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Lipases as Tools in the Synthesis of Prodrugs from Racemic 9-(2,3-Dihydroxypropyl)adenine

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    SYSNO ASEP0384593
    Document TypeJ - Journal Article
    R&D Document TypeJournal Article
    Subsidiary JČlánek ve WOS
    TitleLipases as Tools in the Synthesis of Prodrugs from Racemic 9-(2,3-Dihydroxypropyl)adenine
    Author(s) Brabcová, Jana (UOCHB-X) RID
    Blažek, Jiří (UOCHB-X)
    Janská, Lucie (UOCHB-X)
    Krečmerová, Marcela (UOCHB-X) RID, ORCID
    Zarevúcka, Marie (UOCHB-X) RID
    Number of authors5
    Source TitleMolecules. - : MDPI - ISSN 1420-3049
    Roč. 17, č. 12 (2012), s. 13813-13824
    Number of pages12 s.
    Languageeng - English
    CountryCH - Switzerland
    Keywordslipase ; transesterification ; prodrug ; immobilization of enzymes
    Subject RIVCC - Organic Chemistry
    Institutional supportUOCHB-X - RVO:61388963
    UT WOS000312608200009
    DOI https://doi.org/10.3390/molecules171213813
    AnnotationLipases from Geotrichum candidum 4013 (extracellular lipase and cell-bound lipase) were immobilized by adsorption on chitosan beads. The enzyme preparations were tested in the synthesis of ester prodrugs from racemic 9-(2,3-dihydroxypropyl)adenine in dimethylformamide with different vinyl esters (acetate, butyrate, decanoate, laurate, palmitate). The transesterification activities of these immobilized enzymes were compared with commercially available lipases (lipase from hog pancreas, Aspergillus niger, Candida antarctica, Pseudomonas fluorescens).
    WorkplaceInstitute of Organic Chemistry and Biochemistry
    Contactasep@uochb.cas.cz ; Kateřina Šperková, Tel.: 232 002 584 ; Jana Procházková, Tel.: 220 183 418
    Year of Publishing2013
Number of the records: 1  

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