Number of the records: 1
Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with α-ketoamide warheads
- 1.
SYSNO 0544791 Title Structure-activity relationship and biochemical evaluation of novel fibroblast activation protein and prolyl endopeptidase inhibitors with α-ketoamide warheads Author(s) Šimková, Adéla (UOCHB-X) [220/22] ORCID, RID
Ormsby, Tereza (UOCHB-X) [220/22] ORCID, RID
Sidej, Natan (UOCHB-X) [220/22] ORCID
Poštová Slavětínská, Lenka (UOCHB-X) [910/91] RID
Brynda, Jiří (UOCHB-X) [930/93] RID, ORCID
Beranová, Jana (UOCHB-X) [220/22] ORCID
Šácha, Pavel (UOCHB-X) [220/22] RID, ORCID
Majer, Pavel (UOCHB-X) [390/39]
Konvalinka, Jan (UOCHB-X) [220/22] RID, ORCIDCorespondence/senior Konvalinka, Jan - Korespondující autor Source Title European Journal of Medicinal Chemistry. Roč. 224, Nov 15 (2021). - : Elsevier Article number 113717 Document Type Článek v odborném periodiku Grant GA19-10280S GA ČR - Czech Science Foundation (CSF), CZ - Czech Republic NV15-31379A GA MZd - Ministry of Health (MZ), CZ - Czech Republic EF16_019/0000729 GA MŠMT - Ministry of Education, Youth and Sports (MEYS), CZ - Czech Republic LM2015064 GA MŠMT - Ministry of Education, Youth and Sports (MEYS), CZ - Czech Republic Institutional support UOCHB-X - RVO:61388963 Language eng Country FR Keywords fibroblast activation protein * seprase * FAP inhibitor * serine protease inhibition * prolyl endopeptidase * α-Ketoamide inhibitor Cooperating institutions Univerzita Karlova (Czech Republic) URL https://doi.org/10.1016/j.ejmech.2021.113717 Permanent Link http://hdl.handle.net/11104/0321598
Number of the records: 1