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Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors
- 1.0330291 - FGÚ 2010 RIV GB eng J - Journal Article
Mordvintsev, D.Y. - Polyak, Y.L. - Rodionov, D.I. - Jakubík, Jan - Doležal, Vladimír - Karlsson, E. - Tsetlin, V.I. - Utkin, Y.N.
Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors.
[Slabý toxin WTX z kobry monoklové se váže na receptory pro acetylcholin nikotinového i muskarinového typu.]
FEBS Journal. Roč. 276, č. 18 (2009), s. 5065-5075. ISSN 1742-464X. E-ISSN 1742-4658
R&D Projects: GA MŠMT(CZ) LC554; GA AV ČR(CZ) IAA500110703
Institutional research plan: CEZ:AV0Z50110509
Keywords : acetylcholine receptors * allosteric interaction * toxins
Subject RIV: ED - Physiology
Impact factor: 3.042, year: 2009
Data demonstrate an orthosteric interaction of WTX toxin from Naja kaouthia with nicotinic acetylcholine receptors and an allosteric interaction with muscarinic acetylcholine receptors in micromolar range
Data ukazují ortosterickou vazbu toxinu WTX z kobry monoklové na receptory pro acetylcholin nikotinového typu a alosterickou vazbu na receproty muskarinového typu v mikromolárních koncentracích
Permanent Link: http://hdl.handle.net/11104/0176115
Number of the records: 1