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Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors

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    0330291 - FGÚ 2010 RIV GB eng J - Journal Article
    Mordvintsev, D.Y. - Polyak, Y.L. - Rodionov, D.I. - Jakubík, Jan - Doležal, Vladimír - Karlsson, E. - Tsetlin, V.I. - Utkin, Y.N.
    Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors.
    [Slabý toxin WTX z kobry monoklové se váže na receptory pro acetylcholin nikotinového i muskarinového typu.]
    FEBS Journal. Roč. 276, č. 18 (2009), s. 5065-5075. ISSN 1742-464X. E-ISSN 1742-4658
    R&D Projects: GA MŠMT(CZ) LC554; GA AV ČR(CZ) IAA500110703
    Institutional research plan: CEZ:AV0Z50110509
    Keywords : acetylcholine receptors * allosteric interaction * toxins
    Subject RIV: ED - Physiology
    Impact factor: 3.042, year: 2009

    Data demonstrate an orthosteric interaction of WTX toxin from Naja kaouthia with nicotinic acetylcholine receptors and an allosteric interaction with muscarinic acetylcholine receptors in micromolar range

    Data ukazují ortosterickou vazbu toxinu WTX z kobry monoklové na receptory pro acetylcholin nikotinového typu a alosterickou vazbu na receproty muskarinového typu v mikromolárních koncentracích
    Permanent Link: http://hdl.handle.net/11104/0176115

     
     
Number of the records: 1  

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