Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors

Baltus, C.B., Jorda, R., Marot, C., Berka, K., Bazgier, V., Kryštof, V., Prie, G., Viaud-Massuard, M.C. Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors. European Journal of Medicinal Chemistry. 2016, 108(JAN 27), 701-719. ISSN 0223-5234. E-ISSN 1768-3254. Available: doi: 10.1016/j.ejmech.2015.12.023