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Cellular and behavioural effects of a new steroidal inhibitor of the N-methyl-d-aspartate receptor 3α5β-pregnanolone glutamate
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SYSNO ASEP 0364480 Document Type J - Journal Article R&D Document Type Journal Article Subsidiary J Článek ve WOS Title Cellular and behavioural effects of a new steroidal inhibitor of the N-methyl-d-aspartate receptor 3α5β-pregnanolone glutamate Author(s) Rambousek, Lukáš (FGU-C) RID, ORCID
Bubeníková-Valešová, V. (CZ)
Kačer, P. (CZ)
Syslová, K. (CZ)
Kenney, Jana (FGU-C)
Holubová, Kristína (FGU-C) ORCID, SAI, RID
Najmanová, V. (CZ)
Zach, P. (CZ)
Svoboda, Jan (FGU-C) RID, ORCID
Stuchlík, Aleš (FGU-C) RID, ORCID
Chodounská, Hana (UOCHB-X) RID, ORCID
Kapras, Vojtěch (UOCHB-X)
Adamusová, Eva (FGU-C)
Borovská, Jiřina (FGU-C)
Vyklický ml., Ladislav (FGU-C) RID, ORCID, SAI
Valeš, Karel (FGU-C) RID, ORCID, SAISource Title Neuropharmacology. - : Elsevier - ISSN 0028-3908
Roč. 61, 1-2 (2011), s. 61-68Number of pages 8 s. Language eng - English Country NL - Netherlands Keywords neuroactive steroid ; NMDA ; neuroprotectivity Subject RIV FH - Neurology R&D Projects NS10365 GA MZd - Ministry of Health (MZ) NR9180 GA MZd - Ministry of Health (MZ) GA309/07/0271 GA ČR - Czech Science Foundation (CSF) GA203/08/1498 GA ČR - Czech Science Foundation (CSF) GA309/09/0286 GA ČR - Czech Science Foundation (CSF) 1M0517 GA MŠMT - Ministry of Education, Youth and Sports (MEYS) LC554 GA MŠMT - Ministry of Education, Youth and Sports (MEYS) CEZ AV0Z50110509 - FGU-C (2005-2011) AV0Z40550506 - UOCHB-X (2005-2011) UT WOS 000292408200007 DOI 10.1016/j.neuropharm.2011.02.018 Annotation The results show that 3alfa5betaPregnanolone glutamate, use-dependent NMDA antagonist, is able to cross the blood brain barrier, does not induce psychotomimetic symptoms (such as hyperlocomotion and sensorimotor gating deficit) and reduced an excitotoxic damage of brain tissue and subsequent behavioural impairment in rats Workplace Institute of Physiology Contact Lucie Trajhanová, lucie.trajhanova@fgu.cas.cz, Tel.: 241 062 400 Year of Publishing 2012
Number of the records: 1