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Pregnane-based steroids are novel positive NMDA receptor modulators that may compensate for the effect of loss-of-function disease-associated GRIN mutations

  1. 1.
    SYSNO0558978
    TitlePregnane-based steroids are novel positive NMDA receptor modulators that may compensate for the effect of loss-of-function disease-associated GRIN mutations
    Author(s) Kysilov, Bohdan (FGU-C) ORCID, SAI
    Hrčka Krausová, Barbora (FGU-C) ORCID, RID
    Vyklický, Vojtěch (FGU-C) RID, ORCID, SAI
    Smejkalová, Tereza (FGU-C) RID, ORCID
    Kořínek, Miloslav (FGU-C) RID, ORCID
    Horák, Martin (FGU-C) RID, ORCID
    Chodounská, Hana (UOCHB-X) [370/37] RID, ORCID
    Kudová, Eva (UOCHB-X) [370/37] RID, ORCID
    Černý, Jiří (FGU-C) RID, ORCID
    Vyklický ml., Ladislav (FGU-C) RID, ORCID, SAI
    Corespondence/seniorVyklický ml., Ladislav - Korespondující autor
    Source Title British Journal of Pharmacology. Roč. 179, č. 15 (2022), s. 3970-3990. - : Wiley
    Document TypeČlánek v odborném periodiku
    Grant GA20-17945S GA ČR - Czech Science Foundation (CSF), CZ - Czech Republic
    EF16_025/0007444 GA MZd - Ministry of Health (MZ), CZ - Czech Republic
    TN01000013 GA TA ČR - Technology Agency of the Czech Republic (TA ČR), CZ - Czech Republic
    Institutional supportFGU-C - RVO:67985823 ; UOCHB-X - RVO:61388963
    Languageeng
    CountryGB
    Keywords GRIN channelopathy * NMDA receptor * positive allosteric modulator * steroids * transmembrane domain
    Cooperating institutions Univerzita Karlova v Praze, 3. lékařská fakulta (Czech Republic)
    URLhttps://doi.org/10.1111/bph.15841
    Permanent Linkhttps://hdl.handle.net/11104/0332640
     
Number of the records: 1  

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