0543824 - ÚMG 2022 RIV GB eng J - Journal Article
Oleksak, P. - Psotka, M. - Vančurová, Markéta - Sapega, Olena - Bieblová, Jana - Reiniš, Milan - Ryšánek, David - Mikyšková, Romana - Chalupová, K. - Malinak, D. - Svobodová, J. - Andrýs, R. - Řehulková, H. - Skopek, V. - Ngoc Lam, P. - Bártek, Jiří - Hodný, Zdeněk - Musílek, K.
Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 36, č. 1 (2021), s. 410-424. ISSN 1475-6366. E-ISSN 1475-6374
R&D Projects: GA ČR(CZ) GA18-14259S
Institutional support: RVO:68378050
Keywords : STAT3 signalling pathway * cancer * SH2 domain * inhibitor * structure-activity relationship
OECD category: Biochemistry and molecular biology
Impact factor: 5.756, year: 2021
Method of publishing: Open access
https://www.tandfonline.com/doi/full/10.1080/14756366.2020.1871336
Permanent Link: http://hdl.handle.net/11104/0320942
Oleksak, P. - Psotka, M. - Vančurová, Markéta - Sapega, Olena - Bieblová, Jana - Reiniš, Milan - Ryšánek, David - Mikyšková, Romana - Chalupová, K. - Malinak, D. - Svobodová, J. - Andrýs, R. - Řehulková, H. - Skopek, V. - Ngoc Lam, P. - Bártek, Jiří - Hodný, Zdeněk - Musílek, K.
Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition.
Journal of Enzyme Inhibition and Medicinal Chemistry. Roč. 36, č. 1 (2021), s. 410-424. ISSN 1475-6366. E-ISSN 1475-6374
R&D Projects: GA ČR(CZ) GA18-14259S
Institutional support: RVO:68378050
Keywords : STAT3 signalling pathway * cancer * SH2 domain * inhibitor * structure-activity relationship
OECD category: Biochemistry and molecular biology
Impact factor: 5.756, year: 2021
Method of publishing: Open access
https://www.tandfonline.com/doi/full/10.1080/14756366.2020.1871336
Permanent Link: http://hdl.handle.net/11104/0320942