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Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-L-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery
- 1.NOVOTNÁ, Kateřina, TENORA, Lukáš, PRCHALOVÁ, E., PAULE, J., ALT, J., VEERAVALLI, V., LAM, J., WU, Y., ŠNAJDR, Ivan, GORI, S., METTU, V. S., TSUKAMOTO, T., MAJER, Pavel, SLUSHER, B. S., RAIS, R. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-L-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry. 2023, 66(22), 15493-15510. ISSN 0022-2623. E-ISSN 1520-4804. Available: doi: 10.1021/acs.jmedchem.3c01681.
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