0535283 - ÚEB 2021 RIV FR eng J - Journal Article
Jorda, Radek - Krajčovičová, S. - Králová, P. - Soural, M. - Kryštof, Vladimír
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome.
European Journal of Medicinal Chemistry. Roč. 204, OCT 15 (2020), č. článku 112636. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:61389030
Keywords : Bruton's tyrosine kinase * Protein kinase * Scaffold hopping * Selectivity * Spleen tyrosine kinase
OECD category: Hematology
Impact factor: 6.514, year: 2020
Method of publishing: Open access
http://doi.org/10.1016/j.ejmech.2020.112636
Permanent Link: http://hdl.handle.net/11104/0313353
Jorda, Radek - Krajčovičová, S. - Králová, P. - Soural, M. - Kryštof, Vladimír
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome.
European Journal of Medicinal Chemistry. Roč. 204, OCT 15 (2020), č. článku 112636. ISSN 0223-5234. E-ISSN 1768-3254
Institutional support: RVO:61389030
Keywords : Bruton's tyrosine kinase * Protein kinase * Scaffold hopping * Selectivity * Spleen tyrosine kinase
OECD category: Hematology
Impact factor: 6.514, year: 2020
Method of publishing: Open access
http://doi.org/10.1016/j.ejmech.2020.112636
Permanent Link: http://hdl.handle.net/11104/0313353