alcohol * Hyaluronic acid * Hydroxyapatite * Bone tissue engineering * Biological evaluation * Cell viability
OECD category: Polymer science
Impact factor: 6.208, year: 2021
Method of publishing: Open access
https://www.mdpi.com/1422-0067/22/17/9335
Permanent Link: http://hdl.handle.net/11104/0322896 - 3.0543720 - ÚVGZ 2022 RIV CH eng J - Journal Article
Kos, J. - Strharsky, T. - Štěpánková, Š. - Svrčková, K. - Oravec, Michal - Hošek, J. - Imramovský, A. - Jampílek, J.
Trimethoxycinnamates and Their Cholinesterase Inhibitory Activity.
Applied Sciences-Basel. Roč. 11, č. 10 (2021), č. článku 4691. E-ISSN 2076-3417
R&D Projects: GA MŠMT(CZ) EF16_019/0000797; GA MŠMT(CZ) LM2015061
Research Infrastructure: CzeCOS III - 90123
Institutional support: RVO:86652079
Keywords : biological evaluation * 3,4,5-trimethoxycinnamic acid * butyrylcholinesterase * acetylcholinesterase * derivatives * design * discovery * analogs * hybrids * trimethoxycinnamates * cholinesterase-inhibiting activity * cytotoxicity * structure-activity relationships
OECD category: Organic chemistry
Impact factor: 2.838, year: 2021
Method of publishing: Open access
https://www.mdpi.com/2076-3417/11/10/4691
Permanent Link: http://hdl.handle.net/11104/0320889 - 4.0541528 - ÚMG 2021 RIV US eng J - Journal Article
Jorda, R. - Havlíček, L. - Šturc, A. - Tušková, D. - Daumová, L. - Alam, M. - Škerlová, Jana - Nekardová, M. - Peřina, M. - Pospíšil, T. - Šiiroká, J. - Urbánek, L. - Pachl, P. - Řezáčová, Pavlína - Strnad, M. - Klener, P. - Kryštof, V.
3,5,7-Substituted Pyrazolo[4,3-d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models.
Journal of Medicinal Chemistry. Roč. 62, č. 9 (2019), s. 4606-4623. ISSN 0022-2623. E-ISSN 1520-4804
Institutional support: RVO:68378050
Keywords : biological evaluation * cell-cycle * roscovitine * potent * apoptosis * subgroups * purines * abt-199
OECD category: Biochemistry and molecular biology
Impact factor: 6.205, year: 2019
Method of publishing: Limited access
https://pubs.acs.org/doi/10.1021/acs.jmedchem.9b00189
Permanent Link: http://hdl.handle.net/11104/0319083 - 5.0524320 - BFÚ 2021 RIV GB eng J - Journal Article
Guillon, J. - Cohen, A. - Boudot, C. - Valle, A. - Milano, V. - Das, R.N. - Gudin, A. - Moreau, S. - Ronga, L. - Savrimoutou, S. - Demourgues, A. - Reviriego, E. - Rubio, S. - Ferriez, S. - Agnamey, P. - Pauc, C. - Moukha, S. - Dozolme, P. - Da Nascimento, S. - Laumaille, P. - Bouchut, A. - Azas, N. - Mergny, Jean-Louis - Mullie, C. - Sonnet, P. - Courtioux, B.
Design, synthesis, and antiprotozoal evaluation of new 2,4-bis[(substituted-aminomethyl)phenyl]quinoline, 1,3-bis[(substituted-aminomethyl)phenyl]isoquinoline and 2,4-bis[(substituted-aminomethyl)phenyl]quinazoline derivatives.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 35, č. 1 (2020), s. 432-459. ISSN 1475-6366. E-ISSN 1475-6374
R&D Projects: GA MŠMT EF15_003/0000477
Institutional support: RVO:68081707
Keywords : antimalarial activity * in-vivo * antileishmanial agents * biological evaluation
OECD category: Biochemistry and molecular biology
Impact factor: 5.051, year: 2020
Method of publishing: Open access
http://apps.webofknowledge.com/InboundService.do?customersID=Alerting&mode=FullRecord&IsProductCode=Yes&product=WOS&Init=Yes&Func=Frame&DestFail=http%3A%2F%2Fwww.webofknowledge.com&action=retrieve&SrcApp=Alerting&SrcAuth=Alerting&SID=F3aUiaBOib1sK4fXSDd&UT=WOS%3A000505407000001
Permanent Link: http://hdl.handle.net/11104/0308683 - 6.0510440 - ÚMG 2020 RIV GB eng J - Journal Article
Pavlickova, V. - Jurásek, M. - Rimpelová, S. - Záruba, K. - Sedlák, David - Šimková, M. - Kodr, D. - Staňková, E. - Fahnrich, J. - Rottnerová, Z. - Bartůněk, Petr - Lapčík, O. - Drasar, P. - Ruml, T.
Oxime-based 19-nortestosterone-pheophorbide a conjugate: bimodal controlled release concept for PDT.
Journal of Materials Chemistry B. Roč. 7, č. 36 (2019), s. 5465-5477. ISSN 2050-750X. E-ISSN 2050-7518
R&D Projects: GA MŠMT LO1220; GA MŠMT LM2015063; GA MŠMT(CZ) LO1304
Institutional support: RVO:68378050
Keywords : human breast-cancer * mediated photodynamic therapy * androgen-receptor * prostate-cancer * in-vitro * biological evaluation * pyropheophorbide-a * cellular uptake * pheophorbide * photosensitizers
OECD category: Cell biology
Impact factor: 5.344, year: 2019
Method of publishing: Limited access
https://pubs.rsc.org/en/content/articlelanding/2019/TB/C9TB01301F#!divAbstract
Permanent Link: http://hdl.handle.net/11104/0306733 - 7.0506538 - ÚFCH JH 2020 RIV NL eng J - Journal Article
Haroon, M. - Akhtar, T. - Yousuf, M.J. - Baig, Mirza Wasif - Tahir, M.N. - Rasheed, L.
Synthesis, spectroscopic characterization and crystallographic behavior of ethyl 2-(4-methyl-(2-benzylidenehydraziny1))thiazole-4-carboxylate: Experimental and theoretical (DFT) studies.
Journal of Molecular Structure. Roč. 1167, SEP 2018 (2018), s. 154-160. ISSN 0022-2860. E-ISSN 1872-8014
Institutional support: RVO:61388955
Keywords : density-functional-theory * hartree-fock * mutagenic tautomerization * biological evaluation * dna
OECD category: Physical chemistry
Impact factor: 2.120, year: 2018
Method of publishing: Limited access
Permanent Link: http://hdl.handle.net/11104/0297783File Download Size Commentary Version Access 0506538.pdf 5 2 MB Publisher’s postprint require - 8.0505109 - ÚEB 2020 RIV US eng J - Journal Article
Jorda, Radek - Havlíček, Libor - Šturc, Antonín - Tušková, D. - Daumová, L. - Alam, M. - Škerlová, Jana - Nekardová, Michaela - Peřina, Miroslav - Pospíšil, Tomáš - Široká, Jitka - Urbánek, Lubor - Pachl, Petr - Řezáčová, Pavlína - Strnad, Miroslav - Klener, P. - Kryštof, Vladimír
3,5,7-Substituted Pyrazolo[4,3- d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models.
Journal of Medicinal Chemistry. Roč. 62, č. 9 (2019), s. 4606-4623. ISSN 0022-2623. E-ISSN 1520-4804
R&D Projects: GA ČR GA17-14007S; GA ČR(CZ) GBP208/12/G016
Institutional support: RVO:61389030 ; RVO:61388963
Keywords : BIOLOGICAL EVALUATION * CELL-CYCLE * ROSCOVITINE
OECD category: Hematology; Medicinal chemistry (UOCHB-X)
Impact factor: 6.205, year: 2019
Method of publishing: Limited access
http://doi.org/10.1021/acs.jmedchem.9b00189
Permanent Link: http://hdl.handle.net/11104/0296627File Download Size Commentary Version Access 2019_Jorda_JOURNAL OF MEDICINAL CHEMISTRY_4606.pdf 4 4.5 MB Other require - 9.0495765 - ÚEB 2019 RIV CH eng J - Journal Article
Lasák, J. - Motyka, K. - Kryštof, Vladimír - Stýskala, J.
Synthesis, Bacteriostatic and Anticancer Activity of Novel Phenanthridines Structurally Similar to Benzo[c] phenanthridine Alkaloids.
Molecules. Roč. 23, č. 9 (2018), č. článku 2155. E-ISSN 1420-3049
R&D Projects: GA MŠMT(CZ) LO1304
Institutional support: RVO:61389030
Keywords : topoisomerase-ii inhibitor * biaryl coupling reaction * biological evaluation * chelerythrine * sanguinarine * nk109 * derivatives * analogs * quaternary * arylation * phenanthridines * benzo[c]phenanthridines * radical cyclization * antiproliferative * antibacterial activity
OECD category: Organic chemistry
Impact factor: 3.060, year: 2018
Permanent Link: http://hdl.handle.net/11104/0288686File Download Size Commentary Version Access 2018_Lasak_MOLECULES_2155.pdf 2 1.5 MB Other open-access - 10.0481497 - ÚEB 2018 RIV JP eng J - Journal Article
Cavallaro, V. - Řezníčková, Eva - Jorda, Radek - Alza, N.P. - Murray, A.P. - Kryštof, Vladimír
Semisynthetic Esters of 17-Hydroxycativic Acid with in Vitro Cytotoxic Activity against Leukemia Cell Lines.
Biological & Pharmaceutical Bulletin. Roč. 40, č. 11 (2017), s. 1923-1928. ISSN 0918-6158
R&D Projects: GA MŠMT(CZ) LO1204
Institutional support: RVO:61389030
Keywords : biological evaluation * derivatives * andrographolide * apoptosis * cancer * agents * diterpenes * inhibition * activation * chemistry * diterpenoid * 17-hydroxycativic acid * cytotoxic activity * human cancer cell * apoptosis
OECD category: Hematology
Impact factor: 1.694, year: 2017
Permanent Link: http://hdl.handle.net/11104/0277043File Download Size Commentary Version Access 2017_Cavallaro_BIOLOGICAL & PHARMACEUTICAL BULLETIN_1923.pdf 2 957.7 KB Other open-access